DE3765682D1 - Thiolactam-n-essigsaeure-derivate, ihre herstellung und verwendung. - Google Patents

Thiolactam-n-essigsaeure-derivate, ihre herstellung und verwendung.

Info

Publication number
DE3765682D1
DE3765682D1 DE8787302825T DE3765682T DE3765682D1 DE 3765682 D1 DE3765682 D1 DE 3765682D1 DE 8787302825 T DE8787302825 T DE 8787302825T DE 3765682 T DE3765682 T DE 3765682T DE 3765682 D1 DE3765682 D1 DE 3765682D1
Authority
DE
Germany
Prior art keywords
thiolactam
production
acetic acid
acid derivatives
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE8787302825T
Other languages
English (en)
Inventor
Kanji Meguro
Hitoshi Ikeda
Yujiro Yamamoto
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Senju Pharmaceutical Co Ltd
Takeda Pharmaceutical Co Ltd
Original Assignee
Senju Pharmaceutical Co Ltd
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senju Pharmaceutical Co Ltd, Takeda Chemical Industries Ltd filed Critical Senju Pharmaceutical Co Ltd
Application granted granted Critical
Publication of DE3765682D1 publication Critical patent/DE3765682D1/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/141,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/161,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/12Ophthalmic agents for cataracts
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/341,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/361,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE8787302825T 1986-04-17 1987-04-01 Thiolactam-n-essigsaeure-derivate, ihre herstellung und verwendung. Expired - Fee Related DE3765682D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP8929586 1986-04-17
JP14594186 1986-06-20

Publications (1)

Publication Number Publication Date
DE3765682D1 true DE3765682D1 (de) 1990-11-29

Family

ID=26430721

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8787302825T Expired - Fee Related DE3765682D1 (de) 1986-04-17 1987-04-01 Thiolactam-n-essigsaeure-derivate, ihre herstellung und verwendung.

Country Status (19)

Country Link
US (1) US4771050A (de)
EP (1) EP0243018B1 (de)
JP (1) JPS63107970A (de)
KR (1) KR870010024A (de)
CN (1) CN1020098C (de)
AR (1) AR244674A1 (de)
AU (1) AU602641B2 (de)
CA (1) CA1287629C (de)
DE (1) DE3765682D1 (de)
DK (1) DK184587A (de)
ES (1) ES2022889B3 (de)
FI (1) FI89711C (de)
GR (1) GR3001210T3 (de)
HK (1) HK108293A (de)
HU (1) HU198699B (de)
IE (1) IE60246B1 (de)
NO (1) NO167916C (de)
PT (1) PT84704B (de)
SU (1) SU1538895A3 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2996475B2 (ja) * 1989-12-22 1999-12-27 サントリー株式会社 ベンズオキサジノン誘導体及びそれを有効成分として含有する除草剤
TW200402B (de) * 1990-08-13 1993-02-21 Senju Pharma Co
AU638154B2 (en) * 1990-10-04 1993-06-17 Suntory Limited Benzoxazine derivative and herbicide containing same as an active ingredient
IE914455A1 (en) * 1990-12-27 1992-07-01 Green Cross Corp 1,4-benzothiazine-2-acetic acid derivatives, processes for production thereof
DE69329618T2 (de) * 1992-08-31 2001-05-17 Santen Pharmaceutical Co., Ltd 3-oxo-1,4-benzothiazin-derivate
JP3126541B2 (ja) * 1993-03-26 2001-01-22 千寿製薬株式会社 ベンゾチアゾール誘導体、その製法及びその用途
WO1995013269A1 (fr) * 1993-11-12 1995-05-18 Santen Pharmaceutical Co., Ltd. Derive de 1,4-benzothiazine
HUP0000838A3 (en) * 1997-04-15 2001-04-28 Csir Extract containing steroid-glucosid, process for its isolation and synthesis, pharmaceutical composition containing it having appetite suppressant activity
GB2355657B (en) * 1999-10-27 2004-07-28 Phytopharm Plc Inhibitors Of Gastric Acid Secretion
US6713477B1 (en) 2000-04-19 2004-03-30 Sumitomo Pharmaceuticals Company, Limited Hydroxamic acid derivatives
GB2363985B (en) 2000-06-30 2004-09-29 Phytopharm Plc Extracts,compounds & pharmaceutical compositions having anti-diabetic activity and their use
PL365378A1 (en) 2000-11-30 2005-01-10 Pfizer Products Inc. Combination of gaba agonists and aldose reductase inhibitors
EP1726587B1 (de) * 2004-03-02 2010-09-01 Dainippon Sumitomo Pharma Co., Ltd. Benzothiazin-3-one verbindung und zwischenprodukt dafür
US20110092566A1 (en) * 2004-11-19 2011-04-21 Srivastava Satish K Treatment of cancer with aldose reductase inhibitors
US20070197512A1 (en) * 2006-01-27 2007-08-23 Japan Tobacco Inc. Carboxylic Acid Compounds and Use Thereof
WO2007086504A1 (ja) * 2006-01-27 2007-08-02 Japan Tobacco Inc. カルボン酸化合物及びその用途
US8877717B2 (en) 2007-03-12 2014-11-04 Zadec Aps Anti-diabetic extract of rooibos
US8273746B2 (en) * 2007-03-23 2012-09-25 The Board Of Regents Of The University Of Texas System Methods involving aldose reductase inhibitors
US20090270490A1 (en) * 2008-04-24 2009-10-29 The Board Of Regents Of The University Of Texas System Methods involving aldose reductase inhibition
EP2654749B1 (de) 2010-12-23 2017-05-10 The Board of Regents of The University of Texas System Verfahren zur behandlung von copd
WO2019165195A1 (en) 2018-02-22 2019-08-29 Srivastava Satish Combination therapy for the treatment of cancer

