DK1196427T3 - C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse - Google Patents
C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelseInfo
- Publication number
- DK1196427T3 DK1196427T3 DK00954359T DK00954359T DK1196427T3 DK 1196427 T3 DK1196427 T3 DK 1196427T3 DK 00954359 T DK00954359 T DK 00954359T DK 00954359 T DK00954359 T DK 00954359T DK 1196427 T3 DK1196427 T3 DK 1196427T3
- Authority
- DK
- Denmark
- Prior art keywords
- substituted
- halogen
- androst
- new
- formula
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 150000003431 steroids Chemical class 0.000 title abstract 2
- YEHBIYDOVYBQKX-PAZXDIGFSA-N (8s,10s,13s,14s)-10,13-dimethyl-2,3,4,5,6,7,8,12,14,15,16,17-dodecahydro-1h-cyclopenta[a]phenanthrene Chemical class C([C@H]12)CC3CCCC[C@]3(C)C1=CC[C@@]1(C)[C@H]2CCC1 YEHBIYDOVYBQKX-PAZXDIGFSA-N 0.000 title 1
- 150000001438 androst-9(11)-enes Chemical class 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Steroid Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19934088A DE19934088A1 (de) | 1999-07-15 | 1999-07-15 | Neue C-19-halogensubstituierte Steroide der Androst-9(11)-en-Reihe, Verfahren zu ihrer Herstellung sowie ihre Verwendung |
| PCT/DE2000/002390 WO2001005805A2 (de) | 1999-07-15 | 2000-07-17 | Neue c-19-halogensubstituierte, 5-substituierte, 5-substituierte oder 6,10-carbozyklisch-kondensierte steroide der androst-9(11)-en-reihe, verfahren zu ihrer herstellung sowie ihre verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1196427T3 true DK1196427T3 (da) | 2007-09-10 |
Family
ID=7915474
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK00954359T DK1196427T3 (da) | 1999-07-15 | 2000-07-17 | C-19-halogensubstituerede, 5-substituerede eller 6, 10-carbocyklisk kondenserede steroider af androst-9(11)-en-rækken, fremgangsmåde til deres fremstilling samt deres anvendelse |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US6790843B1 (da) |
| EP (1) | EP1196427B1 (da) |
| JP (1) | JP2003505393A (da) |
| AT (1) | ATE362938T1 (da) |
| AU (1) | AU6684500A (da) |
| DE (2) | DE19934088A1 (da) |
| DK (1) | DK1196427T3 (da) |
| ES (1) | ES2287022T3 (da) |
| PT (1) | PT1196427E (da) |
| WO (1) | WO2001005805A2 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10141937A1 (de) * | 2001-08-28 | 2003-03-27 | Alfred Schmidt | Markierung der Aromatase |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3101356A (en) | 1962-03-13 | 1963-08-20 | Syntex Corp | 19-halo androstenes |
| US5318961A (en) | 1990-08-01 | 1994-06-07 | Merrell Dow Pharmaceuticals Inc. | 4-amino-Δ4-steroids and their use as 5α-reductase inhibitors |
| US5218110A (en) | 1990-08-01 | 1993-06-08 | Merrell Dow Pharmaceuticals | 4-amino-Δ4 -steroids and their use as 5α-reductase inhibitors |
| CN1061987C (zh) * | 1997-08-28 | 2001-02-14 | 中国科学院上海有机化学研究所 | 6,10－亚甲基－19－降－甾体－4－烯－3－酮化合物及其合成 |
-
1999
- 1999-07-15 DE DE19934088A patent/DE19934088A1/de not_active Ceased
-
2000
- 2000-07-17 AT AT00954359T patent/ATE362938T1/de not_active IP Right Cessation
- 2000-07-17 PT PT00954359T patent/PT1196427E/pt unknown
- 2000-07-17 DE DE50014346T patent/DE50014346D1/de not_active Expired - Fee Related
- 2000-07-17 DK DK00954359T patent/DK1196427T3/da active
- 2000-07-17 US US10/031,198 patent/US6790843B1/en not_active Expired - Fee Related
- 2000-07-17 JP JP2001511463A patent/JP2003505393A/ja active Pending
- 2000-07-17 AU AU66845/00A patent/AU6684500A/en not_active Abandoned
- 2000-07-17 EP EP00954359A patent/EP1196427B1/de not_active Expired - Lifetime
- 2000-07-17 WO PCT/DE2000/002390 patent/WO2001005805A2/de active IP Right Grant
- 2000-07-17 ES ES00954359T patent/ES2287022T3/es not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| DE19934088A1 (de) | 2001-01-18 |
| JP2003505393A (ja) | 2003-02-12 |
| EP1196427B1 (de) | 2007-05-23 |
| EP1196427A2 (de) | 2002-04-17 |
| ES2287022T3 (es) | 2007-12-16 |
| US6790843B1 (en) | 2004-09-14 |
| WO2001005805A2 (de) | 2001-01-25 |
| ATE362938T1 (de) | 2007-06-15 |
| AU6684500A (en) | 2001-02-05 |
| WO2001005805A3 (de) | 2001-09-13 |
| DE50014346D1 (de) | 2007-07-05 |
| WO2001005805A9 (de) | 2003-01-23 |
| PT1196427E (pt) | 2007-08-13 |
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