DK0591333T3 - Azanorbornanderivater - Google Patents

Azanorbornanderivater

Info

Publication number
DK0591333T3
DK0591333T3 DK92913342.9T DK92913342T DK0591333T3 DK 0591333 T3 DK0591333 T3 DK 0591333T3 DK 92913342 T DK92913342 T DK 92913342T DK 0591333 T3 DK0591333 T3 DK 0591333T3
Authority
DK
Denmark
Prior art keywords
pct
sec
formula
date
azanorbornane derivatives
Prior art date
Application number
DK92913342.9T
Other languages
Danish (da)
English (en)
Inventor
Brian Thomas Oneill
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK0591333T3 publication Critical patent/DK0591333T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Ink Jet (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Fertilizers (AREA)
DK92913342.9T 1991-06-21 1992-06-11 Azanorbornanderivater DK0591333T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71988491A 1991-06-21 1991-06-21

Publications (1)

Publication Number Publication Date
DK0591333T3 true DK0591333T3 (da) 1997-05-20

Family

ID=24891766

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92913342.9T DK0591333T3 (da) 1991-06-21 1992-06-11 Azanorbornanderivater

Country Status (18)

Country Link
US (1) US5604252A (cg-RX-API-DMAC10.html)
EP (1) EP0591333B1 (cg-RX-API-DMAC10.html)
KR (1) KR940701384A (cg-RX-API-DMAC10.html)
AT (1) ATE149497T1 (cg-RX-API-DMAC10.html)
AU (1) AU2188992A (cg-RX-API-DMAC10.html)
CA (1) CA2111335A1 (cg-RX-API-DMAC10.html)
DE (1) DE69217945T2 (cg-RX-API-DMAC10.html)
DK (1) DK0591333T3 (cg-RX-API-DMAC10.html)
FI (1) FI935726A7 (cg-RX-API-DMAC10.html)
HU (1) HUT68957A (cg-RX-API-DMAC10.html)
IE (1) IE921987A1 (cg-RX-API-DMAC10.html)
IL (1) IL102208A0 (cg-RX-API-DMAC10.html)
MX (1) MX9203053A (cg-RX-API-DMAC10.html)
NO (1) NO934727D0 (cg-RX-API-DMAC10.html)
PT (1) PT100607A (cg-RX-API-DMAC10.html)
TW (1) TW202432B (cg-RX-API-DMAC10.html)
WO (1) WO1993000330A2 (cg-RX-API-DMAC10.html)
ZA (1) ZA924527B (cg-RX-API-DMAC10.html)

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AU4396193A (en) * 1992-08-04 1994-03-03 Pfizer Inc. 3-benzylamino-2-phenyl-piperidine derivatives as substance p receptor antagonists
EP1114823A3 (en) * 1992-08-19 2001-07-18 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
JP2722279B2 (ja) * 1992-12-10 1998-03-04 ファイザー・インク． アミノメチレンで置換した非芳香族複素環式化合物及びサブスタンスｐのアンタゴニストとしての使用
FR2700472B1 (fr) 1993-01-19 1995-02-17 Rhone Poulenc Rorer Sa Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2.
US5340826A (en) * 1993-02-04 1994-08-23 Pfizer Inc. Pharmaceutical agents for treatment of urinary incontinence
US5635510A (en) * 1993-05-06 1997-06-03 Merrell Pharmaceuticals Inc. Substituted pyrrolidin-3-yl-alkyl-piperidines
US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
EP0653208A3 (en) * 1993-11-17 1995-10-11 Pfizer Substance P antagonists for the treatment or prevention of sunburn.
EP0659409A3 (en) * 1993-11-23 1995-08-09 Pfizer Substance P antagonists for the inhibition of angiogenesis.
EP0655246A1 (en) * 1993-11-30 1995-05-31 Pfizer Inc. Substance P antagonists for the treatment of disorders caused by helicobacter pylori or other spiral urease-positive gram-negative bacteria
NZ292683A (en) 1994-08-25 1998-07-28 Merrell Pharma Inc Piperidine derivatives
FR2728165A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
FR2728166A1 (fr) 1994-12-19 1996-06-21 Oreal Composition topique contenant un antagoniste de substance p
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
KR100414321B1 (ko) * 1995-04-13 2004-02-18 아벤티스 파마슈티칼스 인크. 타치키닌수용체길항활성을갖는신규한치환된피페라진유도체
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FR2741262B1 (fr) 1995-11-20 1999-03-05 Oreal Utilisation d'un antagoniste de tnf-alpha pour le traitement des rougeurs cutanees d'origine neurogene
US6194406B1 (en) 1995-12-20 2001-02-27 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease
US6423704B2 (en) 1995-12-20 2002-07-23 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases
US5998439A (en) 1996-02-21 1999-12-07 Hoescht Marion Roussel, Inc. Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
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US5922737A (en) * 1996-02-21 1999-07-13 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases
CA2324116A1 (en) * 1999-10-25 2001-04-25 Susan Beth Sobolov-Jaynes Nk-1 receptor antagonists and eletriptan for the treatment of migraine
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GB8823605D0 (en) * 1988-10-07 1988-11-16 Merck Sharp & Dohme Therapeutic agents
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FI931370L (fi) * 1990-09-28 1993-03-26 Pfizer Kvaeve innehaollande analoger av icke-aromatiska heterocykliska foereningar med en fusionerad ring

Also Published As

Publication number Publication date
ATE149497T1 (de) 1997-03-15
FI935726A0 (fi) 1993-12-20
DE69217945T2 (de) 1997-06-12
NO934727L (no) 1993-12-20
EP0591333A1 (en) 1994-04-13
PT100607A (pt) 1993-08-31
DE69217945D1 (de) 1997-04-10
WO1993000330A2 (en) 1993-01-07
IE921987A1 (en) 1992-12-30
KR940701384A (ko) 1994-05-28
US5604252A (en) 1997-02-18
EP0591333B1 (en) 1997-03-05
IL102208A0 (en) 1993-01-14
HUT68957A (en) 1995-08-28
FI935726L (fi) 1993-12-20
MX9203053A (es) 1992-12-01
WO1993000330A3 (en) 1993-03-04
NO934727D0 (no) 1993-12-20
CA2111335A1 (en) 1993-01-07
AU2188992A (en) 1993-01-25
ZA924527B (en) 1993-12-20
TW202432B (cg-RX-API-DMAC10.html) 1993-03-21
HU9303666D0 (en) 1994-04-28
FI935726A7 (fi) 1993-12-20

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