DK122275B - Fremgangsmåde til fremstilling af 17α-ætynyl-17β-hydroksysteroider af androstan- eller østranrækken. - Google Patents

Fremgangsmåde til fremstilling af 17α-ætynyl-17β-hydroksysteroider af androstan- eller østranrækken.

Info

Publication number
DK122275B
DK122275B DK187367AA DK187367A DK122275B DK 122275 B DK122275 B DK 122275B DK 187367A A DK187367A A DK 187367AA DK 187367 A DK187367 A DK 187367A DK 122275 B DK122275 B DK 122275B
Authority
DK
Denmark
Prior art keywords
hydroxysteroids
androstane
ethynyl
preparation
oestrane series
Prior art date
Application number
DK187367AA
Other languages
English (en)
Inventor
R Ginsig
Original Assignee
Syntex Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Corp filed Critical Syntex Corp
Publication of DK122275B publication Critical patent/DK122275B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/36Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal
    • C07C29/38Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones
    • C07C29/42Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring increasing the number of carbon atoms by reactions with formation of hydroxy groups, which may occur via intermediates being derivatives of hydroxy, e.g. O-metal by reaction with aldehydes or ketones with compounds containing triple carbon-to-carbon bonds, e.g. with metal-alkynes
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/40Ortho- or ortho- and peri-condensed systems containing four condensed rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Steroid Compounds (AREA)
DK187367AA 1966-04-07 1967-03-31 Fremgangsmåde til fremstilling af 17α-ætynyl-17β-hydroksysteroider af androstan- eller østranrækken. DK122275B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54081566A 1966-04-07 1966-04-07

Publications (1)

Publication Number Publication Date
DK122275B true DK122275B (da) 1972-02-14

Family

ID=24157045

Family Applications (1)

Application Number Title Priority Date Filing Date
DK187367AA DK122275B (da) 1966-04-07 1967-03-31 Fremgangsmåde til fremstilling af 17α-ætynyl-17β-hydroksysteroider af androstan- eller østranrækken.

Country Status (7)

Country Link
US (1) US3470217A (da)
CH (1) CH490358A (da)
DE (1) DE1618868C3 (da)
DK (1) DK122275B (da)
GB (1) GB1176229A (da)
NL (1) NL6704744A (da)
SE (1) SE337588B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4614621A (en) * 1984-04-20 1986-09-30 The Upjohn Company Ethynylation of 16-methylene-17-keto steroids
US4618456A (en) * 1984-03-20 1986-10-21 The Upjohn Company Ethynylation of 16-methyl-17-keto steroids
ES2576231T3 (es) 2011-12-23 2016-07-06 Crystal Pharma S.A.U Proceso para alquinilar 17-cetoesteroides 16-sustituidos

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2806030A (en) * 1954-03-20 1957-09-10 Syntex Sa Cyclopentanophenanthrene derivatives and process for the preparation thereof
US2888471A (en) * 1955-03-25 1959-05-26 Syntex Sa Process for preparing 17alpha-ethinyl-delta1, 4-androstadiene-17 beta-ol-3-one
NL123455C (da) * 1964-05-13

Also Published As

Publication number Publication date
DE1618868A1 (de) 1972-07-06
SE337588B (da) 1971-08-16
DE1618868C3 (de) 1973-10-11
CH490358A (de) 1970-05-15
GB1176229A (en) 1970-01-01
US3470217A (en) 1969-09-30
NL6704744A (da) 1967-10-09
DE1618868B2 (de) 1973-03-08

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