DE3536669A1 - Zusammensetzung fuer die perkutane verabreichung von medikamenten und verfahren zur foerderung der perkutanen absorption von medikamenten - Google Patents
Zusammensetzung fuer die perkutane verabreichung von medikamenten und verfahren zur foerderung der perkutanen absorption von medikamentenInfo
- Publication number
- DE3536669A1 DE3536669A1 DE19853536669 DE3536669A DE3536669A1 DE 3536669 A1 DE3536669 A1 DE 3536669A1 DE 19853536669 DE19853536669 DE 19853536669 DE 3536669 A DE3536669 A DE 3536669A DE 3536669 A1 DE3536669 A1 DE 3536669A1
- Authority
- DE
- Germany
- Prior art keywords
- ester
- pca
- carbon atoms
- composition according
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP59226279A JPS61103840A (ja) | 1984-10-26 | 1984-10-26 | 外皮投与用組成物 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE3536669A1 true DE3536669A1 (de) | 1986-04-30 |
Family
ID=16842717
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19853536669 Withdrawn DE3536669A1 (de) | 1984-10-26 | 1985-10-15 | Zusammensetzung fuer die perkutane verabreichung von medikamenten und verfahren zur foerderung der perkutanen absorption von medikamenten |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US4863952A (enExample) |
| JP (1) | JPS61103840A (enExample) |
| DE (1) | DE3536669A1 (enExample) |
Cited By (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0173990A3 (en) * | 1984-09-03 | 1987-05-13 | Teijin Limited | External pharmaceutical composition |
| EP0227531A3 (en) * | 1985-11-29 | 1987-09-16 | Merck & Co. Inc. | Pyroglutamic acid esters used as dermal penetration enhancers for drugs |
| EP0247507A3 (en) * | 1986-05-27 | 1988-02-10 | Hoechst Aktiengesellschaft | Composition for transdermal therapeutical systems of high-ceiling diuretics, and process for producing it |
| EP0260452A1 (en) * | 1986-08-18 | 1988-03-23 | Chugai Seiyaku Kabushiki Kaisha | Pharmaceutical preparation for the transdermal administration of Nicorandil |
| EP0309624A1 (en) * | 1986-03-27 | 1989-04-05 | Nitto Denko Corporation | Composition for enhancing percutaneous administration of medicine |
| EP0342056A3 (en) * | 1988-05-13 | 1990-04-18 | Unilever Plc | Cosmetic composition |
| EP0374218A4 (en) * | 1988-04-08 | 1991-09-11 | Whitby Research Incorporated | Novel transdermal penetration enhancers |
| US5059628A (en) * | 1987-09-28 | 1991-10-22 | Nitto Electric Industrial Co., Ltd. | Medical composition for percutaneous administration |
| WO2007109152A3 (en) * | 2006-03-17 | 2008-01-24 | Croda Inc | Amine/amide-functionalized lipophiles |
| EP1974715A1 (de) * | 2007-03-31 | 2008-10-01 | Zschimmer & Schwarz GmbH & Co KG Chemische Fabriken | Tränklösung für Feuchttücher |
| EP2335480A1 (en) * | 2009-12-15 | 2011-06-22 | Cognis IP Management GmbH | Biocide compositions comprising derivatives of pyroglutamic acid |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS62187415A (ja) * | 1986-02-12 | 1987-08-15 | Lion Corp | 経皮吸収促進用組成物 |
| JPH03232817A (ja) * | 1990-02-07 | 1991-10-16 | Showa Yakuhin Kako Kk | 貼付剤 |
| JP3686434B2 (ja) * | 1993-10-01 | 2005-08-24 | 千寿製薬株式会社 | コンタクトレンズ用剤の安定化方法 |
| US20040033253A1 (en) * | 2002-02-19 | 2004-02-19 | Ihor Shevchuk | Acyl opioid antagonists |
| CN100525767C (zh) | 2002-06-10 | 2009-08-12 | 欧洲凯尔特公司 | 防止所含活性剂被误用的经皮给药器的处置系统 |
| US20040126323A1 (en) * | 2002-08-20 | 2004-07-01 | Ihor Shevchuk | Transdermal dosage form comprising an active agent and a salt and free-base form of an adverse agent |
| US20080020028A1 (en) * | 2003-08-20 | 2008-01-24 | Euro-Celtique S.A. | Transdermal dosage form comprising an active agent and a salt and a free-base form of an adverse agent |
| US20090156565A1 (en) * | 2004-12-03 | 2009-06-18 | The Children's Hospital Of Philadelphia | Composition and use thereof in enhancing a therapeutic effect of an antiepileptic drug |
| FR2908982A1 (fr) * | 2006-11-23 | 2008-05-30 | Oreal | Composition cosmetique comprenant au moins un solvant volatil hydrocarbone aprotique |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2102172A1 (de) * | 1971-01-18 | 1972-07-27 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue Mitel zur Behandlung und Pflege der Haut |
| DE2102173A1 (en) * | 1971-01-18 | 1972-08-17 | Dr. Karl Thomae Gmbh, 7950 Biberach | Pyrrolidone carboxylic acid alkyl esters prepn - having therapeutic and cosmetic activity esp for the skin |
| US3920814A (en) * | 1972-08-18 | 1975-11-18 | Dominique Bocher | Antibiotic composition containing an antibiotic and as a potentiating agent pyrrolidone carboxylic acid or derivative thereof |
| DE2456634A1 (de) * | 1974-11-29 | 1976-08-12 | Thomae Gmbh Dr K | 5-pyrrolidon-(2)-carbonsaeure-phenylalkanolester und deren herstellung, |
