DK108227C - Fremgangsmåde til fremstilling af 3-carbonhydridoxy-17α-halogenethinyl-19-nor-3,5-androstadien-17β-oler. - Google Patents

Fremgangsmåde til fremstilling af 3-carbonhydridoxy-17α-halogenethinyl-19-nor-3,5-androstadien-17β-oler.

Info

Publication number
DK108227C
DK108227C DK267663AA DK267663A DK108227C DK 108227 C DK108227 C DK 108227C DK 267663A A DK267663A A DK 267663AA DK 267663 A DK267663 A DK 267663A DK 108227 C DK108227 C DK 108227C
Authority
DK
Denmark
Prior art keywords
haloethinyl
androstadiene
hydrocarbonoxy
oils
preparation
Prior art date
Application number
DK267663AA
Other languages
English (en)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Application granted granted Critical
Publication of DK108227C publication Critical patent/DK108227C/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/569Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J75/00Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK267663AA 1961-03-02 1961-04-19 Fremgangsmåde til fremstilling af 3-carbonhydridoxy-17α-halogenethinyl-19-nor-3,5-androstadien-17β-oler. DK108227C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US88575A US3072646A (en) 1961-03-02 1961-03-02 Novel 6-chloro-17alpha-haloethynyl-19-norandrostadienes and processes

Publications (1)

Publication Number Publication Date
DK108227C true DK108227C (da) 1967-10-23

Family

ID=22212174

Family Applications (1)

Application Number Title Priority Date Filing Date
DK267663AA DK108227C (da) 1961-03-02 1961-04-19 Fremgangsmåde til fremstilling af 3-carbonhydridoxy-17α-halogenethinyl-19-nor-3,5-androstadien-17β-oler.

Country Status (4)

Country Link
US (1) US3072646A (da)
DE (2) DE1593072C3 (da)
DK (1) DK108227C (da)
NO (1) NO122366B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3248405A (en) * 1962-02-09 1966-04-26 Merck & Co Inc Process for the preparation of 21-halo-19-nor-ethisterones and the 3-enol ethers thereof
DE1249264B (de) * 1962-08-24 1967-09-07 The British Drug Houses Limited London Verfahren zur Her Stellung von neuen YIi Chlorathmyl 17ß alkoxysteroiden
US3409643A (en) * 1966-03-11 1968-11-05 Schering Corp Process for the preparation of 17alpha-alkynl-17beta-alkanoyloxy steroids of the androstane and estrane series
GB1108276A (en) * 1966-03-14 1968-04-03 British Drug Houses Ltd 17ª‡-alka-1',3'-diynyl-oestra-4,9(10)-dien-3-ones
US3471531A (en) * 1966-04-07 1969-10-07 Herchel Smith Synthesis of gona-3,5-dienes

Also Published As

Publication number Publication date
DE1468333A1 (de) 1968-12-19
NO122366B (da) 1971-06-21
DE1593072B2 (de) 1973-08-23
DE1593072A1 (de) 1970-07-30
DE1593072C3 (de) 1974-04-18
US3072646A (en) 1963-01-08

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