DK0611774T3 - Racemiseringsfri fremstilling af amider og peptider i nærværelse af katalytiske mængder af en N-hydroxyforbindelse - Google Patents
Racemiseringsfri fremstilling af amider og peptider i nærværelse af katalytiske mængder af en N-hydroxyforbindelseInfo
- Publication number
- DK0611774T3 DK0611774T3 DK94101784T DK94101784T DK0611774T3 DK 0611774 T3 DK0611774 T3 DK 0611774T3 DK 94101784 T DK94101784 T DK 94101784T DK 94101784 T DK94101784 T DK 94101784T DK 0611774 T3 DK0611774 T3 DK 0611774T3
- Authority
- DK
- Denmark
- Prior art keywords
- amides
- peptides
- hydroxy compound
- racemization
- catalytic amounts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
- C07K1/084—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents containing nitrogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Analytical Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Indole Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH51893 | 1993-02-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
DK0611774T3 true DK0611774T3 (da) | 1999-11-15 |
Family
ID=4188840
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK94101784T DK0611774T3 (da) | 1993-02-19 | 1994-02-07 | Racemiseringsfri fremstilling af amider og peptider i nærværelse af katalytiske mængder af en N-hydroxyforbindelse |
Country Status (8)
Country | Link |
---|---|
US (2) | US5536816A (zh) |
EP (1) | EP0611774B1 (zh) |
JP (1) | JP2524685B2 (zh) |
CN (1) | CN1035873C (zh) |
AT (1) | ATE180491T1 (zh) |
DE (1) | DE59408292D1 (zh) |
DK (1) | DK0611774T3 (zh) |
ES (1) | ES2133428T3 (zh) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE180491T1 (de) * | 1993-02-19 | 1999-06-15 | Hoffmann La Roche | Racemisierungsfreie herstellung von amiden und peptiden in gegenwart katalytischer mengen einer n-hydroxy-verbindung |
GB9424842D0 (en) * | 1994-12-09 | 1995-02-08 | British Tech Group | Pharmaceutical compositions |
EP0823424A1 (de) * | 1996-08-09 | 1998-02-11 | F. Hoffmann-La Roche Ag | Verfahren zur Herstellung von Chinargin |
US5914404A (en) * | 1996-08-09 | 1999-06-22 | Hoffmann-La Roche Inc. | Process for the preparation of quinargine |
DE59709770D1 (de) | 1996-12-11 | 2003-05-15 | Hoffmann La Roche | Verfahren zur Herstellung gemischter Anhydride |
CA2331330A1 (en) * | 1998-06-17 | 1999-12-23 | Magainin Pharmaceuticals, Inc. | Non-enzymatic chemical amidation process |
KR20020002480A (ko) * | 1999-03-17 | 2002-01-09 | 한센 핀 베네드, 안네 제헤르, 웨이콥 마리안느 | 펩티드의 아실화법 및 신규한 아실화제 |
US6719080B1 (en) | 2000-01-10 | 2004-04-13 | The United States Of America As Represented By The Administrator Of The Environmental Protection Agency | Hydraulic hybrid vehicle |
KR100863078B1 (ko) * | 2001-03-19 | 2008-10-10 | 후지모리 고교 가부시키가이샤 | 트롬빈 유도체 및 그 제조방법, 안하이드로트롬빈 유도체및 그 제조방법, 혈소판 응집야기 조성물, 혈소판응집야기 방법, 임상검사약, 임상검사방법, 혈전형성억제제, 흡착체 및 그 제조방법, 정제된 혈액응고 제 ⅷ인자의 제조방법 |
US7423166B2 (en) * | 2001-12-13 | 2008-09-09 | Advanced Technology Materials, Inc. | Stabilized cyclosiloxanes for use as CVD precursors for low-dielectric constant thin films |
US7273921B2 (en) | 2002-09-25 | 2007-09-25 | Novo Nordisk A/S | Method for producing acylated peptides |
US20040077703A1 (en) * | 2002-10-02 | 2004-04-22 | Soll Mark D. | Nodulisporic acid derivative spot-on formulations for combating parasites |
CN103113177B (zh) * | 2013-02-06 | 2015-02-04 | 济南志合医药科技有限公司 | 一种酰胺的制备方法 |
ES2624961T3 (es) | 2013-03-21 | 2017-07-18 | Sanofi-Aventis Deutschland Gmbh | Síntesis de productos de péptido que contienen imida cíclica |
US10087221B2 (en) | 2013-03-21 | 2018-10-02 | Sanofi-Aventis Deutschland Gmbh | Synthesis of hydantoin containing peptide products |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2202613C3 (de) * | 1972-01-20 | 1974-06-20 | Farbwerke Hoechst Ag, Vormals Meister Lucius & Bruening, 6000 Frankfurt | Verfahren zur Herstellung von Peptiden |
