DE69305276D1 - Arylglycinamidderivate, Verfahren zur deren Herstellung und deren Verwendung zur Therapie der Dysurie - Google Patents
Arylglycinamidderivate, Verfahren zur deren Herstellung und deren Verwendung zur Therapie der DysurieInfo
- Publication number
- DE69305276D1 DE69305276D1 DE69305276T DE69305276T DE69305276D1 DE 69305276 D1 DE69305276 D1 DE 69305276D1 DE 69305276 T DE69305276 T DE 69305276T DE 69305276 T DE69305276 T DE 69305276T DE 69305276 D1 DE69305276 D1 DE 69305276D1
- Authority
- DE
- Germany
- Prior art keywords
- carbon atoms
- group
- denotes
- lower alkyl
- substituents
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
- C07C237/20—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
- C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/56—Ring systems containing bridged rings
- C07C2603/58—Ring systems containing bridged rings containing three rings
- C07C2603/70—Ring systems containing bridged rings containing three rings containing only six-membered rings
- C07C2603/74—Adamantanes
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP21969992 | 1992-07-27 | ||
JP19688293A JP3429338B2 (ja) | 1992-07-27 | 1993-07-14 | 新規なアリールグリシンアミド誘導体及びその製造法 |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69305276D1 true DE69305276D1 (de) | 1996-11-14 |
DE69305276T2 DE69305276T2 (de) | 1997-04-30 |
Family
ID=26510045
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69305276T Expired - Fee Related DE69305276T2 (de) | 1992-07-27 | 1993-07-20 | Arylglycinamidderivate, Verfahren zur deren Herstellung und deren Verwendung zur Therapie der Dysurie |
Country Status (11)
Country | Link |
---|---|
US (1) | US5439919A (de) |
EP (1) | EP0581167B1 (de) |
JP (1) | JP3429338B2 (de) |
KR (1) | KR100295027B1 (de) |
AT (1) | ATE143943T1 (de) |
AU (1) | AU658316B2 (de) |
CA (1) | CA2101310C (de) |
DE (1) | DE69305276T2 (de) |
ES (1) | ES2093332T3 (de) |
HU (1) | HU215846B (de) |
TW (1) | TW271435B (de) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5706027A (en) * | 1985-12-18 | 1998-01-06 | Spacetec Imc Corporation | Force and torque converter for use in a computer input device |
CA2179574A1 (en) | 1995-06-26 | 1996-12-27 | Tomomi Okada | Substituted piperidine derivative and medicine comprising the same |
EP0882699A4 (de) * | 1996-08-06 | 2001-03-21 | Taisho Pharmaceutical Co Ltd | Aminoverbindungen und angiotensin iv rezeptor agonisten |
DE10111058A1 (de) * | 2001-03-08 | 2002-09-12 | Boehringer Ingelheim Pharma | Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und NK¶1¶-Rezeptor-Antagonisten |
US6620438B2 (en) | 2001-03-08 | 2003-09-16 | Boehringer Ingelheim Pharma Kg | Pharmaceutical compositions based on anticholinergics and NK1-receptor antagonists |
DE10143009A1 (de) * | 2001-09-03 | 2003-03-20 | Molecular And Clinical Drug Re | Präparat zur Behandlung weiblicher Inkontinenz |
WO2003088204A1 (en) * | 2002-04-12 | 2003-10-23 | Obermeyer Henry K | Multi-axis joystick and transducer means therefore |
WO2004004629A2 (en) | 2002-07-08 | 2004-01-15 | Ranbaxy Laboratories Limited | 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists |
ATE396969T1 (de) | 2002-07-31 | 2008-06-15 | Ranbaxy Lab Ltd | 3,6-disubstituierte azabicyclo (3.1.0)hexanderivate, die sich als muscarinrezeptorantagonisten eignen |
WO2004014363A1 (en) | 2002-08-09 | 2004-02-19 | Ranbaxy Laboratories Limited | 3,6-disubstituted azabicyclo [3.1.0] hexane derivatives useful as muscarinic receptor antagonist |
JP2006501236A (ja) | 2002-08-23 | 2006-01-12 | ランバクシー ラボラトリーズ リミテッド | ムスカリン性レセプター拮抗薬としてのフルオロおよびスルホニルアミノ含有3,6−二置換アザビシクロ(3.1.0)ヘキサン誘導体 |
US7232835B2 (en) | 2002-12-10 | 2007-06-19 | Ranbaxy Laboratories Limited | 3,6-Disubstituted azabicyclo derivatives as muscarinic receptor antagonists |
US7501443B2 (en) | 2002-12-23 | 2009-03-10 | Ranbaxy Laboratories Limited | Flavaxate derivatives as muscarinic receptor antagonists |
EP1583741A1 (de) | 2002-12-23 | 2005-10-12 | Ranbaxy Laboratories, Limited | 1-substituierte-3-pyrrolidin-derivate als muscarinrezeptor-antagonisten |
US7488748B2 (en) | 2003-01-28 | 2009-02-10 | Ranbaxy Laboratories Limited | 3,6-Disubstituted azabicyclo hexane derivatives as muscarinic receptor antagonists |
US7517905B2 (en) | 2003-04-09 | 2009-04-14 | Ranbaxy Laboratories Limited | Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists |
WO2004089363A1 (en) | 2003-04-10 | 2004-10-21 | Ranbaxy Laboratories Limited | Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists |
EP1615887A1 (de) | 2003-04-10 | 2006-01-18 | Ranbaxy Laboratories, Ltd. | 3, 6-disubstitutierte azabicyclohexanderivate als muscarinrezeptorantagonisten |
AU2004228452A1 (en) | 2003-04-11 | 2004-10-21 | Ranbaxy Laboratories Limited | Azabicyclo derivatives as muscarinic receptor antagonists |
EP1740553A1 (de) * | 2004-04-14 | 2007-01-10 | AstraZeneca AB | Arylglycinamidderivate und deren verwendung als nk1-antagonisten und serotoninwiederaufnahmehemmer |
WO2007045979A1 (en) | 2005-10-19 | 2007-04-26 | Ranbaxy Laboratories Limited | Pharmaceutical compositions of muscarinic receptor antagonists |
EP1889612A3 (de) * | 2006-07-24 | 2008-03-19 | Jan Kees Piet Bruinstroop | Verfahren zur Steuerung von Harnlassen |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1269556A (fr) * | 1956-05-14 | 1961-08-18 | Upjohn Co | Procédé de préparation de nu-mono-substituées-alpha-(tertio-aminoalcoyl)-alphaphénylacétamides |
US4783537A (en) * | 1985-11-13 | 1988-11-08 | Pennwalt Corporation | α-(aminoalkyl)-arylacetic acid derivatives |
JPH0783006B2 (ja) * | 1987-12-23 | 1995-09-06 | 株式会社半導体エネルギー研究所 | 薄膜加工方法 |
US5153226A (en) * | 1989-08-31 | 1992-10-06 | Warner-Lambert Company | Acat inhibitors for treating hypocholesterolemia |
-
1993
- 1993-07-14 JP JP19688293A patent/JP3429338B2/ja not_active Expired - Fee Related
- 1993-07-20 HU HUP9302090A patent/HU215846B/hu not_active IP Right Cessation
- 1993-07-20 AT AT93111592T patent/ATE143943T1/de not_active IP Right Cessation
- 1993-07-20 ES ES93111592T patent/ES2093332T3/es not_active Expired - Lifetime
- 1993-07-20 EP EP93111592A patent/EP0581167B1/de not_active Expired - Lifetime
- 1993-07-20 US US08/093,854 patent/US5439919A/en not_active Expired - Fee Related
- 1993-07-20 DE DE69305276T patent/DE69305276T2/de not_active Expired - Fee Related
- 1993-07-23 AU AU42169/93A patent/AU658316B2/en not_active Ceased
- 1993-07-23 TW TW082105885A patent/TW271435B/zh active
- 1993-07-26 KR KR1019930014143A patent/KR100295027B1/ko not_active IP Right Cessation
- 1993-07-26 CA CA002101310A patent/CA2101310C/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
JPH0692921A (ja) | 1994-04-05 |
DE69305276T2 (de) | 1997-04-30 |
CA2101310A1 (en) | 1994-01-28 |
AU658316B2 (en) | 1995-04-06 |
AU4216993A (en) | 1994-02-03 |
ATE143943T1 (de) | 1996-10-15 |
TW271435B (de) | 1996-03-01 |
US5439919A (en) | 1995-08-08 |
JP3429338B2 (ja) | 2003-07-22 |
KR100295027B1 (ko) | 2001-09-17 |
KR940005534A (ko) | 1994-03-21 |
CA2101310C (en) | 2001-07-03 |
EP0581167A1 (de) | 1994-02-02 |
ES2093332T3 (es) | 1996-12-16 |
EP0581167B1 (de) | 1996-10-09 |
HUT64944A (en) | 1994-03-28 |
HU9302090D0 (en) | 1993-10-28 |
HU215846B (hu) | 1999-04-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE69305276T2 (de) | Arylglycinamidderivate, Verfahren zur deren Herstellung und deren Verwendung zur Therapie der Dysurie | |
ATE89263T1 (de) | Naphthalin-derivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische zusammensetzungen. | |
ATE109466T1 (de) | Neue derivate des aminopiperidins, aminopyrrolidins und des aminoperhydroazepins, verfahren zur herstellung und diese enthaltende arzneimittel. | |
DE69627042D1 (de) | Isocumarinderivate und deren verwendung in medikamenten | |
DE69019859D1 (de) | Chinolon-Derivate und deren Salze, Verfahren zu deren Herstellung und diese enthaltende antibakterielle Wirkstoffe. | |
ATE138663T1 (de) | Oxothiolane und derivate, diese enthaltende pharmazeutische zubereitungen und ihre verwendung als arzneimittel | |
GR3034023T3 (en) | Phenyl carboxamide-isoxazole-derivatives and salts, process for their preparation, their use as pharmaceuticals, and pharmaceutical compositions containing them. | |
EP0379483A4 (en) | 1,2,3,4,10,14b-hexahydrodibenzo c,f¨pyrazino- 1,2-a¨azepino derivatives and 10-aza, 10-oxa and 10-thia analogues | |
ATE148128T1 (de) | Anthracyclinglycosid-derivate und verfahren zu ihrer herstellung | |
NO940026L (no) | Mono- og bis alkylamino-antracykliner | |
ATE163649T1 (de) | Peptide, herstellung und deren verwendung | |
DE3465085D1 (en) | Derivatives of 4-(3-alkynyloxy-2-hydroxy-propyl)-piperazin-1-yl-n-phenyl acetamide, their preparation and their therapeutical use | |
AU3309793A (en) | An amphoteric tricyclic compound | |
ATE184282T1 (de) | Cyclopropan-derivate und diese enthaltende antivirale mittel | |
DE69225381T2 (de) | Nootrope Wirkstoffe | |
DE68903893D1 (de) | 20,21-dinoreburnamenin-derivate, substituiert in position 15 durch eine aminogruppe und deren salze, verfahren zu deren herstellung und die auf diese weise erhaltenen zwischenverbindungen, deren anwendung als arzneimittel und diese enthaltende pharmazeutische zusammensetzungen. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |