DK1214292T3 - Tyrosinderivater - Google Patents

Tyrosinderivater

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Publication number
DK1214292T3
DK1214292T3 DK00965417T DK00965417T DK1214292T3 DK 1214292 T3 DK1214292 T3 DK 1214292T3 DK 00965417 T DK00965417 T DK 00965417T DK 00965417 T DK00965417 T DK 00965417T DK 1214292 T3 DK1214292 T3 DK 1214292T3
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DK
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Prior art keywords
tyrosine
alpha4
madcam
vcam
ligands
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DK00965417T
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Danish (da)
English (en)
Inventor
David Y Jackson
Frederick C Sailes
Daniel P Sutherlin
Original Assignee
Genentech Inc
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Publication of DK1214292T3 publication Critical patent/DK1214292T3/da

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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WO2001021584A1 (en) 2001-03-29
AU7613800A (en) 2001-04-24
DE60035204D1 (de) 2007-07-26
CA2385882A1 (en) 2001-03-29
EP1214292A1 (en) 2002-06-19
AU780385B2 (en) 2005-03-17
US6469047B1 (en) 2002-10-22
PT1214292E (pt) 2007-09-14
US20040158076A1 (en) 2004-08-12
DE60035204T2 (de) 2008-02-21
US20090325962A1 (en) 2009-12-31
ES2288871T3 (es) 2008-02-01
JP2003509488A (ja) 2003-03-11
EP1214292B1 (en) 2007-06-13
IL148544A0 (en) 2002-09-12
CY1107721T1 (el) 2013-04-18
ATE364592T1 (de) 2007-07-15
CA2385882C (en) 2009-11-24
US7595399B2 (en) 2009-09-29
US20040110753A1 (en) 2004-06-10

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