DK0700913T3 - 5,6-Dihydro-4H-imidazo[4,5,1,ij]quinoliner, fremgangsmåder til fremstiliing deraf, deres anvendelse som lægemiddel og melle - Google Patents

5,6-Dihydro-4H-imidazo[4,5,1,ij]quinoliner, fremgangsmåder til fremstiliing deraf, deres anvendelse som lægemiddel og melle

Info

Publication number
DK0700913T3
DK0700913T3 DK95113849T DK95113849T DK0700913T3 DK 0700913 T3 DK0700913 T3 DK 0700913T3 DK 95113849 T DK95113849 T DK 95113849T DK 95113849 T DK95113849 T DK 95113849T DK 0700913 T3 DK0700913 T3 DK 0700913T3
Authority
DK
Denmark
Prior art keywords
dihydro
processes
preparation
quinolines
imidazo
Prior art date
Application number
DK95113849T
Other languages
Danish (da)
English (en)
Inventor
Edward J Glamkowski
Brian S Freed
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Application granted granted Critical
Publication of DK0700913T3 publication Critical patent/DK0700913T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK95113849T 1994-09-09 1995-09-04 5,6-Dihydro-4H-imidazo[4,5,1,ij]quinoliner, fremgangsmåder til fremstiliing deraf, deres anvendelse som lægemiddel og melle DK0700913T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/304,041 US5500423A (en) 1994-09-09 1994-09-09 5,6-dihydro-4H-imidazo[4,5,1-ij]quinolines

Publications (1)

Publication Number Publication Date
DK0700913T3 true DK0700913T3 (da) 1999-02-01

Family

ID=23174785

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95113849T DK0700913T3 (da) 1994-09-09 1995-09-04 5,6-Dihydro-4H-imidazo[4,5,1,ij]quinoliner, fremgangsmåder til fremstiliing deraf, deres anvendelse som lægemiddel og melle

Country Status (8)

Country Link
US (2) US5500423A (es)
EP (1) EP0700913B1 (es)
JP (1) JP3117183B2 (es)
AT (1) ATE166876T1 (es)
CA (1) CA2157860C (es)
DE (1) DE69502783T2 (es)
DK (1) DK0700913T3 (es)
ES (1) ES2118483T3 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH11514361A (ja) * 1995-10-16 1999-12-07 藤沢薬品工業株式会社 H+−ATPaseとしての複素環式化合物
TW546302B (en) * 1998-05-08 2003-08-11 Biochemie Sa Improvements in macrolide production
AUPP818099A0 (en) * 1999-01-14 1999-02-11 Fujisawa Pharmaceutical Co., Ltd. New n-containing heterocyclic compounds
PL1731518T3 (pl) 2004-03-31 2014-11-28 Nippon Soda Co Cykliczny związek aminowy oraz środek zwalczający szkodniki
JP4871289B2 (ja) * 2005-10-06 2012-02-08 日本曹達株式会社 環状アミン化合物および有害生物防除剤
GB201220157D0 (en) * 2012-11-08 2012-12-26 Selvita Sa Substitute tricyclic benzimidazoles as kinase inhibitors

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3142679A (en) * 1964-07-28 Pipejazino alkylamevo quinoline deriva-
US3200123A (en) * 1962-01-26 1965-08-10 Richardson Merreil Inc Imidazoquinolines
US3975531A (en) * 1973-10-02 1976-08-17 A. H. Robins Company, Incorporated 4-(5- And 7-)benzoylindolin-2-ones and pharmaceutical uses thereof
US4209519A (en) * 1978-03-13 1980-06-24 The United States Of America As Represented By The Secretary Of The Army Anti-leishmanial lepidine derivatives
IE57646B1 (en) * 1983-12-16 1993-02-10 Wyeth John & Brother Ltd Derivatives of imidazoquinolines and analogues thereof
JPS6354363A (ja) * 1986-08-26 1988-03-08 Ss Pharmaceut Co Ltd キノリン誘導体
US5064852A (en) * 1988-12-16 1991-11-12 Pfizer Inc. Indolinone derivatives
AU675645B2 (en) * 1992-04-27 1997-02-13 Mochida Pharmaceutical Co., Ltd. Tricyclic compound having antiallergic effect
FR2710915B1 (fr) * 1993-10-04 1995-11-24 Synthelabo Dérivés de pipéridine, leur préparation et leur utilisation en thérapeutique.

Also Published As

Publication number Publication date
ATE166876T1 (de) 1998-06-15
EP0700913A1 (en) 1996-03-13
DE69502783D1 (de) 1998-07-09
EP0700913B1 (en) 1998-06-03
US5563272A (en) 1996-10-08
US5500423A (en) 1996-03-19
DE69502783T2 (de) 1998-11-12
CA2157860C (en) 2001-07-17
JP3117183B2 (ja) 2000-12-11
JPH0892251A (ja) 1996-04-09
ES2118483T3 (es) 1998-09-16
CA2157860A1 (en) 1996-03-10

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