DE10304374A1 - Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament - Google Patents
Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament Download PDFInfo
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- DE10304374A1 DE10304374A1 DE10304374A DE10304374A DE10304374A1 DE 10304374 A1 DE10304374 A1 DE 10304374A1 DE 10304374 A DE10304374 A DE 10304374A DE 10304374 A DE10304374 A DE 10304374A DE 10304374 A1 DE10304374 A1 DE 10304374A1
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Obesity (AREA)
- Psychiatry (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Toxicology (AREA)
- Anesthesiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Vascular Medicine (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (18)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10304374A DE10304374A1 (de) | 2003-02-04 | 2003-02-04 | Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| MXPA05007968A MXPA05007968A (es) | 2003-02-04 | 2004-01-20 | Nuevos 2-aminoimidazoles sustituidos, procedimiento para su preparacion, su uso como medicamento o ayuda al diagnostico, y medicamento que los contiene. |
| AT04703371T ATE375982T1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie diese enthaltendes medikament |
| DE502004005260T DE502004005260D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie diese enthaltendes medikament |
| DE502004009771T DE502004009771D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| EP07014956A EP1857445B1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| EP04703371A EP1592669B1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie diese enthaltendes medikament |
| JP2006501561A JP4630269B2 (ja) | 2003-02-04 | 2004-01-20 | 新規な置換された２−アミノイミダゾール、その製造方法、その医薬または診断薬としての使用、および、その化合物を含有する医薬品 |
| BR0407212-0A BRPI0407212A (pt) | 2003-02-04 | 2004-01-20 | 2-aminoimidazóis substituìdos, processos para a sua preparação, sua aplicação como medicamento ou diagnóstico bem como o medicamento contendo os mesmos |
| CA002514028A CA2514028A1 (en) | 2003-02-04 | 2004-01-20 | Substituted 2-aminoimidazoles, method for the production thereof, their use as a medicament or as a diagnostic reagent, and medicament containing these compounds |
| PCT/EP2004/000394 WO2004069806A2 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie sie enthaltendes medikament |
| AU2004208870A AU2004208870A1 (en) | 2003-02-04 | 2004-01-20 | Substituted 2-aminoimidazoles, method for the production thereof, their use as a medicament or as a diagnostic reagent, and medicament containing these compounds |
| PE2004000108A PE20040943A1 (es) | 2003-02-04 | 2004-01-28 | 2-AMINOIMIDAZOLES SUSTITUIDOS COMO INHIBIDORES DEL INTERCAMBIADOR Na/H SUBTIPO 3 (NHE 3) |
| ARP040100314A AR049671A1 (es) | 2003-02-04 | 2004-02-02 | 2-aminoimidazoles sustituidos, procedimiento para su preparacion, su uso como medicamento o ayuda al diagnostico, y medicamento que los contiene |
| TW093102254A TW200508206A (en) | 2003-02-04 | 2004-02-02 | Novel substituted 2-aminoimidazoles, process for their preparation, their use as medicament or diagnostic aid, and medicament containing them |
| US10/771,185 US7442717B2 (en) | 2003-02-04 | 2004-02-03 | Substituted 2-aminoimidazoles, process for their preparation, their use as medicament or diagnostic aid |
| US12/172,380 US20080275098A1 (en) | 2003-02-04 | 2008-07-14 | Novel substituted 2-aminoimidazoles, process for their preparation, their use as medicament or diagnostic aid |
| JP2010196422A JP2011016825A (ja) | 2003-02-04 | 2010-09-02 | 新規な置換された２−アミノイミダゾール、その製造方法、その医薬または診断薬としての使用、および、その化合物を含有する医薬品 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10304374A DE10304374A1 (de) | 2003-02-04 | 2003-02-04 | Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE10304374A1 true DE10304374A1 (de) | 2004-08-05 |
Family
ID=32667986
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE10304374A Withdrawn DE10304374A1 (de) | 2003-02-04 | 2003-02-04 | Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| DE502004005260T Expired - Lifetime DE502004005260D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie diese enthaltendes medikament |
