CZ20031403A3 - Inhibitor proteasy - Google Patents

Inhibitor proteasy Download PDF

Info

Publication number
CZ20031403A3
CZ20031403A3 CZ20031403A CZ20031403A CZ20031403A3 CZ 20031403 A3 CZ20031403 A3 CZ 20031403A3 CZ 20031403 A CZ20031403 A CZ 20031403A CZ 20031403 A CZ20031403 A CZ 20031403A CZ 20031403 A3 CZ20031403 A3 CZ 20031403A3
Authority
CZ
Czechia
Prior art keywords
alkyl
carbon atoms
group
substituted
moiety
Prior art date
Application number
CZ20031403A
Other languages
Czech (cs)
English (en)
Inventor
Dennis S. Yamashita
Daniel F. Veber
Robert W. Marquis
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of CZ20031403A3 publication Critical patent/CZ20031403A3/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CZ20031403A 2000-11-22 2001-11-19 Inhibitor proteasy CZ20031403A3 (cs)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25250800P 2000-11-22 2000-11-22

Publications (1)

Publication Number Publication Date
CZ20031403A3 true CZ20031403A3 (cs) 2003-10-15

Family

ID=22956303

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ20031403A CZ20031403A3 (cs) 2000-11-22 2001-11-19 Inhibitor proteasy

Country Status (17)

Country Link
EP (1) EP1392657A4 (pt)
JP (1) JP2005513083A (pt)
KR (1) KR20040004445A (pt)
CN (1) CN1635903A (pt)
AR (1) AR034278A1 (pt)
AU (1) AU2001298052A1 (pt)
BR (1) BR0115473A (pt)
CA (1) CA2436850A1 (pt)
CZ (1) CZ20031403A3 (pt)
HU (1) HUP0301964A3 (pt)
IL (1) IL155997A0 (pt)
MX (1) MXPA03004542A (pt)
NO (1) NO20032328L (pt)
PL (1) PL366232A1 (pt)
UY (1) UY27032A1 (pt)
WO (1) WO2003053331A2 (pt)
ZA (1) ZA200303848B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030144175A1 (en) 1998-12-23 2003-07-31 Smithkline Beecham Corporation Protease inhibitors
US7071184B2 (en) 2000-03-21 2006-07-04 Smithkline Beecham Corporation Protease inhibitors
AU2001268407A1 (en) * 2000-06-14 2001-12-24 Smithkline Beecham Corporation Protease inhibitors
JPWO2008149971A1 (ja) 2007-06-08 2010-08-26 日本ケミファ株式会社 脳動脈瘤の治療または予防薬
JPWO2009054454A1 (ja) 2007-10-24 2011-03-03 国立大学法人 東京医科歯科大学 カテプシン阻害剤を有効成分として含有するToll様受容体のシグナル伝達の調整剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200101869T2 (tr) * 1998-12-23 2002-01-21 Smithkline Beecham Corporation Proteaz İnhibitörleri.
US7071184B2 (en) * 2000-03-21 2006-07-04 Smithkline Beecham Corporation Protease inhibitors
AU2001268407A1 (en) * 2000-06-14 2001-12-24 Smithkline Beecham Corporation Protease inhibitors

Also Published As

Publication number Publication date
AR034278A1 (es) 2004-02-18
UY27032A1 (es) 2002-07-31
KR20040004445A (ko) 2004-01-13
IL155997A0 (en) 2003-12-23
JP2005513083A (ja) 2005-05-12
MXPA03004542A (es) 2003-09-10
AU2001298052A1 (en) 2003-07-09
NO20032328L (no) 2003-07-02
PL366232A1 (en) 2005-01-24
WO2003053331A2 (en) 2003-07-03
ZA200303848B (en) 2004-06-28
NO20032328D0 (no) 2003-05-22
HUP0301964A2 (en) 2007-02-28
CN1635903A (zh) 2005-07-06
EP1392657A4 (en) 2004-03-10
HUP0301964A3 (en) 2007-09-28
EP1392657A2 (en) 2004-03-03
CA2436850A1 (en) 2003-07-03
WO2003053331A3 (en) 2003-11-13
BR0115473A (pt) 2004-09-28

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