DE69122437D1 - Purinyl und Pyrimidinyltetrahydrofurane - Google Patents

Purinyl und Pyrimidinyltetrahydrofurane

Info

Publication number
DE69122437D1
DE69122437D1 DE69122437T DE69122437T DE69122437D1 DE 69122437 D1 DE69122437 D1 DE 69122437D1 DE 69122437 T DE69122437 T DE 69122437T DE 69122437 T DE69122437 T DE 69122437T DE 69122437 D1 DE69122437 D1 DE 69122437D1
Authority
DE
Germany
Prior art keywords
pyrimidinyltetrahydrofurane
purinyl
chem
exhibited
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69122437T
Other languages
English (en)
Other versions
DE69122437T2 (de
Inventor
Robert Zahler
Val S Goodfellow
Saleem Ahmad
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Application granted granted Critical
Publication of DE69122437D1 publication Critical patent/DE69122437D1/de
Publication of DE69122437T2 publication Critical patent/DE69122437T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DE69122437T 1990-07-02 1991-07-02 Purinyl und Pyrimidinyltetrahydrofurane Expired - Lifetime DE69122437T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54695790A 1990-07-02 1990-07-02

Publications (2)

Publication Number Publication Date
DE69122437D1 true DE69122437D1 (de) 1996-11-07
DE69122437T2 DE69122437T2 (de) 1997-03-13

Family

ID=24182716

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69122437T Expired - Lifetime DE69122437T2 (de) 1990-07-02 1991-07-02 Purinyl und Pyrimidinyltetrahydrofurane

Country Status (14)

Country Link
EP (1) EP0464769B1 (de)
JP (1) JP3055818B2 (de)
AT (1) ATE143662T1 (de)
AU (1) AU633743B2 (de)
CA (1) CA2046002C (de)
DE (1) DE69122437T2 (de)
DK (1) DK0464769T3 (de)
ES (1) ES2093051T3 (de)
GR (1) GR3022158T3 (de)
HU (1) HU209437B (de)
IE (1) IE76731B1 (de)
NZ (1) NZ238708A (de)
PT (1) PT98186B (de)
ZA (1) ZA914894B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5231174A (en) * 1992-02-27 1993-07-27 University Of Iowa Research Foundation 2'isodideoxy-β-D-nucleosides as stable antiviral agents
US5314893A (en) * 1993-01-25 1994-05-24 Bristol-Myers Squibb Co. Antiviral tetrahydropyrans
JPH06263756A (ja) * 1993-03-04 1994-09-20 Asahi Breweries Ltd イソヌクレオシド誘導体
CN110818714A (zh) * 2018-08-14 2020-02-21 连云港润众制药有限公司 一种恩替卡韦中间体的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL89258A0 (en) * 1988-02-16 1989-09-10 Lilly Co Eli 2',3'-dideoxy-2',2'-difluoro-nucleosides
SE8802173D0 (sv) * 1988-06-10 1988-06-10 Astra Ab Pyrimidine derivatives
US5126347A (en) * 1989-02-13 1992-06-30 Hoffmann-La Roche Inc. Isomeric dideoxynuclesides
NZ232993A (en) * 1989-04-24 1992-10-28 Squibb & Sons Inc Purinyl and pyrimidinyl tetrahydrofurans

Also Published As

Publication number Publication date
ZA914894B (en) 1992-04-29
PT98186B (pt) 1998-12-31
CA2046002C (en) 2001-06-12
NZ238708A (en) 1994-04-27
EP0464769B1 (de) 1996-10-02
GR3022158T3 (en) 1997-03-31
HU209437B (en) 1994-06-28
HU912216D0 (en) 1991-12-30
EP0464769A3 (en) 1992-08-05
EP0464769A2 (de) 1992-01-08
IE76731B1 (en) 1997-11-05
PT98186A (pt) 1992-05-29
ATE143662T1 (de) 1996-10-15
DE69122437T2 (de) 1997-03-13
CA2046002A1 (en) 1992-01-03
ES2093051T3 (es) 1996-12-16
JPH04244082A (ja) 1992-09-01
AU7940491A (en) 1992-01-09
AU633743B2 (en) 1993-02-04
IE912243A1 (en) 1992-01-15
HUT58103A (en) 1992-01-28
DK0464769T3 (da) 1996-11-18
JP3055818B2 (ja) 2000-06-26

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition