DE60326060D1 - Nichtvernetzende pyrroloä2,1-cüä1,4übenzodiazepine als potentielle antitumor-agentien und ihre herstellung - Google Patents

Nichtvernetzende pyrroloä2,1-cüä1,4übenzodiazepine als potentielle antitumor-agentien und ihre herstellung

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Publication number
DE60326060D1
DE60326060D1 DE60326060T DE60326060T DE60326060D1 DE 60326060 D1 DE60326060 D1 DE 60326060D1 DE 60326060 T DE60326060 T DE 60326060T DE 60326060 T DE60326060 T DE 60326060T DE 60326060 D1 DE60326060 D1 DE 60326060D1
Authority
DE
Germany
Prior art keywords
preparation
pyrroloa2
crosslinking
antitumor agents
pyrrolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60326060T
Other languages
English (en)
Inventor
Ahmed Kamal
Gujjar Ramesh
Olepu Srinivas
Poddutoori Ramulu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Council of Scientific and Industrial Research CSIR
Original Assignee
Council of Scientific and Industrial Research CSIR
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by Council of Scientific and Industrial Research CSIR filed Critical Council of Scientific and Industrial Research CSIR
Application granted granted Critical
Publication of DE60326060D1 publication Critical patent/DE60326060D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
DE60326060T 2003-03-31 2003-03-31 Nichtvernetzende pyrroloä2,1-cüä1,4übenzodiazepine als potentielle antitumor-agentien und ihre herstellung Expired - Lifetime DE60326060D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/401,782 US6884799B2 (en) 2003-03-31 2003-03-31 Non-cross-linking pyrrolo[2,1-c][1,4]benzodiazepines and process thereof
PCT/IB2003/001182 WO2004087717A1 (en) 2003-03-31 2003-03-31 Non-cross-linking pyrrolo[2,1-c][1,4]benzodiazepines as potential antitumour agents and process thereof

Publications (1)

Publication Number Publication Date
DE60326060D1 true DE60326060D1 (de) 2009-03-19

Family

ID=33477800

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60326060T Expired - Lifetime DE60326060D1 (de) 2003-03-31 2003-03-31 Nichtvernetzende pyrroloä2,1-cüä1,4übenzodiazepine als potentielle antitumor-agentien und ihre herstellung

Country Status (7)

Country Link
US (1) US6884799B2 (de)
EP (1) EP1608664B1 (de)
AT (1) ATE421967T1 (de)
AU (1) AU2003215821B2 (de)
CA (1) CA2520898C (de)
DE (1) DE60326060D1 (de)
WO (1) WO2004087717A1 (de)

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Also Published As

Publication number Publication date
CA2520898C (en) 2009-10-20
AU2003215821A1 (en) 2004-10-25
US6884799B2 (en) 2005-04-26
AU2003215821B2 (en) 2009-04-23
CA2520898A1 (en) 2004-10-14
WO2004087717A1 (en) 2004-10-14
ATE421967T1 (de) 2009-02-15
EP1608664A1 (de) 2005-12-28
EP1608664B1 (de) 2009-01-28
US20040192679A1 (en) 2004-09-30

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