DE3784526D1 - Cembran-diterpene-verbindungen zur herstellung von zusammensetzungen, die inhibitoren der histamin-freisetzung enthalten. - Google Patents
Cembran-diterpene-verbindungen zur herstellung von zusammensetzungen, die inhibitoren der histamin-freisetzung enthalten.Info
- Publication number
- DE3784526D1 DE3784526D1 DE9191106347T DE3784526T DE3784526D1 DE 3784526 D1 DE3784526 D1 DE 3784526D1 DE 9191106347 T DE9191106347 T DE 9191106347T DE 3784526 T DE3784526 T DE 3784526T DE 3784526 D1 DE3784526 D1 DE 3784526D1
- Authority
- DE
- Germany
- Prior art keywords
- cembrane
- compositions containing
- histamine release
- producing compositions
- release inhibitors
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP61292747A JPH0798746B2 (ja) | 1986-12-09 | 1986-12-09 | リソゾ−ム放出抑制剤 |
Publications (2)
Publication Number | Publication Date |
---|---|
DE3784526D1 true DE3784526D1 (de) | 1993-04-08 |
DE3784526T2 DE3784526T2 (de) | 1993-09-09 |
Family
ID=17785809
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8787402578T Expired - Fee Related DE3781653T2 (de) | 1986-12-09 | 1987-11-16 | Verwendung von cembrane-diterpene verbindungen zur herstellung von zusammensetzungen, die inhibitoren der freigabe von lysosomen enthalten. |
DE9191106347T Expired - Fee Related DE3784526T2 (de) | 1986-12-09 | 1987-11-16 | Cembran-diterpene-verbindungen zur herstellung von zusammensetzungen, die inhibitoren der histamin-freisetzung enthalten. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8787402578T Expired - Fee Related DE3781653T2 (de) | 1986-12-09 | 1987-11-16 | Verwendung von cembrane-diterpene verbindungen zur herstellung von zusammensetzungen, die inhibitoren der freigabe von lysosomen enthalten. |
Country Status (4)
Country | Link |
---|---|
US (1) | US4906794A (de) |
EP (2) | EP0271387B1 (de) |
JP (1) | JPH0798746B2 (de) |
DE (2) | DE3781653T2 (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0454140A (ja) * | 1990-06-20 | 1992-02-21 | Mitsubishi Kasei Corp | 共役ジエン化合物 |
US5276217A (en) * | 1992-03-19 | 1994-01-04 | University Of Hawaii | Cyclic anti-tumor promoter compounds, compositions and methods for production and use |
US6204289B1 (en) | 1997-06-05 | 2001-03-20 | Vesna A. Eterovic | Cembranoid inhibitors of nicotinic acetylcholine receptors |
US6489357B1 (en) | 1998-06-04 | 2002-12-03 | University Of Puerto Rico | Tobacco cembranoids block the expression of the behavioral sensitization to nicotine and inhibit neuronal acetylcholine receptors |
WO2000027839A1 (en) * | 1998-11-05 | 2000-05-18 | The Regents Of The University Of California | Rameswaralide and rameswaralide derivatives |
US20040092583A1 (en) * | 2001-01-02 | 2004-05-13 | Elizabeth Shanahan-Prendergast | Treatment for inhibiting neoplastic lesions |
WO2003095404A1 (en) * | 2002-05-09 | 2003-11-20 | University Of Mississippi | Cembranoids with chemopreventive activity |
CN105732656B (zh) * | 2016-03-31 | 2017-10-27 | 中国人民解放军第二军医大学 | 肉芝软珊瑚中的一种四萜类化合物及其用途 |
CN109134184B (zh) * | 2017-06-16 | 2021-03-19 | 中国科学院上海药物研究所 | 二萜类化合物、其制备方法及用途 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS588365B2 (ja) * | 1975-09-22 | 1983-02-15 | キタハラ ヨシオ | フホウワ 14 インカンカゴウブツノ セイホウ |
JPS5522624A (en) * | 1978-08-03 | 1980-02-18 | Mitsubishi Chem Ind Ltd | Preparation of diterpene alcohol |
JPS5661317A (en) * | 1979-10-25 | 1981-05-26 | Mitsubishi Chem Ind Ltd | Cembranolide diterpene |
JPS61109713A (ja) * | 1984-11-05 | 1986-05-28 | Japan Tobacco Inc | 抗腫瘍剤 |
JPH0610177B2 (ja) * | 1985-05-08 | 1994-02-09 | エーザイ株式会社 | キノン化合物 |
JPH0794387B2 (ja) * | 1986-12-09 | 1995-10-11 | 三菱化学株式会社 | 皮膚用製剤 |
