CY1107384T1 - Ταχεως διασπειρομενες μορφες δοσομετρησεως ανευ ζελατινης - Google Patents
Ταχεως διασπειρομενες μορφες δοσομετρησεως ανευ ζελατινηςInfo
- Publication number
- CY1107384T1 CY1107384T1 CY20081100372T CY081100372T CY1107384T1 CY 1107384 T1 CY1107384 T1 CY 1107384T1 CY 20081100372 T CY20081100372 T CY 20081100372T CY 081100372 T CY081100372 T CY 081100372T CY 1107384 T1 CY1107384 T1 CY 1107384T1
- Authority
- CY
- Cyprus
- Prior art keywords
- dosage forms
- solid dosage
- gelatin
- active ingredient
- rapidly dispersible
- Prior art date
Links
- 108010010803 Gelatin Proteins 0.000 title abstract 3
- 229920000159 gelatin Polymers 0.000 title abstract 3
- 239000008273 gelatin Substances 0.000 title abstract 3
- 235000019322 gelatine Nutrition 0.000 title abstract 3
- 235000011852 gelatine desserts Nutrition 0.000 title abstract 3
- 239000002552 dosage form Substances 0.000 title abstract 2
- 239000007909 solid dosage form Substances 0.000 abstract 5
- 229920000881 Modified starch Polymers 0.000 abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 235000019426 modified starch Nutrition 0.000 abstract 2
- 239000004368 Modified starch Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 238000004108 freeze drying Methods 0.000 abstract 1
- 239000011159 matrix material Substances 0.000 abstract 1
- 210000000214 mouth Anatomy 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Zoology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Abstract
Η παρούσα εφεύρεση αφορά ταχέως διασπειρόμενες στερεές μορφές δοσομετρήσεως, οι οποίες κατά προτίμηση διαλύονται εντός της στοματικής κοιλότητος εντός εξήντα (60), κατά μεγαλυτέρα προτίμηση εντός τριάντα (30), κατά μεγίστη προτίμηση εντός δέκα (10) δευτερολέπτων. Νέο χαρακτηριστικό των στερεών μορφών δοσομετρήσεως οφείλεται εις το γεγονός ότι η σύνθεση είναι ουσιαστικά απηλλαγμένη ή απολύτως απηλλαγμένη από ζελατίνη θηλαστικού. Έχει ανακαλυφθεί ότι η χρησιμοποίηση ορισμένων τροποποιημένων αμύλων εις συγκεντρώσεις από 20 έως 90% κατά βάρος της στερεάς μορφής δοσομετρήσεως παρασκευάζει μορφές δοσομετρήσεως, οι οποίες είναι μηχανικά και χημικά σταθερές και ικανές να χορηγήσουν υψηλότερες συγκεντρώσεις δραστικού συστατικού εν συγκρίσει προς τη χρησιμοποιούμενη προς το σκοπό αυτό ζελατίνη ως βάση δια τις διασπειρόμενες στερεές μορφές δοσομετρήσεως. Περαιτέρω, οι στερεές μορφές δοσομετρήσεως συμφώνως προς την εφεύρεση, δύνανται να ληφθούν δι' απομακρύνσεως διαλυτού όπως ύδατος από μίγμα το οποίον περιέχει ενεργό συστατικό, τροποποιημένο άμυλο και παράγοντα διαμορφώσεως μήτρας μέσω λυοφιλοποιήσεως.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9901819.4A GB9901819D0 (en) | 1999-01-27 | 1999-01-27 | Pharmaceutical compositions |
PCT/US2000/001868 WO2000044351A1 (en) | 1999-01-27 | 2000-01-27 | Fast dispersing dosage forms free of gelatin |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1107384T1 true CY1107384T1 (el) | 2012-01-25 |
Family
ID=10846608
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20081100372T CY1107384T1 (el) | 1999-01-27 | 2008-04-02 | Ταχεως διασπειρομενες μορφες δοσομετρησεως ανευ ζελατινης |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP1154757B1 (el) |
JP (1) | JP4863336B2 (el) |
KR (1) | KR100852015B1 (el) |
CN (1) | CN1193740C (el) |
AT (1) | ATE382334T1 (el) |
AU (1) | AU768121B2 (el) |
BG (1) | BG65413B1 (el) |
CA (1) | CA2360647C (el) |
CY (1) | CY1107384T1 (el) |
CZ (1) | CZ301249B6 (el) |
DE (1) | DE60037653T2 (el) |
DK (1) | DK1154757T3 (el) |
ES (1) | ES2298129T3 (el) |
GB (1) | GB9901819D0 (el) |
