DK0789019T3 - Fremgangsmåde til fremstilling af oxoimidazoliniumsalte - Google Patents
Fremgangsmåde til fremstilling af oxoimidazoliniumsalteInfo
- Publication number
- DK0789019T3 DK0789019T3 DK97102004T DK97102004T DK0789019T3 DK 0789019 T3 DK0789019 T3 DK 0789019T3 DK 97102004 T DK97102004 T DK 97102004T DK 97102004 T DK97102004 T DK 97102004T DK 0789019 T3 DK0789019 T3 DK 0789019T3
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- formula
- arylalkyl
- heteroaryl
- cycloalkyl
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 125000001072 heteroaryl group Chemical group 0.000 abstract 2
- 125000003107 substituted aryl group Chemical group 0.000 abstract 2
- CAAMSDWKXXPUJR-UHFFFAOYSA-N 3,5-dihydro-4H-imidazol-4-one Chemical class O=C1CNC=N1 CAAMSDWKXXPUJR-UHFFFAOYSA-N 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 150000001450 anions Chemical class 0.000 abstract 1
- 239000003125 aqueous solvent Substances 0.000 abstract 1
- 125000004446 heteroarylalkyl group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/70—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
- C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
- C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
- C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
- C07C255/42—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
- C07C255/44—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms at least one of the singly-bound nitrogen atoms being acylated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH33296 | 1996-02-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0789019T3 true DK0789019T3 (da) | 2001-09-03 |
Family
ID=4184613
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK97102004T DK0789019T3 (da) | 1996-02-09 | 1997-02-07 | Fremgangsmåde til fremstilling af oxoimidazoliniumsalte |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US5698704A (no) |
| EP (1) | EP0789019B1 (no) |
| JP (1) | JP4224629B2 (no) |
| KR (1) | KR100490220B1 (no) |
| CN (1) | CN1071747C (no) |
| AT (1) | ATE202090T1 (no) |
| CA (1) | CA2196263C (no) |
| CZ (1) | CZ291500B6 (no) |
| DE (1) | DE59703745D1 (no) |
| DK (1) | DK0789019T3 (no) |
| ES (1) | ES2158385T3 (no) |
| GR (1) | GR3036558T3 (no) |
| HU (1) | HU225694B1 (no) |
| NO (1) | NO306674B1 (no) |
| PL (1) | PL191419B1 (no) |
| PT (1) | PT789019E (no) |
| SK (1) | SK282845B6 (no) |
| TW (1) | TW407152B (no) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU218680B (hu) * | 1997-07-25 | 2000-10-30 | Sanofi-Synthelabo | Eljárás 1,3-diaza-spiro[4,4]non-1-én-4-on-származékok előállítására és 1-ciano-1-(acil-amino)-ciklopentán intermedierek |
| HU218681B (hu) * | 1997-07-25 | 2000-10-30 | Sanofi-Synthelabo | Eljárás 1,3-diaza-spiro(4,4)non-1-én-4-on-származékok előállitására és 1-ciano-1-(acil-amino)-ciklopentán intermedierek |
| US6054590A (en) * | 1998-03-25 | 2000-04-25 | Bristol-Myers Squibb Company | Imidazolone anorectic agents: II. phenyl derivatives |
| DE19912383A1 (de) * | 1998-03-27 | 1999-09-30 | Degussa | Verfahren zur Herstellung von cyclischen 4-Oxoamidinen |
| US5910595A (en) * | 1998-06-26 | 1999-06-08 | Salsbury Chemicals, Inc. | Process for preparing oximidazoles |
| US7279478B2 (en) * | 2002-09-04 | 2007-10-09 | Merck Frosst Canada & Co. | Cathepsin cysteine protease inhibitors |
| US9126998B2 (en) | 2012-11-05 | 2015-09-08 | Bayer Pharma AG | Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
| US9624214B2 (en) | 2012-11-05 | 2017-04-18 | Bayer Pharma Aktiengesellschaft | Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
| US8778964B2 (en) | 2012-11-05 | 2014-07-15 | Bayer Pharma Aktiengesellschaft | Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use |
| US8796305B2 (en) | 2012-11-05 | 2014-08-05 | Bayer Pharma Aktiengesellschaft | Carboxy-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
