CY1116664T1 - Χρηση ενος ινδαζολο-μεθοξυ-αλκανοϊκου οξεος για την παρασκευη μιας φαρμακευτικης συνθεσης - Google Patents

Χρηση ενος ινδαζολο-μεθοξυ-αλκανοϊκου οξεος για την παρασκευη μιας φαρμακευτικης συνθεσης

Info

Publication number
CY1116664T1
CY1116664T1 CY20151100184T CY151100184T CY1116664T1 CY 1116664 T1 CY1116664 T1 CY 1116664T1 CY 20151100184 T CY20151100184 T CY 20151100184T CY 151100184 T CY151100184 T CY 151100184T CY 1116664 T1 CY1116664 T1 CY 1116664T1
Authority
CY
Cyprus
Prior art keywords
preparation
pharmaceutical composition
alcohanic
indasol
methoxy
Prior art date
Application number
CY20151100184T
Other languages
Greek (el)
English (en)
Inventor
Angelo Guglielmotti
Giuseppe Biondi
Original Assignee
Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A. filed Critical Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A.
Publication of CY1116664T1 publication Critical patent/CY1116664T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/4161,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Mixers Of The Rotary Stirring Type (AREA)
CY20151100184T 2006-11-24 2015-02-20 Χρηση ενος ινδαζολο-μεθοξυ-αλκανοϊκου οξεος για την παρασκευη μιας φαρμακευτικης συνθεσης CY1116664T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT002254A ITMI20062254A1 (it) 2006-11-24 2006-11-24 Uso di un acido metossi-alcanoico dell'indazolo per preparare una composizione farmaceutca
EP11185914.6A EP2409698B1 (en) 2006-11-24 2007-11-13 Use of an indazolemethoxyalkanoic acid to prepare a pharmaceutical composition

Publications (1)

Publication Number Publication Date
CY1116664T1 true CY1116664T1 (el) 2017-03-15

Family

ID=38198404

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20151100184T CY1116664T1 (el) 2006-11-24 2015-02-20 Χρηση ενος ινδαζολο-μεθοξυ-αλκανοϊκου οξεος για την παρασκευη μιας φαρμακευτικης συνθεσης

Country Status (23)

Country Link
US (2) US8198310B2 (OSRAM)
EP (2) EP2097080B1 (OSRAM)
JP (1) JP5192490B2 (OSRAM)
KR (1) KR101413616B1 (OSRAM)
CN (1) CN101541323B (OSRAM)
AR (1) AR063894A1 (OSRAM)
AU (1) AU2007323351B2 (OSRAM)
BR (1) BRPI0718522A2 (OSRAM)
CA (1) CA2666371C (OSRAM)
CY (1) CY1116664T1 (OSRAM)
DK (2) DK2409698T3 (OSRAM)
EA (1) EA016885B1 (OSRAM)
ES (2) ES2530623T3 (OSRAM)
GE (1) GEP20125570B (OSRAM)
IL (1) IL198286A (OSRAM)
IT (1) ITMI20062254A1 (OSRAM)
MX (1) MX2009004295A (OSRAM)
PL (2) PL2097080T3 (OSRAM)
PT (2) PT2409698E (OSRAM)
SG (1) SG176508A1 (OSRAM)
SI (2) SI2409698T1 (OSRAM)
UA (1) UA97123C2 (OSRAM)
WO (1) WO2008061671A2 (OSRAM)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20062254A1 (it) 2006-11-24 2008-05-25 Acraf Uso di un acido metossi-alcanoico dell'indazolo per preparare una composizione farmaceutca
US8350052B2 (en) 2009-08-03 2013-01-08 Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A. Process for the preparation of 1-benzyl-3-hydroxymethyl-1H-indazole and its derivatives and required magnesium intermediates
US8999292B2 (en) 2012-05-01 2015-04-07 Translatum Medicus Inc. Methods for treating and diagnosing blinding eye diseases
US20170079955A1 (en) * 2014-05-15 2017-03-23 Shelley Romayne Boyd Compositions and methods for treating and diagnosing ocular disorders
CA3144861A1 (en) 2019-06-25 2020-12-30 Translatum Medicus, Inc. Processes of making 2-((1-benzyl-1h-indazol-3-yl)methoxy)-2-methylpropanoic acid and its derivatives
KR20230031322A (ko) 2020-06-27 2023-03-07 크레센타 바이오사이언시즈 세포 물질대사를 조정하는 화합물의 조성물 및 사용 방법
US12138243B2 (en) 2021-12-31 2024-11-12 Crescenta Biosciences Antiviral use of FABP4 modulating compounds

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1131779B (it) * 1980-07-29 1986-06-25 Acraf Sale dell'acido (1-benzil-1h-indazol-3-il)-ossiacetico con la lisina e procedimento per la sua preparazione
IT1230441B (it) * 1989-02-07 1991-10-23 Acraf Eteri della serie dell'indazolo
IT1253703B (it) * 1991-04-22 1995-08-23 Angelini Francesco Ist Ricerca Uso di acidi metossi alcanoici dell'indazolo per preparare un farmaco attivo nel trattamento di malattie autoimmunitarie
IT1276031B1 (it) * 1995-10-31 1997-10-24 Angelini Ricerche Spa Composizione farmaceutica per il trattamento delle malattie autoimmuni
US6077539A (en) * 1996-11-12 2000-06-20 Pozen, Inc. Treatment of migraine headache
IT1293795B1 (it) * 1997-07-28 1999-03-10 Angelini Ricerche Spa Farmaco attivo nel ridurre la produzione di proteina mcp-1
IT1293794B1 (it) 1997-07-28 1999-03-10 Acraf Farmaco attivo nel ridurre la produzione di proteina mcp-1
US6803357B1 (en) * 1998-02-02 2004-10-12 New England Medical Center Hospitals, Inc. Method of regulating glucose metabolism, and reagents related thereto
DE19821625C1 (de) * 1998-05-15 2000-01-05 Merck Patent Gmbh Pharmazeutische Zubereitung
US6197786B1 (en) * 1998-09-17 2001-03-06 Pfizer Inc 4-Carboxyamino-2-substituted-1,2,3,4-tetrahydroquinolines
ITFI20010230A1 (it) * 2001-11-29 2003-05-29 Menarini Int Operations Lu Sa Composizioni farmaceutiche per il trattamento del diabete mellito di tipo ii
US20060030582A1 (en) * 2002-04-29 2006-02-09 Demartino Julie Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity
AU2006243255A1 (en) * 2005-04-29 2006-11-09 Nycomed Gmbh Mutual prodrug compounds for use us antiinflammatory agents with gastrointestinal protective activity
WO2007062469A1 (en) * 2005-12-01 2007-06-07 Flinders Technologies Pty Ltd Methods and compositions for preventing and/or treating pancreatitis
ITMI20062254A1 (it) 2006-11-24 2008-05-25 Acraf Uso di un acido metossi-alcanoico dell'indazolo per preparare una composizione farmaceutca

Also Published As

Publication number Publication date
IL198286A0 (en) 2010-02-17
WO2008061671A3 (en) 2008-11-27
BRPI0718522A2 (pt) 2013-11-12
HK1165275A1 (en) 2012-10-05
CN101541323A (zh) 2009-09-23
HK1129071A1 (en) 2009-11-20
SG176508A1 (en) 2011-12-29
EA200970506A1 (ru) 2009-10-30
ES2530623T3 (es) 2015-03-04
EA016885B1 (ru) 2012-08-30
AU2007323351B2 (en) 2013-05-02
EP2097080B1 (en) 2013-02-20
EP2409698A1 (en) 2012-01-25
WO2008061671A2 (en) 2008-05-29
KR20090081410A (ko) 2009-07-28
DK2097080T3 (da) 2013-05-21
UA97123C2 (uk) 2012-01-10
IL198286A (en) 2016-03-31
EP2097080A2 (en) 2009-09-09
ES2403584T3 (es) 2013-05-20
AR063894A1 (es) 2009-02-25
US8846745B2 (en) 2014-09-30
JP2010510263A (ja) 2010-04-02
JP5192490B2 (ja) 2013-05-08
EP2409698B1 (en) 2015-01-21
PL2097080T3 (pl) 2013-07-31
AU2007323351A1 (en) 2008-05-29
PT2097080E (pt) 2013-04-01
CA2666371A1 (en) 2008-05-29
US8198310B2 (en) 2012-06-12
CN101541323B (zh) 2012-01-04
CA2666371C (en) 2014-05-06
US20100069456A1 (en) 2010-03-18
PL2409698T3 (pl) 2015-06-30
US20120283307A1 (en) 2012-11-08
ITMI20062254A1 (it) 2008-05-25
KR101413616B1 (ko) 2014-07-01
SI2097080T1 (sl) 2013-05-31
MX2009004295A (es) 2009-05-05
DK2409698T3 (en) 2015-04-27
SI2409698T1 (sl) 2015-04-30
GEP20125570B (en) 2012-07-10
PT2409698E (pt) 2015-02-10

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