DD211342A5 - Verfahren zur herstellung polymorpher formen von 5-[3-(2-[2,2,2-trifluor-ethyl] guanidino)pyrazol-1-yl] valeramid - Google Patents

Verfahren zur herstellung polymorpher formen von 5-[3-(2-[2,2,2-trifluor-ethyl] guanidino)pyrazol-1-yl] valeramid Download PDF

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Publication number
DD211342A5
DD211342A5 DD83254489A DD25448983A DD211342A5 DD 211342 A5 DD211342 A5 DD 211342A5 DD 83254489 A DD83254489 A DD 83254489A DD 25448983 A DD25448983 A DD 25448983A DD 211342 A5 DD211342 A5 DD 211342A5
Authority
DD
German Democratic Republic
Prior art keywords
polymorph
ici
solution
starting material
mixture
Prior art date
Application number
DD83254489A
Other languages
German (de)
English (en)
Inventor
Janet Hardie
Ronald Platt
Jonathan Hutton
Peter Warren
Stanley A Lee
Gregory D Harris
Elwyn P Davies
Original Assignee
Ici Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Plc filed Critical Ici Plc
Publication of DD211342A5 publication Critical patent/DD211342A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DD83254489A 1982-09-03 1983-09-02 Verfahren zur herstellung polymorpher formen von 5-[3-(2-[2,2,2-trifluor-ethyl] guanidino)pyrazol-1-yl] valeramid DD211342A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8225154 1982-09-03

Publications (1)

Publication Number Publication Date
DD211342A5 true DD211342A5 (de) 1984-07-11

Family

ID=10532675

Family Applications (1)

Application Number Title Priority Date Filing Date
DD83254489A DD211342A5 (de) 1982-09-03 1983-09-02 Verfahren zur herstellung polymorpher formen von 5-[3-(2-[2,2,2-trifluor-ethyl] guanidino)pyrazol-1-yl] valeramid

Country Status (21)

Country Link
EP (1) EP0115114B1 (fr)
JP (1) JPS5965079A (fr)
AT (1) ATE20740T1 (fr)
AU (1) AU1789783A (fr)
CA (1) CA1198734A (fr)
CS (1) CS236893B2 (fr)
DD (1) DD211342A5 (fr)
DE (1) DE3364524D1 (fr)
DK (1) DK380083D0 (fr)
ES (1) ES525329A0 (fr)
FI (1) FI833074A (fr)
GB (1) GB8320820D0 (fr)
GR (1) GR78940B (fr)
HU (1) HU191091B (fr)
IE (1) IE55805B1 (fr)
IL (1) IL69533A (fr)
NO (1) NO833147L (fr)
NZ (1) NZ205451A (fr)
PT (1) PT77278B (fr)
SU (1) SU1237080A3 (fr)
ZA (1) ZA836196B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8401751D0 (en) * 1984-01-24 1984-02-29 Ici Plc Guanidine derivatives

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1233818A (fr) * 1981-03-09 1988-03-08 David J. Gilman Derives de la guanidine, inhibiteurs des recepteurs h.sub.2 a l'histamine

Also Published As

Publication number Publication date
ES8505738A1 (es) 1985-06-01
AU1789783A (en) 1984-03-08
PT77278A (en) 1983-10-01
ZA836196B (en) 1984-07-25
EP0115114B1 (fr) 1986-07-16
NZ205451A (en) 1985-07-31
NO833147L (no) 1984-03-05
DE3364524D1 (en) 1986-08-21
DK380083D0 (da) 1983-08-19
CA1198734A (fr) 1985-12-31
CS236893B2 (en) 1985-05-15
PT77278B (en) 1986-03-18
SU1237080A3 (ru) 1986-06-07
FI833074A0 (fi) 1983-08-30
GB8320820D0 (en) 1983-09-01
JPS5965079A (ja) 1984-04-13
FI833074A (fi) 1984-03-04
ATE20740T1 (de) 1986-08-15
EP0115114A1 (fr) 1984-08-08
IL69533A (en) 1987-12-31
IE831874L (en) 1984-03-03
IE55805B1 (en) 1991-01-16
HU191091B (en) 1987-01-28
GR78940B (fr) 1984-10-02
ES525329A0 (es) 1985-06-01

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