JPH0794388B2 (ja) * | 1987-03-17 | 1995-10-11 | 三菱化学株式会社 | 乾癬治療剤 |
-
1986
- 1986-12-09 JP JP61292747A patent/JPH0798746B2/ja not_active Expired - Lifetime
-
1987
- 1987-11-16 EP EP87402578A patent/EP0271387B1/de not_active Expired - Lifetime
- 1987-11-16 EP EP91106347A patent/EP0448128B1/de not_active Expired - Lifetime
- 1987-11-16 DE DE8787402578T patent/DE3781653T2/de not_active Expired - Fee Related
- 1987-11-16 DE DE9191106347T patent/DE3784526T2/de not_active Expired - Fee Related
-
1989
- 1989-02-10 US US07/308,476 patent/US4906794A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
DE3784526T2 (de) | 1993-09-09 |
EP0448128A3 (en) | 1991-11-27 |
EP0271387A2 (de) | 1988-06-15 |
DE3781653T2 (de) | 1993-02-18 |
EP0271387A3 (en) | 1990-07-25 |
JPH0798746B2 (ja) | 1995-10-25 |
US4906794A (en) | 1990-03-06 |
DE3781653D1 (de) | 1992-10-15 |
JPS63145224A (ja) | 1988-06-17 |
EP0271387B1 (de) | 1992-09-09 |
EP0448128A2 (de) | 1991-09-25 |
EP0448128B1 (de) | 1993-03-03 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE3581937D1 (de) | Verfahren zur herstellung von modulen, aufgestapelte integrierte schaltungen enthalten. | |
ATE54664T1 (de) | Verfahren zur herstellung von 2-oxo-1,3dioxolanen. | |
DE3585687D1 (de) | Verfahren zur herstellung von 1-hydroxyvitamin-d-verbindungen. | |
DE3784803D1 (de) | Verfahren zur herstellung von mikrokapseln, die polymer-dickungsoel enthalten. | |
DE3767835D1 (de) | Verfahren zur herstellung von fluor-halogen-aethern, ausgehend von fluoroxyverbindungen und halogenierten olefinen. | |
DE3881511D1 (de) | Mechanisch aufgebrachte beschichtungen, die schmiermittel enthalten. | |
DE3586093D1 (de) | Verfahren zur herstellung von aluminiumnitridpulver. | |
DE3861825D1 (de) | Verfahren zur herstellung von (2,2)-paracyclophan. | |
DE3784526D1 (de) | Cembran-diterpene-verbindungen zur herstellung von zusammensetzungen, die inhibitoren der histamin-freisetzung enthalten. | |
DE69013132D1 (de) | Verfahren zur Herstellung von Octa-2,7-dien-1-ol. | |
DE3870065D1 (de) | Zusammensetzungen von polyarylalkanoligomeren, verfahren zu deren herstellung. | |
DE3581884D1 (de) | Verfahren zur herstellung von 2,2'-methylen-bis-(4-hydrocarbyl-6-benzotriazolyl(phenolen). | |
BG38637A3 (en) | Method for preparing 2- exo- hydroxy- 7- oxabicyclo [2, 2, 1] heptanes | |
ATE25520T1 (de) | Verfahren zur herstellung von (-)-2-(1-(2,6de811210 | |
ATE6255T1 (de) | Verfahren zur herstellung von 2,3,5trichlorpyridin. | |
DE3382318D1 (de) | Verfahren zur herstellung von alpha-substituierten beta-dicarbonyl-, beta-cyancarbonyl- und beta-dicyanverbindungen. | |
DE69021907D1 (de) | Verfahren zur Herstellung von kristallinem, sinterfähigem Aluminiumnitridpulver. | |
DE3765956D1 (de) | Verfahren zur herstellung von 1-methyl-3,5,7-triaza-1-azoniatricyclodecan-halogeniden. | |
DE3887212D1 (de) | Verfahren zur Herstellung von Derivaten von 6,7-Diazyl-7-desacetylforskolin. | |
DE3773240D1 (de) | Hydrochinolinverbindungen, diese enthaltende zusammensetzungen und verfahren zu ihrer herstellung. | |
DE3674161D1 (de) | Verfahren zum gewinnen von nuetzlichen verbindungen, die mindestens dimethylterephthalat enthalten aus den hochsiedenden beiprodukten der herstellung von dimethylterephthalat. | |
AT381703B (de) | Verfahren zur herstellung von 1-(1,3-benzodioxol-5-yl)-2-pyrrolidinon | |
DE3766127D1 (de) | Verfahren zur herstellung von blockcopolymeren aus propylen. | |
ATE9800T1 (de) | Verfahren zur herstellung von 4-amino-6tert.butyl-3-mercapto-1,2,4-triazin-5-on. | |
DE3578066D1 (de) | Verfahren zur herstellung von alpha, beta-diaminoacrylnitrilen. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |