CY1108187T1 - Μεθοδος για την παρασκευη παραγωγων της (3-οξο 2,3-διυδρο-1η-ισοϊνδολ-1-υλο)-ακετυλογουανιδινης - Google Patents
Μεθοδος για την παρασκευη παραγωγων της (3-οξο 2,3-διυδρο-1η-ισοϊνδολ-1-υλο)-ακετυλογουανιδινηςInfo
- Publication number
- CY1108187T1 CY1108187T1 CY20081100727T CY081100727T CY1108187T1 CY 1108187 T1 CY1108187 T1 CY 1108187T1 CY 20081100727 T CY20081100727 T CY 20081100727T CY 081100727 T CY081100727 T CY 081100727T CY 1108187 T1 CY1108187 T1 CY 1108187T1
- Authority
- CY
- Cyprus
- Prior art keywords
- derivatives
- products
- producing
- isoindol
- dihydro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/06—Free radical scavengers or antioxidants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Toxicology (AREA)
- Biochemistry (AREA)
- Oncology (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Gastroenterology & Hepatology (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Η παρούσα εφεύρεση αφορά μία μέθοδο για την παρασκευή παραγώγων της (3-οξο -2,3-διυδρο -1Η-ισοϊνδολ -1-υλο)-ακετυλογουανιδίνης του τύπου (I) μέσω παραγώγων της 3-υδροξυ -2,3-διυδρο -1Η-ισοϊνδολ -1-όνης ή παραγώγων εστέρων του 3-(2-καρβαμοϋλο -φαινυλο) -ακρυλικού οξέος ως ενδιάμεσων βαθμίδων, σε μια μέθοδο για τον διαχωρισμό των ρακεμικών μειγμάτων, καθώς και σε ενδιάμεσα προϊόντα της σύμφωνα με την εφεύρεση μεθόδου.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10356717A DE10356717A1 (de) | 2003-12-02 | 2003-12-02 | Verfahren zur Herstellung von (3-Oxo-2,3-dihydro-1H-isoindol-1-yl)-acetylguanidin-Derivaten |
EP04803188A EP1692105B1 (de) | 2003-12-02 | 2004-11-19 | VERFAHREN ZUR HERSTELLUNG VON (3-OXO-2,3-DIHYDRO-1H-ISOINDOL-1-Yl)-ACETYLGUANIDIN-DERIVATEN |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1108187T1 true CY1108187T1 (el) | 2014-02-12 |
Family
ID=34638338
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20081100727T CY1108187T1 (el) | 2003-12-02 | 2008-07-11 | Μεθοδος για την παρασκευη παραγωγων της (3-οξο 2,3-διυδρο-1η-ισοϊνδολ-1-υλο)-ακετυλογουανιδινης |
Country Status (38)
Country | Link |
---|---|
EP (1) | EP1692105B1 (el) |
JP (1) | JP4809774B2 (el) |
KR (1) | KR101202604B1 (el) |
CN (1) | CN100526297C (el) |
AR (1) | AR046733A1 (el) |
AT (1) | ATE395334T1 (el) |
AU (1) | AU2004295056B2 (el) |
BR (1) | BRPI0417147A (el) |
CA (1) | CA2548020C (el) |
CR (1) | CR8376A (el) |
CY (1) | CY1108187T1 (el) |
DE (2) | DE10356717A1 (el) |
DK (1) | DK1692105T3 (el) |
EC (1) | ECSP066597A (el) |
EG (1) | EG25498A (el) |
ES (1) | ES2304634T3 (el) |
HK (1) | HK1097525A1 (el) |
HR (1) | HRP20080253T3 (el) |
IL (1) | IL175834A (el) |
JO (1) | JO2498B1 (el) |
MA (1) | MA28220A1 (el) |
MY (1) | MY136467A (el) |
NO (1) | NO20063058L (el) |
NZ (1) | NZ547625A (el) |
OA (1) | OA13293A (el) |
PA (1) | PA8618701A1 (el) |
PE (1) | PE20051037A1 (el) |
PL (1) | PL1692105T3 (el) |
PT (1) | PT1692105E (el) |
RS (1) | RS50571B (el) |
RU (1) | RU2397159C2 (el) |
SI (1) | SI1692105T1 (el) |
TN (1) | TNSN06167A1 (el) |
TW (1) | TWI334348B (el) |
UA (1) | UA83883C2 (el) |
UY (1) | UY28648A1 (el) |
WO (1) | WO2005054195A1 (el) |
ZA (1) | ZA200603338B (el) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200812962A (en) * | 2006-07-12 | 2008-03-16 | Astrazeneca Ab | New compounds I/418 |
CA2725230C (en) * | 2008-04-16 | 2016-05-17 | Kissei Pharmaceutical Co., Ltd. | Hemifumarate of a pyrazole derivative |
RU2518740C1 (ru) * | 2013-03-22 | 2014-06-10 | Федеральное государственное автономное образовательное учреждение высшего профессионального образования "ЮЖНЫЙ ФЕДЕРАЛЬНЫЙ УНИВЕРСИТЕТ" | СРЕДСТВО, ИНГИБИРУЮЩЕЕ Na+/H+-ОБМЕН, И ДИГИДРОХЛОРИД 2-(3,4-МЕТИЛЕНДИОКСИФЕНИЛ)-9-МОРФОЛИНОЭТИЛИМИДАЗО[1,2-a]БЕНЗИМИДАЗОЛА |
CN107778238B (zh) * | 2016-08-29 | 2022-07-22 | 中山大学 | 一种3,4-二氢异喹啉-1-酮的合成新方法 |
CN107286074B (zh) * | 2017-08-16 | 2019-08-20 | 厦门华厦学院 | 3-羟基异吲哚-1-酮衍生物及其制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU581324B2 (en) * | 1985-07-05 | 1989-02-16 | Smith Kline & French Laboratories Limited | Substituted 6-phenyl-4,5-dihydro pyradazin-3-ones |
DE19737224A1 (de) * | 1997-08-27 | 1999-03-18 | Hoechst Marion Roussel De Gmbh | Pharmazeutisches Kombinationspräparat aus einem Inhibitor des Natrium-Wasserstoff-Austauschers und einem Arzneimittel zur Behandlung von Herz-Kreislauferkrankungen |
DE19832429A1 (de) * | 1998-07-18 | 2000-01-20 | Hoechst Marion Roussel De Gmbh | Imidazolderivate mit Biphenylsulfonylsubstitution, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
EP1767525A1 (en) | 2001-04-09 | 2007-03-28 | Novartis Vaccines and Diagnostics, Inc. | Guanidino compounds as melanocortin-4 receptor (MC4-R) agonists |
FR2840302B1 (fr) * | 2002-06-03 | 2004-07-16 | Aventis Pharma Sa | Derives d'isoindolones, procede de preparation et intermediaire de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant |
-
2003
- 2003-12-02 DE DE10356717A patent/DE10356717A1/de not_active Withdrawn
-
2004
- 2004-11-04 JO JO2004155A patent/JO2498B1/en active
- 2004-11-19 JP JP2006541829A patent/JP4809774B2/ja not_active Expired - Fee Related
- 2004-11-19 AT AT04803188T patent/ATE395334T1/de active
- 2004-11-19 CN CNB2004800348122A patent/CN100526297C/zh not_active Expired - Fee Related
- 2004-11-19 PL PL04803188T patent/PL1692105T3/pl unknown
- 2004-11-19 OA OA1200600177A patent/OA13293A/en unknown
- 2004-11-19 EP EP04803188A patent/EP1692105B1/de active Active
- 2004-11-19 PT PT04803188T patent/PT1692105E/pt unknown
- 2004-11-19 SI SI200430747T patent/SI1692105T1/sl unknown
- 2004-11-19 DE DE502004007177T patent/DE502004007177D1/de active Active
- 2004-11-19 RU RU2006123410/04A patent/RU2397159C2/ru not_active IP Right Cessation
- 2004-11-19 BR BRPI0417147-0A patent/BRPI0417147A/pt not_active IP Right Cessation
- 2004-11-19 DK DK04803188T patent/DK1692105T3/da active
- 2004-11-19 UA UAA200607292A patent/UA83883C2/ru unknown
- 2004-11-19 KR KR1020067010920A patent/KR101202604B1/ko not_active IP Right Cessation
- 2004-11-19 CA CA2548020A patent/CA2548020C/en not_active Expired - Fee Related
- 2004-11-19 RS RSP-2008/0311A patent/RS50571B/sr unknown
- 2004-11-19 WO PCT/EP2004/013153 patent/WO2005054195A1/de active Application Filing
- 2004-11-19 ES ES04803188T patent/ES2304634T3/es active Active
- 2004-11-19 NZ NZ547625A patent/NZ547625A/en not_active IP Right Cessation
- 2004-11-19 AU AU2004295056A patent/AU2004295056B2/en not_active Ceased
- 2004-11-29 PE PE2004001175A patent/PE20051037A1/es not_active Application Discontinuation
- 2004-11-30 AR ARP040104450A patent/AR046733A1/es not_active Application Discontinuation
- 2004-11-30 TW TW093136804A patent/TWI334348B/zh not_active IP Right Cessation
- 2004-12-01 PA PA20048618701A patent/PA8618701A1/es unknown
- 2004-12-01 MY MYPI20044973A patent/MY136467A/en unknown
- 2004-12-02 UY UY28648A patent/UY28648A1/es not_active Application Discontinuation
-
2006
- 2006-04-26 ZA ZA200603338A patent/ZA200603338B/en unknown
- 2006-04-28 CR CR8376A patent/CR8376A/es unknown
- 2006-05-22 IL IL175834A patent/IL175834A/en not_active IP Right Cessation
- 2006-06-01 TN TNP2006000167A patent/TNSN06167A1/en unknown
- 2006-06-01 EC EC2006006597A patent/ECSP066597A/es unknown
- 2006-06-01 EG EGNA2006000508 patent/EG25498A/xx active
- 2006-06-02 MA MA29077A patent/MA28220A1/fr unknown
- 2006-06-30 NO NO20063058A patent/NO20063058L/no unknown
-
2007
- 2007-03-09 HK HK07102616.3A patent/HK1097525A1/xx not_active IP Right Cessation
-
2008
- 2008-06-09 HR HR20080253T patent/HRP20080253T3/xx unknown
- 2008-07-11 CY CY20081100727T patent/CY1108187T1/el unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1122238T1 (el) | Νεα 1-ναφθυλ-3-αζαδικυκλο[3.1.0]εξανia: παρασκευη και χρηση για τη θεραπεια νευροψυχιατρικων διαταραχων | |
EA200000358A1 (ru) | Способ получения диарилпиридинов, полезных в качестве ингибиторов cox-2 | |
CY1109104T1 (el) | 1,2,3,4 τετρα-υποκατεστημενη ινδολη για την αντιμετωπιση ασθενειων του αναπνευστικου | |
ATE497013T1 (de) | Verfahren zur herstellung von glutaminsäurederivaten | |
CY1110318T1 (el) | Παραγωγα φαινοξυοξικου οξεος | |
ATE440087T1 (de) | 2,4-diaminopyrimidinderivate, die sich als inhibitoren von pkc-theta eignen | |
EA200001102A1 (ru) | Способ синтеза ингибиторов сох-2 (циклооксигеназы-2) | |
SE0303180D0 (sv) | Novel compounds | |
SE0302232D0 (sv) | Novel Compounds | |
CY1109760T1 (el) | Παραγωγα ινδολης-3-θειου | |
CY1105836T1 (el) | 12, 13-τροποποιημενα παραγωγα εποθιλονης | |
DE602004024900D1 (de) | Substituierte 2,3-dihydro-1h-isoindol-1-one derivate und anwendungsverfahren | |
EA200600621A1 (ru) | Производные тетрагидронафталина, способ их получения и их применение в качестве противовоспалительных средств | |
CY1108770T1 (el) | Νεα παραγωγα του ινδολιου και χρηση τους ως φαρμακων | |
CY1109227T1 (el) | Παραγωγα της 5-φαινυλο-4-μεθυλο-θειαζολ-2-υλ-αμινης ως αναστολεις των ενζυμων κινασης της φωσφατιδυλινοσιτολης 3 (p13) για την θεραπεια των φλεγμονωδων ασθενειων των αεραγωγων | |
NO20071577L (no) | Bifenyloksyiddiksyrederivater for behandling av luftveissykdommer | |
CY1108187T1 (el) | Μεθοδος για την παρασκευη παραγωγων της (3-οξο 2,3-διυδρο-1η-ισοϊνδολ-1-υλο)-ακετυλογουανιδινης | |
NO20073839L (no) | Kinolinderivat, fremgangsmate for fremstilling og anvendelse av dette, og legemiddel inneholdende dette | |
EA200800785A1 (ru) | 4-арил-1,4-дигидро-3(2н)-изохинолиноны и 4-арил-1,2,3,4-тетрагидроизохинолины в качестве ингибиторов igf-1r и в качестве фармакологического средства в тест-системах, фармацевтическая композиция и изделие на их основе и способ лечения заболеваний, опосредованных igf-1 рецептором | |
ATE424892T1 (de) | Verfahren zur herstellung von derivaten des 4a,5, 9,10,11,12-hexahydrobenzofuro ä3a,3,2üä 2 ü- benzazepins | |
CY1110458T1 (el) | Παραγωγα βενγαμιδης και η χρηση τους στην αγωγη καρκινικων παθησεων | |
NO994049L (no) | Metode for aa fremstille farmasöytiske forbindelser | |
CY1112080T1 (el) | Μεθοδος διεργασιων για την παρασκευη παραγωγων του διαρυλοκυκλοαλκυλιου | |
ATE421961T1 (de) | Piperidinderivate, verfahren zu deren herstellung und pharmazeutische zusammensetzung zur behandlung von alzheimer-krankheit, die diese derivate enthält | |
ATE348801T1 (de) | Verfahren zur herstellung von disubstituierten 9- alkylidenfluorenen und deren derivaten. |