DE60106281T2 - Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms - Google Patents

Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms Download PDF

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Publication number
DE60106281T2
DE60106281T2 DE60106281T DE60106281T DE60106281T2 DE 60106281 T2 DE60106281 T2 DE 60106281T2 DE 60106281 T DE60106281 T DE 60106281T DE 60106281 T DE60106281 T DE 60106281T DE 60106281 T2 DE60106281 T2 DE 60106281T2
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Germany
Prior art keywords
rapamycin
carbon atoms
antiestrogen
use according
product
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60106281T
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German (de)
English (en)
Other versions
DE60106281D1 (de
Inventor
Yixian Zhang
Michelle Tammy SADLER
Philip Frost
Martin Lee GREENBERGER
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
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Wyeth LLC
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22840171&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE60106281(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth LLC filed Critical Wyeth LLC
Publication of DE60106281D1 publication Critical patent/DE60106281D1/de
Application granted granted Critical
Publication of DE60106281T2 publication Critical patent/DE60106281T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE60106281T 2000-08-11 2001-08-06 Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms Expired - Fee Related DE60106281T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22432600P 2000-08-11 2000-08-11
US224326P 2000-08-11
PCT/US2001/024615 WO2002013802A2 (en) 2000-08-11 2001-08-06 Method of treating estrogen receptor positive carcinoma

Publications (2)

Publication Number Publication Date
DE60106281D1 DE60106281D1 (de) 2004-11-11
DE60106281T2 true DE60106281T2 (de) 2005-02-24

Family

ID=22840171

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60106281T Expired - Fee Related DE60106281T2 (de) 2000-08-11 2001-08-06 Verfahren zur Behandlung eines Östrogenrezeptor-positiven Karzinoms

Country Status (14)

Country Link
US (1) US6511986B2 (cg-RX-API-DMAC7.html)
EP (1) EP1318837B1 (cg-RX-API-DMAC7.html)
JP (1) JP2004507465A (cg-RX-API-DMAC7.html)
CN (1) CN100448487C (cg-RX-API-DMAC7.html)
AR (1) AR033555A1 (cg-RX-API-DMAC7.html)
AT (1) ATE278421T1 (cg-RX-API-DMAC7.html)
AU (1) AU2001283139A1 (cg-RX-API-DMAC7.html)
CA (1) CA2416976C (cg-RX-API-DMAC7.html)
DE (1) DE60106281T2 (cg-RX-API-DMAC7.html)
DK (1) DK1318837T3 (cg-RX-API-DMAC7.html)
ES (1) ES2228932T3 (cg-RX-API-DMAC7.html)
MX (1) MXPA03001245A (cg-RX-API-DMAC7.html)
PT (1) PT1318837E (cg-RX-API-DMAC7.html)
WO (1) WO2002013802A2 (cg-RX-API-DMAC7.html)

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Publication number Publication date
HK1056687A1 (en) 2004-02-27
WO2002013802A2 (en) 2002-02-21
CA2416976C (en) 2008-05-20
ES2228932T3 (es) 2005-04-16
EP1318837A2 (en) 2003-06-18
PT1318837E (pt) 2004-12-31
US6511986B2 (en) 2003-01-28
AR033555A1 (es) 2003-12-26
DK1318837T3 (da) 2005-01-10
CA2416976A1 (en) 2002-02-21
DE60106281D1 (de) 2004-11-11
US20020045638A1 (en) 2002-04-18
CN1446106A (zh) 2003-10-01
CN100448487C (zh) 2009-01-07
WO2002013802A3 (en) 2003-03-27
MXPA03001245A (es) 2003-05-27
ATE278421T1 (de) 2004-10-15
EP1318837B1 (en) 2004-10-06
JP2004507465A (ja) 2004-03-11
AU2001283139A1 (en) 2002-02-25

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