DK127556B - Analogifremgangsmåde til fremstilling af quinazolinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af quinazolinderivater eller syreadditionssalte deraf.

Info

Publication number
DK127556B
DK127556B DK397770AA DK397770A DK127556B DK 127556 B DK127556 B DK 127556B DK 397770A A DK397770A A DK 397770AA DK 397770 A DK397770 A DK 397770A DK 127556 B DK127556 B DK 127556B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
quinazoline derivatives
analogous process
Prior art date
Application number
DK397770AA
Other languages
Danish (da)
English (en)
Inventor
S Inaba
M Yamamoto
K Ishizumi
K Mori
H Yamamoto
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP653170A external-priority patent/JPS5138714B1/ja
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of DK127556B publication Critical patent/DK127556B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • C07D239/82Oxygen atoms with an aryl radical attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK397770AA 1969-08-02 1970-07-31 Analogifremgangsmåde til fremstilling af quinazolinderivater eller syreadditionssalte deraf. DK127556B (da)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
JP6122269 1969-08-02
JP6187269 1969-08-04
JP7045369 1969-09-04
JP9883669 1969-12-08
JP9919669 1969-12-09
JP10281069 1969-12-19
JP653170A JPS5138714B1 (de) 1970-01-23 1970-01-23
JP662870 1970-01-24
JP1406970 1970-02-17

Publications (1)

Publication Number Publication Date
DK127556B true DK127556B (da) 1973-11-26

Family

ID=27576527

Family Applications (1)

Application Number Title Priority Date Filing Date
DK397770AA DK127556B (da) 1969-08-02 1970-07-31 Analogifremgangsmåde til fremstilling af quinazolinderivater eller syreadditionssalte deraf.

Country Status (12)

Country Link
US (1) US3712892A (de)
CH (3) CH553190A (de)
DE (1) DE2037693C3 (de)
DK (1) DK127556B (de)
FI (1) FI54301C (de)
FR (1) FR2060075B1 (de)
GB (1) GB1313789A (de)
IL (1) IL35035A (de)
NL (1) NL151704B (de)
NO (1) NO128277B (de)
PL (1) PL81273B1 (de)
YU (1) YU3277A (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3925359A (en) * 1967-03-30 1975-12-09 Hoffmann La Roche Novel 2{8 2-(1,3-diazacycloalk-2-enyl){9 benzophenone derivatives and novel 1,3-diazacycloalkenyl{8 2,1-1{9 isoindole derivatives
US3929766A (en) * 1967-03-30 1975-12-30 Hoffmann La Roche Novel 2{8 2-(1,3-diazacycloalk-2-enyl){9 benzophenone derivatives and novel 1,3-diazacycloalkenyl{8 2,1-A{9 isoindole derivatives
DE2118315C3 (de) * 1970-04-20 1975-04-03 Sumitomo Chemical Co., Ltd., Osaka (Japan) 2-(1H)-Chinazolinonderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DK129348B (da) * 1970-07-13 1974-09-30 Sumitomo Chemical Co Analogifremgangsmåde til fremstilling af 1-substituerede 3,4-dihydro-2(1H)-quinazolinonderivater.
DE2050640A1 (de) * 1970-10-15 1972-04-20 Cassella Farbwerke Mainkur Ag, 6000 Frankfurt Basisch substituierte Derivate des (lH,3H)-Chinazolin-2-thion-4-ons
DE2162327C3 (de) * 1970-12-23 1975-09-18 Sumitomo Chemical Co., Ltd., Osaka (Japan) Verfahren zur Herstellung von 3,4-Oihydro-2(1 H)-chinazolinonen
DK135044B (da) * 1971-05-06 1977-02-28 Sandoz Ag Analogifremgangsmåde til fremstilling af 4-phenyl- eller 4-(2'-thienyl)-6,7-methylendioxy-2(1H)-quinazolinoner eller -2(1H)-quinazolinthioner.
US4202895A (en) * 1971-06-04 1980-05-13 Sumitomo Chemical Company, Limited 1-Polyhaloalkyl-2(1H)-quinazolinone derivatives
BE795519A (fr) * 1972-02-18 1973-06-18 Sumitomo Chemical Co Procede de preparation d'un agent uricosurique
JPS5426556B2 (de) * 1972-03-24 1979-09-04
JPS5427356B2 (de) * 1972-03-31 1979-09-10
DE2225218C2 (de) * 1972-05-24 1983-01-13 Morishita Pharmaceutical Co., Ltd., Osaka 2-Alkyl-4-äthoxy-5-morpholino-3(2H)-pyridazinone und Verfahren zu deren Herstellung
JPS5418269B2 (de) * 1972-07-20 1979-07-06
JPS5537554B2 (de) * 1972-07-24 1980-09-29
JPS555506B2 (de) * 1972-09-07 1980-02-07
US4067868A (en) * 1973-04-17 1978-01-10 Sumitomo Chemical Company, Limited Production of quinazolinone compounds
US3927011A (en) * 1973-05-10 1975-12-16 Yoshitomi Pharmaceutical 2-Aminoalkyl-1-(pyridylcarbonylphenyl)imidazole compounds
JPS5724789B2 (de) * 1973-08-14 1982-05-26
JPS5046680A (de) * 1973-08-20 1975-04-25
GB1494340A (en) * 1974-12-03 1977-12-07 Wyeth John & Brother Ltd Process for preparation of substituted n-phenylcarbamate esters
JPS521036A (en) 1975-06-23 1977-01-06 Sumitomo Chem Co Ltd Antiphlogistic with extremely low reaction to digestive canals
US4247554A (en) * 1977-05-11 1981-01-27 Sumitomo Chemical Company, Limited Method for the prevention of gastro-intestinal ulcer caused by a non-steroidal anti-inflammatory agent
AR038658A1 (es) * 2001-06-15 2005-01-26 Novartis Ag Derivados de 4-aril-2(1h) quinazolinona y 4-aril-quinazolina 2-sustituidas, un proceso para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la preparacion de un medicamento
GB0230015D0 (en) 2002-12-23 2003-01-29 Novartis Ag Organic compounds
WO2005042501A1 (en) * 2003-11-03 2005-05-12 Warner-Lambert Company Llc Novel norepinephrine reuptake inhibitors for the treatment of central nervous system disorders
US20070111906A1 (en) * 2005-11-12 2007-05-17 Milner Jeffrey L Relatively low viscosity transmission fluids
US7682491B2 (en) * 2007-03-26 2010-03-23 Nalco Company Antifoulant for hydrocarbon processing equipment

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RO56665A (de) * 1968-07-01 1974-06-01

Also Published As

Publication number Publication date
US3712892A (en) 1973-01-23
FI54301C (fi) 1978-11-10
FI54301B (fi) 1978-07-31
FR2060075A1 (de) 1971-06-11
IL35035A0 (en) 1970-09-17
PL81273B1 (en) 1975-08-30
DE2037693B2 (de) 1974-05-22
FR2060075B1 (de) 1974-08-30
GB1313789A (en) 1973-04-18
NL151704B (nl) 1976-12-15
CH553791A (de) 1974-09-13
CH553190A (de) 1974-08-30
NL7011359A (de) 1971-02-04
DE2037693C3 (de) 1975-01-16
IL35035A (en) 1973-01-30
DE2037693A1 (de) 1971-02-25
CH554877A (de) 1974-10-15
YU3277A (en) 1982-06-30
NO128277B (de) 1973-10-22

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Legal Events

Date Code Title Description
PBP Patent lapsed