DK1082119T3 - Mikroemulsionsforkoncentrater indeholdende en piperidinsubstans P-antagonist - Google Patents

Mikroemulsionsforkoncentrater indeholdende en piperidinsubstans P-antagonist

Info

Publication number
DK1082119T3
DK1082119T3 DK99927760T DK99927760T DK1082119T3 DK 1082119 T3 DK1082119 T3 DK 1082119T3 DK 99927760 T DK99927760 T DK 99927760T DK 99927760 T DK99927760 T DK 99927760T DK 1082119 T3 DK1082119 T3 DK 1082119T3
Authority
DK
Denmark
Prior art keywords
antagonist
microemulsion preconcentrates
piperidine substance
preconcentrates containing
piperidine
Prior art date
Application number
DK99927760T
Other languages
Danish (da)
English (en)
Inventor
Steffen Lang
Kurt Liechti
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9811200.6A external-priority patent/GB9811200D0/en
Priority claimed from GBGB9818105.0A external-priority patent/GB9818105D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK1082119T3 publication Critical patent/DK1082119T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK99927760T 1998-05-26 1999-05-26 Mikroemulsionsforkoncentrater indeholdende en piperidinsubstans P-antagonist DK1082119T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9811200.6A GB9811200D0 (en) 1998-05-26 1998-05-26 Organic compounds
GBGB9818105.0A GB9818105D0 (en) 1998-08-19 1998-08-19 Organic compounds
PCT/EP1999/003623 WO1999061025A1 (fr) 1998-05-26 1999-05-26 Preconcentres de microemulsion contenant un antagoniste de la substance p a base de piperidine

Publications (1)

Publication Number Publication Date
DK1082119T3 true DK1082119T3 (da) 2004-04-13

Family

ID=26313736

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99927760T DK1082119T3 (da) 1998-05-26 1999-05-26 Mikroemulsionsforkoncentrater indeholdende en piperidinsubstans P-antagonist

Country Status (31)

Country Link
US (2) US20020156099A1 (fr)
EP (1) EP1082119B1 (fr)
JP (1) JP4083985B2 (fr)
KR (1) KR20010043669A (fr)
CN (1) CN1270714C (fr)
AR (1) AR018376A1 (fr)
AT (1) ATE257380T1 (fr)
AU (1) AU755134B2 (fr)
BE (1) BE1012143A5 (fr)
BR (1) BR9910696A (fr)
CA (1) CA2333154C (fr)
DE (2) DE19983247T1 (fr)
DK (1) DK1082119T3 (fr)
ES (1) ES2214859T3 (fr)
FR (1) FR2779145B1 (fr)
GB (1) GB2353473A (fr)
HK (1) HK1035137A1 (fr)
HU (1) HUP0102202A3 (fr)
ID (1) ID27096A (fr)
IL (1) IL139501A0 (fr)
IT (1) IT1313551B1 (fr)
NO (1) NO20005920L (fr)
NZ (1) NZ508325A (fr)
PE (1) PE20000537A1 (fr)
PL (1) PL344245A1 (fr)
PT (1) PT1082119E (fr)
RU (1) RU2240121C2 (fr)
SK (1) SK17752000A3 (fr)
TR (1) TR200003502T2 (fr)
TW (1) TW537894B (fr)
WO (1) WO1999061025A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR018376A1 (es) 1998-05-26 2001-11-14 Novartis Ag Composiciones farmaceuticas que se pueden dispersar de una manera espontanea y el uso de las mismas para la manufactura de un medicamento
US7202282B2 (en) * 2002-04-22 2007-04-10 University Of Florida Microemulsions for selective molecular separation
GB0220953D0 (en) * 2002-09-10 2002-10-23 Novartis Ag Organic compounds
US7842791B2 (en) 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
FR2935001B1 (fr) * 2008-08-14 2011-12-30 Commissariat Energie Atomique Emulsion fluorescente
FR2934953B1 (fr) 2008-08-14 2011-01-21 Commissariat Energie Atomique Nanoemulsions de nanocristaux
FR2934955B1 (fr) 2008-08-14 2011-07-08 Commissariat Energie Atomique Encapsulation d'agents therapeutiques lipophiles ou amphiphiles dans des nanoemulsions
FR2934954B1 (fr) 2008-08-14 2011-07-22 Commissariat Energie Atomique Emulsion fluorescente de vert d'indocyanine
EP2938324B1 (fr) * 2012-12-31 2023-11-08 JRX Biotechnology, Inc. Formulations de nano-émulsion pharmaceutiques topiques liquides