| US9776997B2 (en) | 2013-06-04 | 2017-10-03 | Bayer Pharma Aktiengesellschaft | 3-aryl-substituted imidazo[1,2-A]pyridines and their use |
| CA2920565A1 (en) | 2013-08-08 | 2015-02-12 | Bayer Pharma Aktiengesellschaft | Substituted pyrazolo[1,5-a]pyridine-3-carboxamides and use thereof |
| CN106459090A (zh) | 2014-02-19 | 2017-02-22 | 拜耳制药股份公司 | 3‑(嘧啶‑2‑基)咪唑并[1,2‑a]吡啶 |
| WO2015140199A1 (de) | 2014-03-21 | 2015-09-24 | Bayer Pharma Aktiengesellschaft | Cyano-substituierte imidazo[1,2-a]pyridincarboxamide und ihre verwendung |
| WO2016087343A1 (de) | 2014-12-02 | 2016-06-09 | Bayer Pharma Aktiengesellschaft | Heteroaryl-substituierte imidazo[1,2-a]pyridine und ihre verwendung |
| EP3227286B1 (de) | 2014-12-02 | 2018-12-26 | Bayer Pharma Aktiengesellschaft | Substituierte pyrazolo[1,5-a]pyridine und imidazo[1,2-a]pyrazine und ihre verwendung |
| JP2018505885A (ja) | 2015-02-05 | 2018-03-01 | バイエル・ファルマ・アクティエンゲゼルシャフト | 置換ピラゾロ［１，５−ａ］−ピリジン−３−カルボキサミドおよびその使用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4709036A (en) * | 1985-06-13 | 1987-11-24 | American Cyanamid Company | Process for the preparation of herbicidal 2-(4,4-disubstituted-5-oxo-2-imidazolin-2-yl)benzoic, nicotinic and quinoline-3-carboxylic acids, esters and salts |
| TW201738B (no) * | 1990-03-20 | 1993-03-11 | Sanofi Co | |
| CZ36294A3 (en) * | 1991-08-19 | 1994-07-13 | Du Pont | Substituted imidazilonone derivatives and pharmaceutical preparations based thereon |
-
1997
- 1997-01-29 CA CA002196263A patent/CA2196263C/en not_active Expired - Fee Related
- 1997-01-30 TW TW086101034A patent/TW407152B/zh not_active IP Right Cessation
- 1997-01-31 JP JP01815397A patent/JP4224629B2/ja not_active Expired - Fee Related
- 1997-02-03 US US08/794,641 patent/US5698704A/en not_active Expired - Lifetime
- 1997-02-05 SK SK160-97A patent/SK282845B6/sk not_active IP Right Cessation
- 1997-02-05 CN CN97102520A patent/CN1071747C/zh not_active Expired - Fee Related
- 1997-02-06 KR KR1019970003797A patent/KR100490220B1/ko not_active Expired - Fee Related
- 1997-02-07 DK DK97102004T patent/DK0789019T3/da active
- 1997-02-07 CZ CZ1997386A patent/CZ291500B6/cs not_active IP Right Cessation
- 1997-02-07 AT AT97102004T patent/ATE202090T1/de active
- 1997-02-07 HU HU9700380A patent/HU225694B1/hu not_active IP Right Cessation
- 1997-02-07 PL PL318370A patent/PL191419B1/pl not_active IP Right Cessation
- 1997-02-07 DE DE59703745T patent/DE59703745D1/de not_active Expired - Lifetime
- 1997-02-07 NO NO970581A patent/NO306674B1/no not_active IP Right Cessation
- 1997-02-07 EP EP97102004A patent/EP0789019B1/de not_active Expired - Lifetime
- 1997-02-07 PT PT97102004T patent/PT789019E/pt unknown
- 1997-02-07 ES ES97102004T patent/ES2158385T3/es not_active Expired - Lifetime
-
2001
- 2001-09-06 GR GR20010401412T patent/GR3036558T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US5698704A (en) | 1997-12-16 |
| HU9700380D0 (en) | 1997-03-28 |
| EP0789019A1 (de) | 1997-08-13 |
| SK16097A3 (en) | 1997-09-10 |
| CN1162595A (zh) | 1997-10-22 |
| NO970581D0 (no) | 1997-02-07 |
| NO970581L (no) | 1997-08-11 |
| ES2158385T3 (es) | 2001-09-01 |
| HUP9700380A2 (en) | 1997-10-28 |
| CZ38697A3 (en) | 1997-08-13 |
| CA2196263C (en) | 2004-10-26 |
| GR3036558T3 (en) | 2001-12-31 |
| NO306674B1 (no) | 1999-12-06 |
| JPH09227527A (ja) | 1997-09-02 |
| KR970061874A (ko) | 1997-09-12 |
| PL318370A1 (en) | 1997-08-18 |
| CZ291500B6 (cs) | 2003-03-12 |
| PL191419B1 (pl) | 2006-05-31 |
| PT789019E (pt) | 2001-11-30 |
| TW407152B (en) | 2000-10-01 |
| ATE202090T1 (de) | 2001-06-15 |
| KR100490220B1 (ko) | 2005-09-08 |
| EP0789019B1 (de) | 2001-06-13 |
| HUP9700380A3 (en) | 1998-04-28 |
| SK282845B6 (sk) | 2002-12-03 |
| DE59703745D1 (de) | 2001-07-19 |
| JP4224629B2 (ja) | 2009-02-18 |
| CN1071747C (zh) | 2001-09-26 |
| HU225694B1 (en) | 2007-06-28 |
| CA2196263A1 (en) | 1997-08-10 |
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