DK1196427T3 - C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse - Google Patents

C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse

Info

Publication number
DK1196427T3
DK1196427T3 DK00954359T DK00954359T DK1196427T3 DK 1196427 T3 DK1196427 T3 DK 1196427T3 DK 00954359 T DK00954359 T DK 00954359T DK 00954359 T DK00954359 T DK 00954359T DK 1196427 T3 DK1196427 T3 DK 1196427T3
Authority
DK
Denmark
Prior art keywords
substituted
halogen
androst
new
formula
Prior art date
Application number
DK00954359T
Other languages
English (en)
Inventor
Guenter Neef
Roland Golde
Karl-Heinrich Fritzemeier
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Application granted granted Critical
Publication of DK1196427T3 publication Critical patent/DK1196427T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36Antigestagens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK00954359T 1999-07-15 2000-07-17 C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse DK1196427T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19934088A DE19934088A1 (de) 1999-07-15 1999-07-15 Neue C-19-halogensubstituierte Steroide der Androst-9(11)-en-Reihe, Verfahren zu ihrer Herstellung sowie ihre Verwendung
PCT/DE2000/002390 WO2001005805A2 (de) 1999-07-15 2000-07-17 Neue c-19-halogensubstituierte, 5-substituierte, 5-substituierte oder 6,10-carbozyklisch-kondensierte steroide der androst-9(11)-en-reihe, verfahren zu ihrer herstellung sowie ihre verwendung

Publications (1)

Publication Number Publication Date
DK1196427T3 true DK1196427T3 (da) 2007-09-10

Family

ID=7915474

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00954359T DK1196427T3 (da) 1999-07-15 2000-07-17 C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse

Country Status (10)

Country Link
US (1) US6790843B1 (da)
EP (1) EP1196427B1 (da)
JP (1) JP2003505393A (da)
AT (1) ATE362938T1 (da)
AU (1) AU6684500A (da)
DE (2) DE19934088A1 (da)
DK (1) DK1196427T3 (da)
ES (1) ES2287022T3 (da)
PT (1) PT1196427E (da)
WO (1) WO2001005805A2 (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10141937A1 (de) * 2001-08-28 2003-03-27 Alfred Schmidt Markierung der Aromatase

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3101356A (en) 1962-03-13 1963-08-20 Syntex Corp 19-halo androstenes
US5318961A (en) 1990-08-01 1994-06-07 Merrell Dow Pharmaceuticals Inc. 4-amino-Δ4-steroids and their use as 5α-reductase inhibitors
US5218110A (en) 1990-08-01 1993-06-08 Merrell Dow Pharmaceuticals 4-amino-Δ4 -steroids and their use as 5α-reductase inhibitors
CN1061987C (zh) * 1997-08-28 2001-02-14 中国科学院上海有机化学研究所 6,10-亚甲基-19-降-甾体-4-烯-3-酮化合物及其合成

Also Published As

Publication number Publication date
DE19934088A1 (de) 2001-01-18
JP2003505393A (ja) 2003-02-12
EP1196427B1 (de) 2007-05-23
EP1196427A2 (de) 2002-04-17
ES2287022T3 (es) 2007-12-16
US6790843B1 (en) 2004-09-14
WO2001005805A2 (de) 2001-01-25
ATE362938T1 (de) 2007-06-15
AU6684500A (en) 2001-02-05
WO2001005805A3 (de) 2001-09-13
DE50014346D1 (de) 2007-07-05
WO2001005805A9 (de) 2003-01-23
PT1196427E (pt) 2007-08-13

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