| DE502004009771T Expired - Lifetime DE502004009771D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE502004005260T Expired - Lifetime DE502004005260D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-aminoimidazole, verfahren zu ihrer herstellung, ihre verwendung als medikament oder diagnostikum sowie diese enthaltendes medikament |
| DE502004009771T Expired - Lifetime DE502004009771D1 (de) | 2003-02-04 | 2004-01-20 | Substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US7442717B2 (https=) |
| EP (2) | EP1592669B1 (https=) |
| JP (2) | JP4630269B2 (https=) |
| AR (1) | AR049671A1 (https=) |
| AT (1) | ATE375982T1 (https=) |
| AU (1) | AU2004208870A1 (https=) |
| BR (1) | BRPI0407212A (https=) |
| CA (1) | CA2514028A1 (https=) |
| DE (3) | DE10304374A1 (https=) |
| MX (1) | MXPA05007968A (https=) |
| PE (1) | PE20040943A1 (https=) |
| TW (1) | TW200508206A (https=) |
| WO (1) | WO2004069806A2 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007083207A1 (en) * | 2006-01-19 | 2007-07-26 | Pfizer Limited | Substituted imidazoles and their use as pesticides |
| CN109422695A (zh) * | 2017-08-28 | 2019-03-05 | 扬子江药业集团有限公司 | 一种盐酸苯达莫司汀粗品的制备方法 |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050054705A1 (en) * | 2003-02-04 | 2005-03-10 | Aventis Pharma Deutschland Gmbh | N-substituted (benzoimidazol-2-yl) phenylamines, process for their preparation, their use as medicament or diagnostic aid, and medicament comprising them |
| WO2005107470A2 (en) * | 2004-04-29 | 2005-11-17 | University Of Florida Research Foundation, Inc. | Use of carbonic anhydrase inhibitors for insect control and malaria treatment |
| US20120088737A2 (en) * | 2009-10-02 | 2012-04-12 | Ajinomoto Co., Inc | Novel acyl guanidine derivatives |
| ME03311B (me) | 2014-07-25 | 2019-10-20 | Taisho Pharmaceutical Co Ltd | Fenil teтrahidroizokvinolinsko jedinjenje supsтituisano heteroarilom |
| CN118619883B (zh) * | 2024-05-24 | 2025-11-11 | 河北圣泰材料股份有限公司 | 一种4,5-二氰基-2-三氟甲基咪唑锂的制备方法 |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4275072A (en) * | 1978-08-16 | 1981-06-23 | Farmos Group, Ltd. | 2,6-Dichlorophenyl-substituted amino-imidazole derivatives and use as hypertensive agents |
| EP0254259A2 (en) * | 1986-07-21 | 1988-01-27 | Otsuka Pharmaceutical Factory, Inc. | p-Aminophenol derivatives |
| WO1990014338A1 (en) * | 1989-05-20 | 1990-11-29 | Fisons Plc | Anti-inflammatory 4-aminophenol derivatives |
| WO1995019968A1 (en) * | 1994-01-24 | 1995-07-27 | Allergan | Aromatic 2-amino-imidazole derivatives as alpha-2a adrenoceptor agonists |
| WO2001021160A2 (en) * | 1999-09-23 | 2001-03-29 | Axxima Pharmaceuticals Aktiengesellschaft | Carboxymide and aniline derivatives as selective inhibitors of pathogens |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3459763A (en) | 1966-01-25 | 1969-08-05 | Geigy Chem Corp | Certain amino imidazole derivatives |
| JPS5547663A (en) * | 1978-08-16 | 1980-04-04 | Farmos Oy | 2*66dichlorophenyl substituted aminoo imidazole derivative*its acid addition salt* their manufacture and therapy of mammal using them |
| DE19633966A1 (de) * | 1996-08-22 | 1998-02-26 | Hoechst Ag | Phenylsubstituierte Alkenylcarbonsäure-guanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| DE19945302A1 (de) | 1999-09-22 | 2001-03-29 | Merck Patent Gmbh | Biphenylderivate als NHE-3-Inhibitoren |
| DE19960204A1 (de) * | 1999-12-14 | 2001-06-28 | Aventis Pharma Gmbh | Substituierte Norlbornylamino-Derivate, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| DE10015248A1 (de) | 2000-03-28 | 2001-10-04 | Merck Patent Gmbh | Bisamidino-Verbindungen als NHE-3 Inhibitoren |
| DE10019062A1 (de) | 2000-04-18 | 2001-10-25 | Merck Patent Gmbh | 2-Guanidino-4-aryl-chinazoline als NHE-3 Inhibitoren |
| DE10043667A1 (de) | 2000-09-05 | 2002-03-14 | Merck Patent Gmbh | 2-Guanidino-4-aryl-chinazoline |
| EP1578341A2 (en) * | 2000-10-11 | 2005-09-28 | Tularik Inc. | Modulation of ccr4 function |
| DE10060292A1 (de) * | 2000-12-05 | 2002-06-20 | Aventis Pharma Gmbh | Verwendung substituierter Benzimidazole zur Herstellung eines Medikaments zur Behandlung von Krankheiten, welche durch Inhibierung des Na+/H+-Austauschers beeinflusst werden können und sie enthaltendes Medikament |
| US20030187045A1 (en) * | 2001-12-21 | 2003-10-02 | Uwe Heinelt | Substituted imidazolidines, process for their preparation, and their use as a medicament or diagnostic |
