DK0911030T3 - Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor - Google Patents

Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor

Info

Publication number
DK0911030T3
DK0911030T3 DK98117009T DK98117009T DK0911030T3 DK 0911030 T3 DK0911030 T3 DK 0911030T3 DK 98117009 T DK98117009 T DK 98117009T DK 98117009 T DK98117009 T DK 98117009T DK 0911030 T3 DK0911030 T3 DK 0911030T3
Authority
DK
Denmark
Prior art keywords
beta
antimicrobial compositions
lactamase inhibitor
vinyl pyrrolidinone
carbapenem antibiotic
Prior art date
Application number
DK98117009T
Other languages
Danish (da)
English (en)
Inventor
Peter Angehrn
Ingrid Heinze-Krauss
Malcolm Page
G F Hans Richter
Original Assignee
Basilea Pharmaceutica Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basilea Pharmaceutica Ag filed Critical Basilea Pharmaceutica Ag
Application granted granted Critical
Publication of DK0911030T3 publication Critical patent/DK0911030T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/74Synthetic polymeric materials
    • A61K31/785Polymers containing nitrogen
    • A61K31/787Polymers containing nitrogen containing heterocyclic rings having nitrogen as a ring hetero atom
    • A61K31/79Polymers of vinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DK98117009T 1997-09-15 1998-09-09 Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor DK0911030T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP97115997 1997-09-15
EP98117009A EP0911030B1 (en) 1997-09-15 1998-09-09 Antimicrobial composition comprising a vinyyl pyrrolidinon derivative and a carbapenem antibiotic or a beta-lactamase inhibitor

Publications (1)

Publication Number Publication Date
DK0911030T3 true DK0911030T3 (da) 2005-08-01

Family

ID=8227350

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98117009T DK0911030T3 (da) 1997-09-15 1998-09-09 Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor

Country Status (16)

Country Link
US (1) US6150350A (enExample)
EP (1) EP0911030B1 (enExample)
JP (1) JP4621311B2 (enExample)
KR (1) KR100630012B1 (enExample)
CN (1) CN1186021C (enExample)
AR (1) AR013490A1 (enExample)
AT (1) ATE292994T1 (enExample)
AU (1) AU747285B2 (enExample)
BR (1) BR9803443A (enExample)
CA (1) CA2247232C (enExample)
DE (1) DE69829720T2 (enExample)
DK (1) DK0911030T3 (enExample)
ES (1) ES2241084T3 (enExample)
PT (1) PT911030E (enExample)
TR (1) TR199801835A2 (enExample)
ZA (1) ZA988399B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2335288A1 (en) * 1998-06-22 1999-12-29 F. Hoffmann-La Roche Ag Propenyl cephalosporin derivatives
WO2000032605A1 (en) * 1998-12-03 2000-06-08 F. Hoffmann-La Roche Ag Bi-pyrrolidinylvinl (carba) cephalosporins
JP4583559B2 (ja) * 2000-07-24 2010-11-17 栄研化学株式会社 Mrsaスクリーニング用培地
CN100384857C (zh) * 2003-11-28 2008-04-30 浙江永宁制药厂 耐β-内酰胺酶的头孢菌素酯化合物及其盐
CN112608369A (zh) * 2020-12-30 2021-04-06 中国海洋大学 一种具有抑菌活性的细菌素及其生产方法及用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0347122A (ja) * 1989-02-21 1991-02-28 Banyu Pharmaceut Co Ltd 抗菌性組成物
DE69019395D1 (de) * 1989-02-21 1995-06-22 Banyu Pharma Co Ltd Zusammensetzung gegen Mikroben.
GB9019743D0 (en) * 1990-09-10 1990-10-24 Beecham Group Plc Novel compounds
KR100214288B1 (ko) * 1993-04-16 1999-08-02 성재갑 안개서림 방지용 내마모성 피복조성물 및 이를 도포한 합성수지 성형품
EP0620225B1 (en) * 1993-04-16 2002-11-13 Basilea Pharmaceutica AG Cephalosporin derivatives
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors
US5464616A (en) * 1994-08-04 1995-11-07 Synphar Laboratories, Ind. 6β-substituted penicillanic acids as beta-lactamase inhibitors
WO1996026943A1 (en) * 1995-02-27 1996-09-06 F.Hoffmann-La Roche Ag Derivatives of 3-pyrrolidylidene-2-one-cephalosporines
DK0841339T3 (da) * 1996-11-06 2007-07-02 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporinderivater

Also Published As

Publication number Publication date
KR19990029769A (ko) 1999-04-26
BR9803443A (pt) 2000-02-08
CA2247232C (en) 2007-08-28
JP4621311B2 (ja) 2011-01-26
JPH11140087A (ja) 1999-05-25
US6150350A (en) 2000-11-21
EP0911030A3 (en) 1999-10-13
TR199801835A3 (tr) 1999-04-21
CA2247232A1 (en) 1999-03-15
KR100630012B1 (ko) 2006-11-30
TR199801835A2 (xx) 1999-04-21
CN1186021C (zh) 2005-01-26
AU747285B2 (en) 2002-05-16
DE69829720T2 (de) 2006-03-09
ATE292994T1 (de) 2005-04-15
AU8425198A (en) 1999-04-01
PT911030E (pt) 2005-08-31
CN1216246A (zh) 1999-05-12
AR013490A1 (es) 2000-12-27
EP0911030B1 (en) 2005-04-13
DE69829720D1 (de) 2005-05-19
EP0911030A2 (en) 1999-04-28
ES2241084T3 (es) 2005-10-16
ZA988399B (en) 1999-03-15

Similar Documents

Publication Publication Date Title
DK0922697T3 (da) Substituerede pyrazolylbenzensulfonamider og anvendelse deraf som cyclooxygenase II-inhibitorer
NO942064D0 (no) yminhibitorer
FI931796A7 (fi) Portabelt krafthjaelpdon som skall haollas i handen
DE59606915D1 (de) Schraubendreher oder Schraubendrehereinsatz
FI944804A7 (fi) Pyrimidinyyliasetamideja elastaasin estäjinä
AU7145294A (en) Heterocyclic thrombin inhibitors
DE19581468T1 (de) Drehmomentschlüssel
KR970707039A (ko) 알루미노-실리케이트 유도체(alumino-silicate derivatives)
DE69415077D1 (de) Impuls-Drehmomentschlüssel
DE59600423D1 (de) Schraubgerät
FI955795A7 (fi) Aromaattisia asetyylikoliiniesteraasin inhibiittoreita
DE59600801D1 (de) Schraubgerät
FI961044L (fi) Kininogeeni-inhibiittorit
ID17792A (id) Penghambat penghambat metaloproreinase matriks
AU6183494A (en) Guanidinyl- or amidinyl-substituted heterocyclic thrombin inhibitors
DE69601302D1 (de) Drehmomentschlussel
DE69410640D1 (de) Verbesserungen bei Dichtungsmassen
NO954321L (no) 4-aryl-4-hydroksy-tetrahydropyraner og 3-aryl-3-hydroksy-tetrahydrofuraner som 5-lipoksygenase-inhibitorer
DK0911030T3 (da) Antimikrobielle præparater som omfatter et vinylpyrrolidinonderivat og et carbapenemantibiotikum eller en beta-lactamaseinhibitor
DE69404666D1 (de) Schraubenschlüssel
DE69431454D1 (de) Amylase Inhibitoren
NO961901D0 (no) 6-okso-nucleosider som er anvendbare immunoundertrykkende midler
DK0675681T3 (da) Arylamino-alkoiminoderivater og deres anvendelse som fungicider
NO950327D0 (no) Pyridoindolobenzodiazepiner og derivater som antipsykotiske midler
AU8138994A (en) Phenyl propane derivatives as antibiotics and lipoxygenase inhibitors