| DE2707814A1 (de) * | 1976-02-26 | 1977-09-01 | Unilever Nv | Mittel zur pflege und behandlung der haut und verfahren zur herstellung der mittel |
| EP0123948A1 (en) * | 1983-04-04 | 1984-11-07 | Teijin Limited | External pharmaceutical composition |
| EP0173990A2 (en) * | 1984-09-03 | 1986-03-12 | Teijin Limited | External pharmaceutical composition |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3975399A (en) * | 1974-08-06 | 1976-08-17 | E. I. Du Pont De Nemours And Company | 1,5-Disubstituted-2-pyrrolidinones, -3-pyrrolin-2-ones, and -4-pyrrolin-2-ones |
| GB1563199A (en) * | 1975-09-10 | 1980-03-19 | Ici Ltd | 1,2,4 triazole compounds and their use as pesticides |
| US4428883A (en) * | 1981-03-06 | 1984-01-31 | The University Of Kentucky Research Foundation | Novel method of administering β-blockers and novel dosage forms containing same |
-
1984
- 1984-10-26 JP JP59226279A patent/JPS61103840A/ja active Granted
-
1985
- 1985-10-04 US US06/784,303 patent/US4863952A/en not_active Expired - Lifetime
- 1985-10-15 DE DE19853536669 patent/DE3536669A1/de not_active Withdrawn
Patent Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2102172A1 (de) * | 1971-01-18 | 1972-07-27 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue Mitel zur Behandlung und Pflege der Haut |
| DE2102173A1 (en) * | 1971-01-18 | 1972-08-17 | Dr. Karl Thomae Gmbh, 7950 Biberach | Pyrrolidone carboxylic acid alkyl esters prepn - having therapeutic and cosmetic activity esp for the skin |
| US3920814A (en) * | 1972-08-18 | 1975-11-18 | Dominique Bocher | Antibiotic composition containing an antibiotic and as a potentiating agent pyrrolidone carboxylic acid or derivative thereof |
| DE2456634A1 (de) * | 1974-11-29 | 1976-08-12 | Thomae Gmbh Dr K | 5-pyrrolidon-(2)-carbonsaeure-phenylalkanolester und deren herstellung, |
| DE2707814A1 (de) * | 1976-02-26 | 1977-09-01 | Unilever Nv | Mittel zur pflege und behandlung der haut und verfahren zur herstellung der mittel |
| EP0123948A1 (en) * | 1983-04-04 | 1984-11-07 | Teijin Limited | External pharmaceutical composition |
| EP0173990A2 (en) * | 1984-09-03 | 1986-03-12 | Teijin Limited | External pharmaceutical composition |
Cited By (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0173990A3 (en) * | 1984-09-03 | 1987-05-13 | Teijin Limited | External pharmaceutical composition |
| EP0227531A3 (en) * | 1985-11-29 | 1987-09-16 | Merck & Co. Inc. | Pyroglutamic acid esters used as dermal penetration enhancers for drugs |
| EP0309624A1 (en) * | 1986-03-27 | 1989-04-05 | Nitto Denko Corporation | Composition for enhancing percutaneous administration of medicine |
| EP0247507A3 (en) * | 1986-05-27 | 1988-02-10 | Hoechst Aktiengesellschaft | Composition for transdermal therapeutical systems of high-ceiling diuretics, and process for producing it |
| EP0260452A1 (en) * | 1986-08-18 | 1988-03-23 | Chugai Seiyaku Kabushiki Kaisha | Pharmaceutical preparation for the transdermal administration of Nicorandil |
| BE1000477A3 (fr) * | 1986-08-18 | 1988-12-20 | Chugai Pharmaceutical Co Ltd | Compositions pharmaceutiques pour l'administration par absorption percutanee et procede pour les preparer. |
| US5211943A (en) * | 1986-08-18 | 1993-05-18 | Chugai Seiyaku Kabushili Kaisha | Pharmaceutical preparation for administration by percutaneous absorption and a method for their manufacture |
| US5059628A (en) * | 1987-09-28 | 1991-10-22 | Nitto Electric Industrial Co., Ltd. | Medical composition for percutaneous administration |
| EP0374218A4 (en) * | 1988-04-08 | 1991-09-11 | Whitby Research Incorporated | Novel transdermal penetration enhancers |
| EP0342056A3 (en) * | 1988-05-13 | 1990-04-18 | Unilever Plc | Cosmetic composition |
| WO2007109152A3 (en) * | 2006-03-17 | 2008-01-24 | Croda Inc | Amine/amide-functionalized lipophiles |
| US7781391B2 (en) | 2006-03-17 | 2010-08-24 | Croda, Inc. | Amine/amide-functionalized lipophiles |
| EP1974715A1 (de) * | 2007-03-31 | 2008-10-01 | Zschimmer & Schwarz GmbH & Co KG Chemische Fabriken | Tränklösung für Feuchttücher |
| EP2335480A1 (en) * | 2009-12-15 | 2011-06-22 | Cognis IP Management GmbH | Biocide compositions comprising derivatives of pyroglutamic acid |
| WO2011072811A3 (en) * | 2009-12-15 | 2012-03-29 | Cognis Ip Management Gmbh | Biocide compositions comprising derivatives of pyroglutamic acid |
| US8927460B2 (en) | 2009-12-15 | 2015-01-06 | Cognis Ip Management Gmbh | Biocide compositions comprising derivatives of pyroglutamic acid |
Also Published As
| Publication number | Publication date |
|---|---|
| JPS61103840A (ja) | 1986-05-22 |
| US4863952A (en) | 1989-09-05 |
| JPH0570610B2 (enExample) | 1993-10-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8110 | Request for examination paragraph 44 | ||
| 8125 | Change of the main classification |
Ipc: A61K 47/18 |
|
| 8130 | Withdrawal |