| US7049333B2 (en) * | 2002-06-04 | 2006-05-23 | Sanofi-Aventis Deutschland Gmbh | Substituted thiophenes: compositions, processes of making, and uses in disease treatment and diagnosis |
-
2003
- 2003-02-04 DE DE10304374A patent/DE10304374A1/de not_active Withdrawn
-
2004
- 2004-01-20 JP JP2006501561A patent/JP4630269B2/ja not_active Expired - Fee Related
- 2004-01-20 AT AT04703371T patent/ATE375982T1/de not_active IP Right Cessation
- 2004-01-20 MX MXPA05007968A patent/MXPA05007968A/es unknown
- 2004-01-20 EP EP04703371A patent/EP1592669B1/de not_active Expired - Lifetime
- 2004-01-20 EP EP07014956A patent/EP1857445B1/de not_active Expired - Lifetime
- 2004-01-20 DE DE502004005260T patent/DE502004005260D1/de not_active Expired - Lifetime
- 2004-01-20 CA CA002514028A patent/CA2514028A1/en not_active Abandoned
- 2004-01-20 DE DE502004009771T patent/DE502004009771D1/de not_active Expired - Lifetime
- 2004-01-20 BR BR0407212-0A patent/BRPI0407212A/pt not_active IP Right Cessation
- 2004-01-20 WO PCT/EP2004/000394 patent/WO2004069806A2/de not_active Ceased
- 2004-01-20 AU AU2004208870A patent/AU2004208870A1/en not_active Abandoned
- 2004-01-28 PE PE2004000108A patent/PE20040943A1/es not_active Application Discontinuation
- 2004-02-02 TW TW093102254A patent/TW200508206A/zh unknown
- 2004-02-02 AR ARP040100314A patent/AR049671A1/es unknown
- 2004-02-03 US US10/771,185 patent/US7442717B2/en not_active Expired - Fee Related
-
2008
- 2008-07-14 US US12/172,380 patent/US20080275098A1/en not_active Abandoned
-
2010
- 2010-09-02 JP JP2010196422A patent/JP2011016825A/ja not_active Abandoned
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4275072A (en) * | 1978-08-16 | 1981-06-23 | Farmos Group, Ltd. | 2,6-Dichlorophenyl-substituted amino-imidazole derivatives and use as hypertensive agents |
| EP0254259A2 (en) * | 1986-07-21 | 1988-01-27 | Otsuka Pharmaceutical Factory, Inc. | p-Aminophenol derivatives |
| WO1990014338A1 (en) * | 1989-05-20 | 1990-11-29 | Fisons Plc | Anti-inflammatory 4-aminophenol derivatives |
| WO1995019968A1 (en) * | 1994-01-24 | 1995-07-27 | Allergan | Aromatic 2-amino-imidazole derivatives as alpha-2a adrenoceptor agonists |
| WO2001021160A2 (en) * | 1999-09-23 | 2001-03-29 | Axxima Pharmaceuticals Aktiengesellschaft | Carboxymide and aniline derivatives as selective inhibitors of pathogens |
Cited By (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2007083207A1 (en) * | 2006-01-19 | 2007-07-26 | Pfizer Limited | Substituted imidazoles and their use as pesticides |
| US7544706B2 (en) | 2006-01-19 | 2009-06-09 | Pfizer Limited | Substituted imidazoles |
| US7547718B2 (en) | 2006-01-19 | 2009-06-16 | Pfizer Limited | Substituted imidazoles |
| US7592362B2 (en) | 2006-01-19 | 2009-09-22 | Pfizer Limited | Substituted imidazoles |
| US7825149B2 (en) | 2006-01-19 | 2010-11-02 | Pfizer Limited | Substituted imidazoles |
| EA015738B1 (ru) * | 2006-01-19 | 2011-10-31 | Пфайзер Лимитед | Замещенные имидазолы и их применение в качестве пестицидов |
| EP2423199A1 (en) * | 2006-01-19 | 2012-02-29 | Pfizer Limited | Substituted imidazoles and their use as pesticides |
| NO341141B1 (no) * | 2006-01-19 | 2017-08-28 | Zoetis Uk Ltd | Substituerte imidazoler og deres anvendelse som pesticider |
| CN109422695A (zh) * | 2017-08-28 | 2019-03-05 | 扬子江药业集团有限公司 | 一种盐酸苯达莫司汀粗品的制备方法 |
| CN109422695B (zh) * | 2017-08-28 | 2022-03-18 | 扬子江药业集团有限公司 | 一种盐酸苯达莫司汀粗品的制备方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004208870A1 (en) | 2004-08-19 |
| CA2514028A1 (en) | 2004-08-19 |
| WO2004069806A2 (de) | 2004-08-19 |
| WO2004069806A3 (de) | 2004-10-28 |
| MXPA05007968A (es) | 2005-09-20 |
| EP1857445A3 (de) | 2007-12-19 |
| ATE375982T1 (de) | 2007-11-15 |
| EP1857445A2 (de) | 2007-11-21 |
| TW200508206A (en) | 2005-03-01 |
| JP2006516576A (ja) | 2006-07-06 |
| EP1592669B1 (de) | 2007-10-17 |
| US20080275098A1 (en) | 2008-11-06 |
| DE502004009771D1 (de) | 2009-08-27 |
| US20040259927A1 (en) | 2004-12-23 |
| BRPI0407212A (pt) | 2006-01-24 |
| PE20040943A1 (es) | 2005-02-07 |
| DE502004005260D1 (de) | 2007-11-29 |
| EP1592669A2 (de) | 2005-11-09 |
| US7442717B2 (en) | 2008-10-28 |
| JP4630269B2 (ja) | 2011-02-09 |
| AR049671A1 (es) | 2006-08-30 |
| EP1857445B1 (de) | 2009-07-15 |
| JP2011016825A (ja) | 2011-01-27 |
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