CY1113473T1 - ΠΡΟΣΤΑΤΕΥΤΙΚΟΣ ΠΑΡΑΓΩΝ ΓΙΑ ΑΜΦΙΒΛΗΣΤΡΟΕΙΔΙΚΟ ΝΕΥΡΩΝΙΚΟ ΚΥΤΤΑΡΟ ΠΟΥ ΠΕΡΙΕΧΕΙ ΠΑΡΑΓΩΓΟ ΠΡΟΣΤΑΓΛΑΝΔΙΝΗΣ F2α ΩΣ ΔΡΑΣΤΙΚΟ ΣΥΣΤΑΤΙΚΟ - Google Patents
ΠΡΟΣΤΑΤΕΥΤΙΚΟΣ ΠΑΡΑΓΩΝ ΓΙΑ ΑΜΦΙΒΛΗΣΤΡΟΕΙΔΙΚΟ ΝΕΥΡΩΝΙΚΟ ΚΥΤΤΑΡΟ ΠΟΥ ΠΕΡΙΕΧΕΙ ΠΑΡΑΓΩΓΟ ΠΡΟΣΤΑΓΛΑΝΔΙΝΗΣ F2α ΩΣ ΔΡΑΣΤΙΚΟ ΣΥΣΤΑΤΙΚΟInfo
- Publication number
- CY1113473T1 CY1113473T1 CY20121100958T CY121100958T CY1113473T1 CY 1113473 T1 CY1113473 T1 CY 1113473T1 CY 20121100958 T CY20121100958 T CY 20121100958T CY 121100958 T CY121100958 T CY 121100958T CY 1113473 T1 CY1113473 T1 CY 1113473T1
- Authority
- CY
- Cyprus
- Prior art keywords
- prostaglantine
- dilutic
- product
- active ingredient
- cell containing
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Ophthalmology & Optometry (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Ένα αντικείμενο της παρούσας εφεύρεσης είναι να βρεθεί μια νέα φαρμακευτική εφαρμογή για ένα παράγωγο προσταγλανδίνης F2α. Έχει βρεθεί ότι το παράγωγο προσταλανδίνης F2α αναστέλλει τον προκαλούμενο από γλουταμικό θάνατο αμφιβληστροειδικού νευρωνικού κυττάρου με τρόπο που εξαρτάται από την συγκέντρωση σε εμβρυϊκά αμφιβληστροειδικά νευρωνικά κύτταρα αρουραίου, με άλλα λόγια, το παράγωγο προσταγλανδίνης F2α δρα απευθείας επί των αμφιβληστροειδικών νευρωνικών κυττάρων και δεικνύει προστατευτικό αποτέλεσμα. Ακολούθως, το παράγωγο προσταγλανδίνης F2α είναι χρήσιμο για την αποτροπή ή την θεραπεία μιας οφθαλμικής ασθένειας που συνδυάζεται με βλάβη αμφιβληστροειδικού νευρωνικού κυττάρου.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2005100348 | 2005-03-31 | ||
EP06730774A EP1864666B1 (en) | 2005-03-31 | 2006-03-31 | Protective agent for retinal neuronal cell containing prostaglandin f2 alpha derivative as active ingredient |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1113473T1 true CY1113473T1 (el) | 2016-06-22 |
Family
ID=37073466
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20121100958T CY1113473T1 (el) | 2005-03-31 | 2012-10-16 | ΠΡΟΣΤΑΤΕΥΤΙΚΟΣ ΠΑΡΑΓΩΝ ΓΙΑ ΑΜΦΙΒΛΗΣΤΡΟΕΙΔΙΚΟ ΝΕΥΡΩΝΙΚΟ ΚΥΤΤΑΡΟ ΠΟΥ ΠΕΡΙΕΧΕΙ ΠΑΡΑΓΩΓΟ ΠΡΟΣΤΑΓΛΑΝΔΙΝΗΣ F2α ΩΣ ΔΡΑΣΤΙΚΟ ΣΥΣΤΑΤΙΚΟ |
Country Status (14)
Country | Link |
---|---|
US (2) | US20090234005A1 (el) |
EP (1) | EP1864666B1 (el) |
KR (1) | KR101396731B1 (el) |
CN (2) | CN101151034B (el) |
CA (1) | CA2602573C (el) |
CY (1) | CY1113473T1 (el) |
DK (1) | DK1864666T3 (el) |
ES (1) | ES2389500T3 (el) |
NO (1) | NO339794B1 (el) |
PL (1) | PL1864666T3 (el) |
PT (1) | PT1864666E (el) |
RU (1) | RU2414904C2 (el) |
SI (1) | SI1864666T1 (el) |
WO (1) | WO2006106915A1 (el) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI348386B (en) * | 2003-08-12 | 2011-09-11 | R Tech Ueno Ltd | Composition and method for promoting hair growth |
US7666912B2 (en) | 2006-03-23 | 2010-02-23 | Massachusetts Eye And Ear Infirmary | Compositions and methods for reducing body fat |
WO2008133021A1 (ja) * | 2007-04-12 | 2008-11-06 | R-Tech Ueno, Ltd. | プロスタグランジンF2α化合物を有効成分として含む視神経障害改善剤組成物 |
JP5894364B2 (ja) * | 2007-08-16 | 2016-03-30 | ザ スキーペンズ アイ リサーチ インスティチュート インコーポレイテッド | 眼および付属器組織の炎症を処置するための治療組成物 |
KR101628415B1 (ko) * | 2008-09-04 | 2016-06-08 | 산텐 세이야꾸 가부시키가이샤 | 15,15-디플루오로프로스타글란딘 F2α 유도체를 유효 성분으로서 함유하는 모발 성장 촉진제 |
US20120014970A1 (en) * | 2009-01-09 | 2012-01-19 | Reza Dana | Therapeutic Compositions for Treatment of Corneal Disorders |
JP2012515164A (ja) | 2009-01-09 | 2012-07-05 | ザ スキーペンズ アイ リサーチ インスティチュート インコーポレイテッド | 角膜障害を処置するための治療組成物 |
CA2764063C (en) | 2009-06-03 | 2019-05-14 | Forsight Labs, Llc | Anterior segment drug delivery |
SG187770A1 (en) | 2010-08-12 | 2013-03-28 | Univ Nanyang Tech | A liposomal formulation for ocular drug delivery |
EP2982373B1 (en) | 2011-01-19 | 2018-06-13 | Topokine Therapeutics, Inc. | Methods and compostions for reducing body fat |
WO2013040426A2 (en) | 2011-09-14 | 2013-03-21 | Forsight Labs, Llc | Ocular insert apparatus and methods |
US8426471B1 (en) * | 2011-12-19 | 2013-04-23 | Topokine Therapeutics, Inc. | Methods and compositions for reducing body fat and adipocytes |
CN104884006B (zh) | 2012-10-26 | 2017-12-15 | 弗赛特影像5股份有限公司 | 用于持续释放药物到眼睛的眼科系统 |
NO2753788T3 (el) | 2013-05-10 | 2018-06-16 | ||
US9820993B2 (en) | 2013-05-15 | 2017-11-21 | Topokine Therapeutics, Inc. | Methods and compositions for topical delivery of prostaglandins to subcutaneous fat |
US9956195B2 (en) | 2014-01-07 | 2018-05-01 | Nanyang Technological University | Stable liposomal formulations for ocular drug delivery |
WO2015200425A1 (en) | 2014-06-27 | 2015-12-30 | Topokine Therapeutics, Inc. | Topical dosage regimen |
US20160296532A1 (en) | 2015-04-13 | 2016-10-13 | Forsight Vision5, Inc. | Ocular Insert Composition of a Semi-Crystalline or Crystalline Pharmaceutically Active Agent |
Family Cites Families (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4599353A (en) | 1982-05-03 | 1986-07-08 | The Trustees Of Columbia University In The City Of New York | Use of eicosanoids and their derivatives for treatment of ocular hypertension and glaucoma |
US4822820A (en) * | 1986-11-24 | 1989-04-18 | Alcon Laboratories, Inc. | Use of tri-methyl PG-F2 a and derivatives in glaucoma therapy |
JPH0251225A (ja) | 1988-08-15 | 1990-02-21 | Shin Etsu Chem Co Ltd | 半導体拡散炉用炉芯管 |
ES2213504T1 (es) | 1988-09-06 | 2004-09-01 | Pfizer Health Ab | Derivados de prostaglandina para el tratamiento del glaucoma o hipertension ocular. |
US5352708A (en) | 1992-09-21 | 1994-10-04 | Allergan, Inc. | Non-acidic cyclopentane heptanoic acid, 2-cycloalkyl or arylalkyl derivatives as therapeutic agents |
US5510383A (en) | 1993-08-03 | 1996-04-23 | Alcon Laboratories, Inc. | Use of cloprostenol, fluprostenol and their salts and esters to treat glaucoma and ocular hypertension |
TW420611B (en) * | 1995-03-10 | 2001-02-01 | R Tech Ueno Ltd | Pharmaceutical composition containing prostanoic acid compounds for the treatment of optic nerve disorder |
JP3501310B2 (ja) | 1995-03-10 | 2004-03-02 | 日産ディーゼル工業株式会社 | ディーゼルエンジンの燃料噴射管の保持装置 |
JP3625946B2 (ja) * | 1995-03-10 | 2005-03-02 | 株式会社アールテック・ウエノ | 視神経障害改善剤 |
ZA9610741B (en) * | 1995-12-22 | 1997-06-24 | Warner Lambert Co | 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists |
DE69714698T2 (de) * | 1996-06-10 | 2002-12-05 | Sucampo Ag | Endothelin-antagonisten |
JPH1087607A (ja) | 1996-09-17 | 1998-04-07 | Asahi Glass Co Ltd | 含フッ素プロスタグランジン誘導体の製造方法 |
WO1998012175A1 (fr) | 1996-09-17 | 1998-03-26 | Asahi Glass Company Ltd. | Derives de prostaglandine fluores et medicaments |
JP4004109B2 (ja) * | 1996-09-17 | 2007-11-07 | 参天製薬株式会社 | 含フッ素プロスタグランジン誘導体および医薬 |
JPH10259179A (ja) | 1996-09-19 | 1998-09-29 | Santen Pharmaceut Co Ltd | 多置換アリールオキシ基を有するプロスタグランジン類およびその用途 |
JP3480549B2 (ja) | 1996-12-26 | 2003-12-22 | 参天製薬株式会社 | ジフルオロプロスタグランジン誘導体およびその用途 |
US5877211A (en) * | 1997-11-21 | 1999-03-02 | Allergan | EP2 receptor agonists as neuroprotective agents for the eye |
US6225348B1 (en) * | 1998-08-20 | 2001-05-01 | Alfred W. Paulsen | Method of treating macular degeneration with a prostaglandin derivative |
MXPA01003761A (es) * | 1998-10-13 | 2003-07-21 | Kyowa Hakko Kogyo Kk | Agente para tratar oftalmopatia. |
JP4372905B2 (ja) | 1999-09-02 | 2009-11-25 | 興和株式会社 | 網膜神経細胞保護剤 |
EP1252895A4 (en) | 2000-01-31 | 2003-04-16 | Santen Pharmaceutical Co Ltd | REMEDIES FOR OPHTHALMIC DISORDERS |
US7217722B2 (en) | 2000-02-01 | 2007-05-15 | Kirin Beer Kabushiki Kaisha | Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same |
CA2403086C (en) * | 2000-03-24 | 2010-08-17 | Sucampo Ag | Apoptosis inhibiting composition comprising a 15-keto-prostaglandin or derivative thereof |
DE60143615D1 (de) | 2000-09-13 | 2011-01-20 | Asahi Glass Co Ltd | Augentropfen |
JP2002293771A (ja) | 2001-03-30 | 2002-10-09 | Asahi Glass Co Ltd | 新規なエーテル型ジフルオロプロスタグランジン誘導体またはその塩 |
CA2443918C (en) | 2001-04-11 | 2012-06-05 | Senju Pharmaceutical Co., Ltd. | Visual function disorder improving agents containing rho kinase inhibitors |
JPWO2002100833A1 (ja) | 2001-06-12 | 2004-09-24 | 住友製薬株式会社 | Rhoキナーゼ阻害剤 |
EP1410808A4 (en) | 2001-07-02 | 2009-07-29 | Santen Pharmaceutical Co Ltd | MEDIUM FOR THE PROTECTION OF THE SEHNERV WITH ALPHA 1 RECEPTOR BLOCKER AS AN ACTIVE SUBSTANCE |
JP2003146904A (ja) | 2001-11-08 | 2003-05-21 | Nippon Shinyaku Co Ltd | 緑内障治療薬 |
JP2003321442A (ja) | 2002-04-24 | 2003-11-11 | Santen Pharmaceut Co Ltd | 新規なジフルオロプロスタグランジンアミド誘導体 |
ES2426288T3 (es) | 2003-10-15 | 2013-10-22 | Ube Industries, Ltd. | Novedoso derivado de imidazol |
-
2006
- 2006-03-31 PT PT06730774T patent/PT1864666E/pt unknown
- 2006-03-31 DK DK06730774.4T patent/DK1864666T3/da active
- 2006-03-31 CN CN2006800107892A patent/CN101151034B/zh active Active
- 2006-03-31 ES ES06730774T patent/ES2389500T3/es active Active
- 2006-03-31 PL PL06730774T patent/PL1864666T3/pl unknown
- 2006-03-31 KR KR1020077023372A patent/KR101396731B1/ko active IP Right Grant
- 2006-03-31 US US11/887,037 patent/US20090234005A1/en not_active Abandoned
- 2006-03-31 WO PCT/JP2006/306826 patent/WO2006106915A1/ja active Application Filing
- 2006-03-31 CA CA2602573A patent/CA2602573C/en active Active
- 2006-03-31 SI SI200631410T patent/SI1864666T1/sl unknown
- 2006-03-31 RU RU2007140309/15A patent/RU2414904C2/ru active
- 2006-03-31 CN CN201110176745A patent/CN102293774A/zh active Pending
- 2006-03-31 EP EP06730774A patent/EP1864666B1/en active Active
-
2007
- 2007-10-29 NO NO20075464A patent/NO339794B1/no not_active IP Right Cessation
-
2011
- 2011-09-02 US US13/199,598 patent/US9138438B2/en active Active
-
2012
- 2012-10-16 CY CY20121100958T patent/CY1113473T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
RU2414904C2 (ru) | 2011-03-27 |
US20090234005A1 (en) | 2009-09-17 |
CN101151034B (zh) | 2012-06-06 |
US20120010288A1 (en) | 2012-01-12 |
KR20070116632A (ko) | 2007-12-10 |
CN101151034A (zh) | 2008-03-26 |
DK1864666T3 (da) | 2012-10-29 |
CA2602573C (en) | 2013-10-08 |
NO20075464L (no) | 2007-12-18 |
NO339794B1 (no) | 2017-01-30 |
PL1864666T3 (pl) | 2013-02-28 |
EP1864666A1 (en) | 2007-12-12 |
WO2006106915A1 (ja) | 2006-10-12 |
US9138438B2 (en) | 2015-09-22 |
PT1864666E (pt) | 2012-09-06 |
KR101396731B1 (ko) | 2014-05-19 |
EP1864666B1 (en) | 2012-08-15 |
SI1864666T1 (sl) | 2012-10-30 |
EP1864666A4 (en) | 2008-04-02 |
ES2389500T3 (es) | 2012-10-26 |
RU2007140309A (ru) | 2009-05-10 |
CN102293774A (zh) | 2011-12-28 |
CA2602573A1 (en) | 2006-10-12 |
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