EP0662078B1 (en) * | 1992-09-28 | 2003-05-02 | Research Corporation Technologies, Inc. | Reagents for peptide couplings |
ATE180491T1 (de) * | 1993-02-19 | 1999-06-15 | Hoffmann La Roche | Racemisierungsfreie herstellung von amiden und peptiden in gegenwart katalytischer mengen einer n-hydroxy-verbindung |
-
1994
- 1994-02-07 AT AT94101784T patent/ATE180491T1/de not_active IP Right Cessation
- 1994-02-07 ES ES94101784T patent/ES2133428T3/es not_active Expired - Lifetime
- 1994-02-07 DK DK94101784T patent/DK0611774T3/da not_active Application Discontinuation
- 1994-02-07 EP EP94101784A patent/EP0611774B1/de not_active Revoked
- 1994-02-07 DE DE59408292T patent/DE59408292D1/de not_active Expired - Fee Related
- 1994-02-15 JP JP6039301A patent/JP2524685B2/ja not_active Expired - Lifetime
- 1994-02-15 US US08/196,750 patent/US5536816A/en not_active Expired - Fee Related
- 1994-02-18 CN CN94101380A patent/CN1035873C/zh not_active Expired - Fee Related
-
1996
- 1996-02-23 US US08/606,104 patent/US5750649A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
ES2133428T3 (es) | 1999-09-16 |
ATE180491T1 (de) | 1999-06-15 |
US5750649A (en) | 1998-05-12 |
EP0611774B1 (de) | 1999-05-26 |
JP2524685B2 (ja) | 1996-08-14 |
JPH06256225A (ja) | 1994-09-13 |
DE59408292D1 (de) | 1999-07-01 |
CN1035873C (zh) | 1997-09-17 |
US5536816A (en) | 1996-07-16 |
CN1111237A (zh) | 1995-11-08 |
EP0611774A1 (de) | 1994-08-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK0611774T3 (da) | Racemiseringsfri fremstilling af amider og peptider i nærværelse af katalytiske mængder af en N-hydroxyforbindelse | |
ATE179166T1 (de) | N'-substituierte-n,n'diacylhydrazin-insektizide | |
AU634294B2 (en) | Fibrinogen receptor antagonists | |
DK0422937T3 (da) | Fibrinogenreceptorantagonister | |
NO930193D0 (no) | Biarylsubstituerte 4-aminosmoersyreamider | |
DE69132435D1 (de) | Inhibitoren retroviraler Proteasen | |
DK0623589T3 (da) | Koblingsreagens og fremgangsmåde til kobling af aminer med carboxylsyrer | |
FI102966B (fi) | Menetelmä terapeuttisesti käyttökelpoisten guanidiinien valmistamiseks i | |
EP0742209A3 (en) | Process for the preparation of an optically active quinoline demevalonolacton and process for the preparation of a salt of an optically active quinoline demevalolon | |
DE69415353D1 (de) | Verfahren zur Herstellung von Maleinamidsäure | |
EP1048694A4 (en) | AZO COMPOUNDS AND METHOD FOR THE PRODUCTION THEREOF | |
DK20980A (da) | Fremgangsmaade til fremstilling af carboxylsyreamider og peptider | |
TW228520B (zh) | ||
DK0510625T3 (da) | Fremgangsmåde til fremstilling af lysstabilisatorer med hindrede aminogrupper | |
DE59301060D1 (de) | Substituierte Aminosäureamide. | |
DK0640608T3 (da) | Mellemprodukter til syntese af cephalosporiner | |
NO178231C (no) | Umettede polyesterharpiksblandinger og anvendelse av disse | |
NZ514653A (en) | Process for producing an amide compound by reacting a compound with an amino group with a polyaminocarboxylic acid anhydride | |
ZA948631B (en) | 5-arylisoxazol-4-yl-substituted 2-amino carboxylic acid compounds | |
DK659188A (da) | Fremgangsmaade til fremstiling af isothiazoloner | |
EP0684227A3 (zh) | ||
DE3164897D1 (en) | Process for preparing 1-amino-3-aryloxy-2-propanols and 1-amino-2-aryl-2-ethanols | |
ATE161263T1 (de) | 2,4-diamino-1,3,5-triazinyl-6- phosphonsäurederivate | |
DE69406382D1 (de) | Verfahren zur Herstellung von N-Phenyl-N-(4-Piperidinyl)Amid-Derivaten | |
DE69427343D1 (de) | Verfahren zur herstellung von 3-substituierten cephem-derivaten |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |