DK0799239T3 - Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener - Google Patents

Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Info

Publication number
DK0799239T3
DK0799239T3 DK95942689T DK95942689T DK0799239T3 DK 0799239 T3 DK0799239 T3 DK 0799239T3 DK 95942689 T DK95942689 T DK 95942689T DK 95942689 T DK95942689 T DK 95942689T DK 0799239 T3 DK0799239 T3 DK 0799239T3
Authority
DK
Denmark
Prior art keywords
antiandrogens
thioxo
aza
oxo
diastereomerically pure
Prior art date
Application number
DK95942689T
Other languages
Danish (da)
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Vincenzo Olgiati
Ambrogio Magni
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of DK0799239T3 publication Critical patent/DK0799239T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK95942689T 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener DK0799239T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (fr) 1994-12-23 1995-12-18 Derives diastereomeriquement purs du 3-oxo et du 3-thioxo-4-aza-androstane et emploi de ceux-ci comme androgenes

Publications (1)

Publication Number Publication Date
DK0799239T3 true DK0799239T3 (da) 2001-12-10

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95942689T DK0799239T3 (da) 1994-12-23 1995-12-18 Diastereomert rene 3-oxo- og 3-thioxo-4-aza-androstan-derivater og anvendelse deraf som antiandrogener

Country Status (10)

Country Link
US (1) US6147213A (fr)
EP (1) EP0799239B1 (fr)
AT (1) ATE207929T1 (fr)
AU (1) AU4387296A (fr)
DE (1) DE69523622T2 (fr)
DK (1) DK0799239T3 (fr)
ES (1) ES2163538T3 (fr)
IT (1) IT1271325B (fr)
PT (1) PT799239E (fr)
WO (1) WO1996020210A2 (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
US7835136B2 (en) 2006-11-15 2010-11-16 Energ2, Inc. Electric double layer capacitance device
PL2532648T3 (pl) * 2007-05-03 2014-07-31 Univ Yale Działające miejscowo „miękkie” antyandrogeny
CN105226284B (zh) 2009-07-01 2017-11-28 巴斯夫欧洲公司 超纯合成碳材料
US20110159375A1 (en) * 2009-12-11 2011-06-30 Energ2, Inc. Carbon materials comprising an electrochemical modifier
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
WO2012045002A1 (fr) 2010-09-30 2012-04-05 Energ2 Technologies, Inc. Agrégation améliorée de particules d'accumulation d'énergie
CN103370756B (zh) 2010-12-28 2018-05-11 巴斯福股份公司 包含增强的电化学特性的碳材料
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
CN103947017B (zh) 2011-06-03 2017-11-17 巴斯福股份公司 用于混合能量存储装置中的碳‑铅共混物
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
WO2014143213A1 (fr) 2013-03-14 2014-09-18 Energ2 Technologies, Inc. Matériaux composites carbonés comprenant des modificateurs électrochimiques d'alliage au lithium
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
WO2015137980A1 (fr) 2014-03-14 2015-09-17 Energ2 Technologies, Inc. Nouveaux procédés pour la polymérisation sol-gel en l'absence de solvant et création de structure de carbone adaptable à partir de ceux-ci
US10763501B2 (en) 2015-08-14 2020-09-01 Group14 Technologies, Inc. Nano-featured porous silicon materials
EP4286355A3 (fr) 2015-08-28 2024-05-01 Group14 Technologies, Inc. Nouveaux matériaux à insertion extrêmement durable de lithium et leurs procédés de fabrication
WO2018165610A1 (fr) 2017-03-09 2018-09-13 Group 14 Technologies, Inc. Décomposition de précurseurs contenant du silicium sur des matériaux d'échafaudage poreux
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
DE69523622T2 (de) 2002-05-29
PT799239E (pt) 2002-02-28
WO1996020210A3 (fr) 1996-09-06
DE69523622D1 (de) 2001-12-06
EP0799239A2 (fr) 1997-10-08
EP0799239B1 (fr) 2001-10-31
US6147213A (en) 2000-11-14
ITMI942626A0 (it) 1994-12-23
IT1271325B (it) 1997-05-27
ATE207929T1 (de) 2001-11-15
ITMI942626A1 (it) 1996-06-23
WO1996020210A2 (fr) 1996-07-04
ES2163538T3 (es) 2002-02-01
AU4387296A (en) 1996-07-19

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