DK0705240T3 - Fremgangsmåde til fremstilling af (S)-4-aminohepta-5,6-diensyre og mellemprodukter derfor - Google Patents

Fremgangsmåde til fremstilling af (S)-4-aminohepta-5,6-diensyre og mellemprodukter derfor

Info

Publication number
DK0705240T3
DK0705240T3 DK94917458.5T DK94917458T DK0705240T3 DK 0705240 T3 DK0705240 T3 DK 0705240T3 DK 94917458 T DK94917458 T DK 94917458T DK 0705240 T3 DK0705240 T3 DK 0705240T3
Authority
DK
Denmark
Prior art keywords
aminohepta
preparation
diacetic acid
intermediates therefor
preparing
Prior art date
Application number
DK94917458.5T
Other languages
Danish (da)
English (en)
Inventor
H Michael Kolb
Original Assignee
Merrell Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Pharma Inc filed Critical Merrell Pharma Inc
Application granted granted Critical
Publication of DK0705240T3 publication Critical patent/DK0705240T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
    • C07D207/262-Pyrrolidones
    • C07D207/2732-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/30Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/36Oxygen or sulfur atoms
    • C07D207/402,5-Pyrrolidine-diones
    • C07D207/4042,5-Pyrrolidine-diones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms, e.g. succinimide

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK94917458.5T 1993-06-23 1994-05-23 Fremgangsmåde til fremstilling af (S)-4-aminohepta-5,6-diensyre og mellemprodukter derfor DK0705240T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8172393A 1993-06-23 1993-06-23

Publications (1)

Publication Number Publication Date
DK0705240T3 true DK0705240T3 (da) 1998-02-09

Family

ID=22165982

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94917458.5T DK0705240T3 (da) 1993-06-23 1994-05-23 Fremgangsmåde til fremstilling af (S)-4-aminohepta-5,6-diensyre og mellemprodukter derfor

Country Status (20)

Country Link
US (2) US5654477A (zh)
EP (1) EP0705240B1 (zh)
JP (1) JP3671252B2 (zh)
KR (1) KR100338207B1 (zh)
CN (2) CN1054369C (zh)
AT (1) ATE161822T1 (zh)
AU (1) AU672315B2 (zh)
CA (1) CA2166061C (zh)
DE (1) DE69407789T2 (zh)
DK (1) DK0705240T3 (zh)
ES (1) ES2114199T3 (zh)
FI (1) FI113859B (zh)
GR (1) GR3026123T3 (zh)
HU (1) HU223066B1 (zh)
IL (1) IL110073A (zh)
NO (1) NO306155B1 (zh)
NZ (1) NZ267007A (zh)
TW (1) TW401398B (zh)
WO (1) WO1995000470A1 (zh)
ZA (1) ZA944381B (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6750527B1 (en) * 1996-05-30 2004-06-15 Kabushiki Kaisha Toshiba Semiconductor integrated circuit device having a plurality of wells, test method of testing the semiconductor integrated circuit device, and test device which executes the test method
WO2011161529A2 (en) 2010-06-24 2011-12-29 Edge-To-Edge Global Investments Limited Nutritional supplement
CN105777586A (zh) * 2016-04-14 2016-07-20 安徽省逸欣铭医药科技有限公司 S(+)氨己烯酸酯衍生物及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2120244B (en) * 1982-05-17 1985-05-01 Merrell Toraude & Co Aminoalkadiene derivative
US4668703A (en) * 1983-07-07 1987-05-26 Syntex (U.S.A.) Inc. γ-allenyl-γ-aminobutyric acids
US4661510A (en) * 1983-08-17 1987-04-28 Syntex (U.S.A.) Inc. α-allenic-α-amino acids as enzyme inhibitors
IL100360A (en) * 1990-12-17 1998-08-16 Merrell Dow Pharma HISTORY OF PYROLIDINONE USED AS SUBSTANCE (S) -Vinyl and Alanyl GABA

Also Published As

Publication number Publication date
JPH08511801A (ja) 1996-12-10
CN1093853C (zh) 2002-11-06
WO1995000470A1 (en) 1995-01-05
CA2166061C (en) 1999-02-23
FI956247A0 (fi) 1995-12-22
US5654477A (en) 1997-08-05
AU672315B2 (en) 1996-09-26
HU223066B1 (hu) 2004-03-01
CN1256266A (zh) 2000-06-14
GR3026123T3 (en) 1998-05-29
EP0705240B1 (en) 1998-01-07
FI956247A (fi) 1995-12-22
DE69407789T2 (de) 1998-07-09
CA2166061A1 (en) 1995-01-05
HUT73629A (en) 1996-08-28
ATE161822T1 (de) 1998-01-15
NO955253D0 (no) 1995-12-22
KR100338207B1 (ko) 2003-02-11
IL110073A (en) 2000-09-28
NO306155B1 (no) 1999-09-27
TW401398B (en) 2000-08-11
AU6917294A (en) 1995-01-17
EP0705240A1 (en) 1996-04-10
JP3671252B2 (ja) 2005-07-13
ES2114199T3 (es) 1998-05-16
NO955253L (no) 1996-02-21
NZ267007A (en) 1996-12-20
IL110073A0 (en) 1994-10-07
ZA944381B (en) 1995-02-09
FI113859B (fi) 2004-06-30
CN1125937A (zh) 1996-07-03
DE69407789D1 (de) 1998-02-12
US5756762A (en) 1998-05-26
CN1054369C (zh) 2000-07-12
HU9503708D0 (en) 1996-02-28

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