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1173942A (en) * 1967-06-06 1969-12-10 Bellon Labor Sa Roger New 2,3-Dihydro-1,4-Benzoxazines
US3923709A (en) * 1974-08-30 1975-12-02 Monsanto Co 3,4-Dihydro-3-oxo-2H-1,4-benzothiazines and benzoxazines
IE58312B1 (en) * 1984-05-18 1993-09-08 Union Pharma Scient Appl Heterocyclic derivatives, processes for their preparation and drugs in which they are present, which are useful especially as aldose reductase inhibitors

Also Published As

Publication number Publication date
DK184587A (da) 1987-10-18
PT84704B (pt) 1989-11-30
EP0243018B1 (de) 1990-10-24
AR244674A1 (es) 1993-11-30
ES2022889B3 (es) 1991-12-16
FI89711C (fi) 1993-11-10
AU602641B2 (en) 1990-10-18
HK108293A (en) 1993-10-22
HU198699B (en) 1989-11-28
JPS63107970A (ja) 1988-05-12
IE60246B1 (en) 1994-06-15
NO167916C (no) 1991-12-27
CN1020098C (zh) 1993-03-17
DK184587D0 (da) 1987-04-10
FI871719A (fi) 1987-10-18
EP0243018A1 (de) 1987-10-28
PT84704A (en) 1987-05-01
NO871526L (no) 1987-10-19
GR3001210T3 (en) 1992-07-30
CN87102891A (zh) 1987-11-04
IE871012L (en) 1987-10-17
SU1538895A3 (ru) 1990-01-23
US4771050A (en) 1988-09-13
CA1287629C (en) 1991-08-13
KR870010024A (ko) 1987-11-30
HUT45515A (en) 1988-07-28
JPH034550B2 (de) 1991-01-23
NO167916B (no) 1991-09-16
NO871526D0 (no) 1987-04-10
AU7073087A (en) 1987-10-22
FI89711B (fi) 1993-07-30
FI871719A0 (fi) 1987-04-16

Similar Documents

Publication Publication Date Title
ATE89560T1 (de) Makrolid-derivate, ihre herstellung und ihre verwendung.
DE3768922D1 (de) Anthrapyridon-verbindungen, ihre herstellung und ihre verwendung.
DE3578418D1 (de) Chinonderivate, ihre herstellung und verwendung.
DE3777366D1 (de) 2,3-dihydro-cumaron-derivate, ihre herstellung und verwendung.
DE3780329D1 (de) Chinoloncarbonsaeure-derivate und ihre herstellung.
DE3885534D1 (de) Arylphosphorderivate, ihre Herstellung und Verwendung.
DE3587366D1 (de) Benzimidazol-derivate, ihre herstellung und verwendung.
DE3765682D1 (de) Thiolactam-n-essigsaeure-derivate, ihre herstellung und verwendung.
DE69008454D1 (de) Nitrolsothiolderivate, ihre Herstellung und Verwendung.
DE3879024D1 (de) Pyridinium-derivate, ihre herstellung und verwendung.
DE3777604D1 (de) Makrolid-verbindungen, ihre herstellung und ihre verwendung.
DE3688477D1 (de) Antibakterielle verbindungen, ihre herstellung und verwendung.
ATE73762T1 (de) N-aminobutyl-n-phenylarylamid-derivate, ihre herstellung und ihre verwendung in der heilkunde.
DE3784602D1 (de) Inonos-derivate, ihre herstellung und verwendung.
DE3773722D1 (de) Inosose-derivate und ihre herstellung.
DE3770020D1 (de) Sulfoxidderivate und ihre herstellung.
DE3774718D1 (de) Benzothiazolylazolidine und ihre herstellung und verwendung.
DE3883297D1 (de) Phenolderivate, ihre herstellung und verwendung.
DE3863191D1 (de) Substituierte aminderivate, ihre herstellung und verwendung.
DE68908389D1 (de) Amidofluoroverbindungen, ihre herstellung und ihre verwendung.
DE3879328D1 (de) Stannosilikate, ihre herstellung und verwendung.
DE3770299D1 (de) 1,2,4-triazinonderivate, ihre herstellung und verwendung.
DE3886225D1 (de) Pyruvat-Oxidase, ihre Herstellung und Verwendung.
DE3671033D1 (de) Monoazofarbstoffe, ihre herstellung und verwendung.
DE3686632D1 (de) Antibiotische derivate, ihre herstellung und verwendung.

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee