DK128352B - Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner. - Google Patents

Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner.

Info

Publication number
DK128352B
DK128352B DK569770AA DK569770A DK128352B DK 128352 B DK128352 B DK 128352B DK 569770A A DK569770A A DK 569770AA DK 569770 A DK569770 A DK 569770A DK 128352 B DK128352 B DK 128352B
Authority
DK
Denmark
Prior art keywords
oxazolidinoxazines
hydroxypregna
dione
diene
fluoro
Prior art date
Application number
DK569770AA
Other languages
English (en)
Inventor
G Nathansohn
G Winters
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of DK128352B publication Critical patent/DK128352B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036Nitrogen-containing hetero ring
    • C07J71/0057Nitrogen and oxygen
    • C07J71/0068Nitrogen and oxygen at position 16(17)
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011Unsubstituted amino radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
DK569770AA 1968-05-03 1970-11-10 Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner. DK128352B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1602968 1968-05-03

Publications (1)

Publication Number Publication Date
DK128352B true DK128352B (da) 1974-04-16

Family

ID=11148457

Family Applications (2)

Application Number Title Priority Date Filing Date
DK224769AA DK124680B (da) 1968-05-03 1969-04-24 Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken.
DK569770AA DK128352B (da) 1968-05-03 1970-11-10 Analogifremgangsmåde til fremstilling af 9α-fluor-11β-hydroxypregna-1,4-dien-3,20-dion-[17α,16α-d]-oxazolidinoxaziner.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK224769AA DK124680B (da) 1968-05-03 1969-04-24 Fremgangsmåde til fremstilling af 2'-substituerede steroid-[16α, 17α-d]-oxazoliner af pregnanrækken.

Country Status (16)

Country Link
US (1) US3631033A (da)
AT (2) AT291450B (da)
BE (1) BE731718A (da)
BR (1) BR6908511D0 (da)
CH (1) CH511823A (da)
DE (1) DE1921778A1 (da)
DK (2) DK124680B (da)
ES (2) ES366738A1 (da)
FI (3) FI46374C (da)
FR (1) FR2007756B1 (da)
GB (1) GB1254487A (da)
IL (1) IL31997A (da)
LU (1) LU58451A1 (da)
NL (2) NL6906149A (da)
NO (1) NO128608B (da)
SE (4) SE373578B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7107998A (da) * 1970-07-09 1972-01-11
IT1134455B (it) * 1980-11-26 1986-08-13 Lepetit Spa Procedimento per la preparazione di derivati 16alfa-idrossi-17alfa-aminopregnanici
US20030083231A1 (en) * 1998-11-24 2003-05-01 Ahlem Clarence N. Blood cell deficiency treatment method
US20050101581A1 (en) * 2002-08-28 2005-05-12 Reading Christopher L. Therapeutic treatment methods 2
JP2006506445A (ja) * 2002-08-28 2006-02-23 ホリス − イーデン ファーマスーティカルズ、 インコーポレイテッド 治療処置の方法
KR101451486B1 (ko) * 2009-09-11 2014-10-22 키에시 파르마슈티시 엣스. 피. 에이. N-치환된 이속사졸리딘 링과 함께 16, 17 위치 내에 응축된 항염증제로서의 프레그난 유도체
TWI658047B (zh) 2011-03-15 2019-05-01 吉斯藥品公司 異唑啶衍生物
CA2829982A1 (en) 2011-03-15 2012-09-20 Chiesi Farmaceutici S.P.A. Isoxazolidine derivatives
US9155747B2 (en) * 2012-09-13 2015-10-13 Chiesi Farmaceutici S.P.A. Isoxazolidine derivatives

Also Published As

Publication number Publication date
SE373131B (da) 1975-01-27
FR2007756A1 (da) 1970-01-09
DK124680B (da) 1972-11-13
IL31997A0 (en) 1969-06-25
GB1254487A (en) 1971-11-24
FI46376B (da) 1972-11-30
NO128608B (da) 1973-12-17
NL6906149A (da) 1969-11-05
CH511823A (fr) 1971-08-31
FI46377B (da) 1972-11-30
IL31997A (en) 1974-03-14
FR2007756B1 (da) 1975-10-10
DE1921778A1 (de) 1969-11-20
FI46377C (fi) 1973-03-12
ES371991A1 (es) 1971-12-01
SE373578B (sv) 1975-02-10
DE1965963B2 (de) 1973-02-08
AT300218B (de) 1972-07-25
BE731718A (da) 1969-10-01
FI46374B (da) 1972-11-30
AT291450B (de) 1971-07-12
BR6908511D0 (pt) 1973-02-08
SE363098B (da) 1974-01-07
LU58451A1 (da) 1969-07-21
DE1965963A1 (de) 1970-12-23
SE378250B (da) 1975-08-25
ES366738A1 (es) 1971-03-16
FI46374C (fi) 1973-03-12
FI46376C (fi) 1973-03-12
US3631033A (en) 1971-12-28
NL7709675A (nl) 1977-12-30

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