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3305689A1 (de) 1983-02-18 1984-08-23 Mack Chem Pharm Pharmazeutische zubereitung mit retardwirkung
US5342625A (en) * 1988-09-16 1994-08-30 Sandoz Ltd. Pharmaceutical compositions comprising cyclosporins
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
DE4220616C2 (de) 1992-06-24 1994-12-22 Byk Gulden Lomberg Chem Fab Dexniguldipin zur intravenösen Verabreichung
EP0589843B1 (fr) 1992-09-25 2001-11-28 Novartis AG Compositions pharmaceutiques comprenant de la cyclosporine
GB2278780B (en) * 1993-05-27 1998-10-14 Sandoz Ltd Macrolide formulations
CA2185803C (fr) * 1994-03-18 2006-07-11 Edward M. Rudnic Systemes d'administration de medicaments emulsionnes
TW397825B (en) * 1994-10-14 2000-07-11 Novartis Ag Aroyl-piperidine derivatives
GB2308545B (en) 1994-10-26 1999-06-02 Novartis Ag Pharmaceutical microemulsion preconcentrates
FR2728165A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728169A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
AU696948B2 (en) * 1995-03-27 1998-09-24 Hisamitsu Pharmaceutical Co., Inc. Piperidine derivatives
NZ280689A (en) 1995-12-15 1997-08-22 Bernard Charles Sherma Sherman Pharmaceutical composition comprising a cyclosporipharmaceutical composition comprising a cyclosporin; a tocol, tocopherol or tocotrienol; and propylen; a tocol, tocopherol or tocotrienol; and propylene carbonate or polyethylene glycol ne carbonate or polyethylene glycol
GB9601120D0 (en) 1996-01-19 1996-03-20 Sandoz Ltd Organic compounds
WO1997045119A1 (fr) 1996-05-24 1997-12-04 Novartis Ag Utilisation d'antagonistes de la substance p pour traiter la phobie sociale
AR018376A1 (es) 1998-05-26 2001-11-14 Novartis Ag Composiciones farmaceuticas que se pueden dispersar de una manera espontanea y el uso de las mismas para la manufactura de un medicamento

Also Published As

Publication number Publication date
WO1999061025A1 (fr) 1999-12-02
NO20005920L (no) 2001-01-25
HUP0102202A3 (en) 2003-01-28
GB0028506D0 (en) 2001-01-10
JP2002516280A (ja) 2002-06-04
TR200003502T2 (tr) 2001-04-20
AR018376A1 (es) 2001-11-14
JP4083985B2 (ja) 2008-04-30
EP1082119A1 (fr) 2001-03-14
ITMI991164A1 (it) 2000-11-26
PE20000537A1 (es) 2000-07-10
DE69914077D1 (de) 2004-02-12
ATE257380T1 (de) 2004-01-15
AU755134B2 (en) 2002-12-05
EP1082119B1 (fr) 2004-01-07
ID27096A (id) 2001-03-01
DE19983247T1 (de) 2001-05-31
CN1270714C (zh) 2006-08-23
PT1082119E (pt) 2004-05-31
AU4500899A (en) 1999-12-13
US20020156099A1 (en) 2002-10-24
US6949257B2 (en) 2005-09-27
CN1303285A (zh) 2001-07-11
RU2240121C2 (ru) 2004-11-20
FR2779145B1 (fr) 2004-07-30
HK1035137A1 (en) 2001-11-16
ES2214859T3 (es) 2004-09-16
GB2353473A (en) 2001-02-28
KR20010043669A (ko) 2001-05-25
FR2779145A1 (fr) 1999-12-03
DE69914077T2 (de) 2004-06-09
IT1313551B1 (it) 2002-09-09
BR9910696A (pt) 2001-01-30
US20030152626A1 (en) 2003-08-14
HUP0102202A2 (hu) 2001-11-28
TW537894B (en) 2003-06-21
NO20005920D0 (no) 2000-11-23
PL344245A1 (en) 2001-10-08
CA2333154A1 (fr) 1999-12-02
IL139501A0 (en) 2001-11-25
SK17752000A3 (sk) 2001-05-10
CA2333154C (fr) 2008-07-08
NZ508325A (en) 2003-06-30
BE1012143A5 (fr) 2000-05-02

Similar Documents

Publication Publication Date Title
DE59811302D1 (de) Mikroemulsion
DE69839399D1 (de) Lymphozyten funktion antigen-1 antagonisten
NO960081D0 (no) Östrogen-agonist/antagonister
NO20000939L (no) Pæleramming
ATE278695T1 (de) Piperidinderivate
NO20000542L (no) Endothelin-antagonister
DE69834598D1 (de) Seismische Vermessung
DK1082119T3 (da) Mikroemulsionsforkoncentrater indeholdende en piperidinsubstans P-antagonist
ATE290546T1 (de) Tachykinin antagoniste
DE29722403U1 (de) Bagger
DE29800958U1 (de) Schneideinsätze
NO20002236L (no) ROV-installerte sugepæler
SE0702704L (sv) Borrskär
DE29711259U1 (de) Reflexionslichtschranke
DE69821642D1 (de) Substituierte oxime als neurokinin antagonisten
SI1082119T1 (en) Microemulsion preconcentrates containing a piperidine substance p antagonist
NO995005D0 (no) En ny fremgangsmåte
DE29716724U1 (de) Bohrgerät
ATA87997A (de) Bagger
NO20001778D0 (no) Substituerte piperidinderivater
FR2776692B1 (fr) Machine a platrer les plafonds
IT245016Y1 (it) Cesti portascarpe a marsupio
DK0964867T3 (da) Tachykininantagonister
FR2770999B1 (fr) Poincon a algies
DK1037892T3 (da) Piperidinderivater