DE4120109A1 - 3-aryl- oder 3-hetaryl-(beta)-carboline, deren herstellung und verwendung in arzneimitteln - Google Patents
3-aryl- oder 3-hetaryl-(beta)-carboline, deren herstellung und verwendung in arzneimittelnInfo
- Publication number
- DE4120109A1 DE4120109A1 DE4120109A DE4120109A DE4120109A1 DE 4120109 A1 DE4120109 A1 DE 4120109A1 DE 4120109 A DE4120109 A DE 4120109A DE 4120109 A DE4120109 A DE 4120109A DE 4120109 A1 DE4120109 A1 DE 4120109A1
- Authority
- DE
- Germany
- Prior art keywords
- carboline
- methoxymethyl
- benzyloxy
- alkyl
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Priority Applications (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4120109A DE4120109A1 (de) | 1991-06-15 | 1991-06-15 | 3-aryl- oder 3-hetaryl-(beta)-carboline, deren herstellung und verwendung in arzneimitteln |
PCT/DE1992/000497 WO1992022549A1 (fr) | 1991-06-15 | 1992-06-12 | 3-ARYL- OU 3-HETARYL-β-CARBOLINES, LEUR FABRICATION ET LEUR UTILISATION DANS DES MEDICAMENTS |
JP5500741A JPH06501956A (ja) | 1991-06-15 | 1992-06-12 | 3―アリール―または3―ヘテロアリール―β―カルボリン、その製造および薬剤としての使用 |
EP92912055A EP0543968A1 (fr) | 1991-06-15 | 1992-06-12 | 3-ARYL- OU 3-HETARYL-$g(b)-CARBOLINES, LEUR FABRICATION ET LEUR UTILISATION DANS DES MEDICAMENTS |
CA002089569A CA2089569A1 (fr) | 1991-06-15 | 1992-06-12 | 3-aryl- ou 3-hetaryl-.beta.-carbolines; preparation et utilisation dans des agents pharmaceutiques |
PT100593A PT100593A (pt) | 1991-06-15 | 1992-06-15 | 3-aril-beta-carbolinas ou 3-heteroaril-beta-carbolinas, processos para a sua preparacao e composicoes farmaceuticas que as contem |
US08/329,051 US5543519A (en) | 1991-06-15 | 1994-10-25 | 3-aryl or 3-hetaryl-β-carbolines, their production and use in pharmaceutical agents |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4120109A DE4120109A1 (de) | 1991-06-15 | 1991-06-15 | 3-aryl- oder 3-hetaryl-(beta)-carboline, deren herstellung und verwendung in arzneimitteln |
Publications (1)
Publication Number | Publication Date |
---|---|
DE4120109A1 true DE4120109A1 (de) | 1992-12-17 |
Family
ID=6434220
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE4120109A Withdrawn DE4120109A1 (de) | 1991-06-15 | 1991-06-15 | 3-aryl- oder 3-hetaryl-(beta)-carboline, deren herstellung und verwendung in arzneimitteln |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP0543968A1 (fr) |
JP (1) | JPH06501956A (fr) |
CA (1) | CA2089569A1 (fr) |
DE (1) | DE4120109A1 (fr) |
PT (1) | PT100593A (fr) |
WO (1) | WO1992022549A1 (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1134221A1 (fr) * | 2000-03-15 | 2001-09-19 | Aventis Pharma Deutschland GmbH | Bêta-carbolines substituées comme inhibiteurs de lkB kinase |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4330175A1 (de) * | 1993-08-31 | 1995-03-02 | Schering Ag | Alkoxy-substituierte beta-Carboline |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57123180A (en) * | 1980-12-17 | 1982-07-31 | Schering Ag | 3-substituted beta-carboline, manufacture and psychotropic drug containing same |
DE3240511A1 (de) * | 1982-10-29 | 1984-05-03 | Schering AG, 1000 Berlin und 4709 Bergkamen | Verfahren zur herstellung von ss-carbolinderivaten |
DE3322895A1 (de) * | 1983-06-23 | 1985-01-03 | Schering AG, 1000 Berlin und 4709 Bergkamen | Neue ss-carboline, verfahren zur ihrer herstellung und ihre verwendung als arzneimittel (s) |
DK240084D0 (da) * | 1984-05-15 | 1984-05-15 | Ferrosan As | New beta-carboline-3-oxadiazolyl derivatives |
DE3540654A1 (de) * | 1985-11-13 | 1987-05-14 | Schering Ag | Phenoxy-substituierte ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel |
DE3608089A1 (de) * | 1986-03-08 | 1987-09-10 | Schering Ag | Heteroaryl-oxy-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel |
AU619203B2 (en) * | 1987-08-28 | 1992-01-23 | Schering Aktiengesellschaft | Isoxazole-beta-carboline derivatives |
DE3903753A1 (de) * | 1989-02-06 | 1990-08-23 | Schering Ag | Verfahren zur herstellung waessriger mischmicelloesungen |
DE3943225A1 (de) * | 1989-12-23 | 1991-06-27 | Schering Ag | Neue ss-carboline, verfahren zu deren herstellung und deren verwendung in arzneimitteln |
-
1991
- 1991-06-15 DE DE4120109A patent/DE4120109A1/de not_active Withdrawn
-
1992
- 1992-06-12 CA CA002089569A patent/CA2089569A1/fr not_active Abandoned
- 1992-06-12 WO PCT/DE1992/000497 patent/WO1992022549A1/fr not_active Application Discontinuation
- 1992-06-12 EP EP92912055A patent/EP0543968A1/fr not_active Withdrawn
- 1992-06-12 JP JP5500741A patent/JPH06501956A/ja active Pending
- 1992-06-15 PT PT100593A patent/PT100593A/pt not_active Application Discontinuation
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1134221A1 (fr) * | 2000-03-15 | 2001-09-19 | Aventis Pharma Deutschland GmbH | Bêta-carbolines substituées comme inhibiteurs de lkB kinase |
Also Published As
Publication number | Publication date |
---|---|
PT100593A (pt) | 1993-08-31 |
WO1992022549A1 (fr) | 1992-12-23 |
CA2089569A1 (fr) | 1992-12-16 |
JPH06501956A (ja) | 1994-03-03 |
EP0543968A1 (fr) | 1993-06-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8127 | New person/name/address of the applicant |
Owner name: SCHERING AG, 13353 BERLIN, DE |
|
8130 | Withdrawal |