HK (1) | HK1037536A1 (el) |
HU (1) | HU226557B1 (el) |
IL (2) | IL144412A0 (el) |
IS (1) | IS2678B (el) |
NO (1) | NO331253B1 (el) |
PL (1) | PL197462B1 (el) |
PT (1) | PT1154757E (el) |
RU (1) | RU2242968C2 (el) |
TR (1) | TR200102504T2 (el) |
WO (1) | WO2000044351A1 (el) |
ZA (1) | ZA200105930B (el) |
Families Citing this family (38)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9904049D0 (en) * | 1999-02-22 | 1999-04-14 | Quadrant Holdings Cambridge | Rapidly-soluble compositions |
US7550156B2 (en) | 2001-11-23 | 2009-06-23 | Rohm And Haas Company | Optimised pellet formulations |
GB0210397D0 (en) | 2002-05-07 | 2002-06-12 | Ferring Bv | Pharmaceutical formulations |
DE60307082T4 (de) * | 2002-05-07 | 2015-04-30 | Ferring B.V. | In der mundhöhle dispergierbare phamarzeutische zusammensetzung mit desmopressin |
DE10237459A1 (de) * | 2002-08-16 | 2004-02-26 | Beiersdorf Ag | Wirkstoffhaltige kosmetische Zubereitung |
MXPA05005528A (es) * | 2002-11-26 | 2006-04-05 | Alk Abello As | Producto farmaceutico de alergeno. |
UA93479C2 (en) * | 2002-11-26 | 2011-02-25 | Альк-Абелло A/C | Allergen dosage form |
US8012505B2 (en) | 2003-02-28 | 2011-09-06 | Alk-Abello A/S | Dosage form having a saccharide matrix |
WO2004075875A1 (en) | 2003-02-28 | 2004-09-10 | Alk-Abello A/S | Dosage form having a saccharide matrix |
ITRM20030288A1 (it) * | 2003-06-10 | 2004-12-11 | Valerio Cioli | Somministrazione sublinguale di antinfiammatori non steroidei (fans) |
EP2322197A2 (en) | 2003-11-10 | 2011-05-18 | Reprise Biopharmaceutics, LLC | Pharmaceutical compositions including low dosages of desmopressin |
DE20321887U1 (de) | 2003-11-10 | 2012-01-20 | Allergan, Inc. | Arzneimittel umfassend niedrige Dosierungen von Desmopressin |
EP1530967B1 (en) | 2003-11-13 | 2006-05-03 | Ferring B.V. | Blister pack and solid dosage form comprising desmopressin |
US20060210590A1 (en) | 2005-02-03 | 2006-09-21 | Alk-Abello A/S | Minor allergen control to increase safety of immunotherapy |
RU2008117396A (ru) | 2005-10-04 | 2009-11-10 | Альк-Абелло А/С (Dk) | Твердая вакцинная композиция |
CN101548958B (zh) * | 2008-04-03 | 2012-10-17 | 万特制药(海南)有限公司 | 一种含有盐酸特比萘芬的分散片 |
US20100286045A1 (en) | 2008-05-21 | 2010-11-11 | Bjarke Mirner Klein | Methods comprising desmopressin |
PT2296686E (pt) | 2008-05-21 | 2014-05-23 | Ferring Bv | Desmopressina orodispersível para aumentar o período inicial de sono não perturbado por noctúria |
US11963995B2 (en) | 2008-05-21 | 2024-04-23 | Ferring B.V. | Methods comprising desmopressin |
DE102008051579A1 (de) * | 2008-10-14 | 2010-04-15 | Rhodia Acetow Gmbh | Biologisch abbaubarer Kunststoff und Verwendung desselben |
JP5752677B2 (ja) | 2009-05-19 | 2015-07-22 | セルジーン コーポレイション | 4−アミノ−2−(2,6−ジオキソピペリジン−3−イル)イソインドリン−1,3−ジオンの製剤 |
EP2442821B1 (en) | 2009-06-18 | 2017-06-14 | Allergan, Inc. | Safe desmopressin administration |
PL2493457T3 (pl) | 2009-10-30 | 2018-01-31 | Ix Biopharma Ltd | Szybko rozpuszczalna stała postać dawkowana |
US10548839B2 (en) * | 2010-03-16 | 2020-02-04 | Wei Tian | Process of manufacturing a lyophilized fast dissolving, multi-phasic dosage form |
JP5602936B2 (ja) * | 2010-03-29 | 2014-10-08 | フイルメニツヒ ソシエテ アノニム | 噴霧乾燥した結晶性活性成分 |
JO3112B1 (ar) | 2010-03-29 | 2017-09-20 | Ferring Bv | تركيبة دوائية سريعة التحلل |
RU2566269C2 (ru) | 2010-03-29 | 2015-10-20 | Ферринг Б.В. | Быстрорастворимая фармацевтическая композиция |
JP6061859B2 (ja) * | 2010-10-08 | 2017-01-18 | アール.ピー. シェーラー テクノロジーズ エルエルシー | デンプンを使用する経口ワクチン速溶性剤型 |
BR112014005134A2 (pt) | 2011-09-16 | 2017-04-18 | Ferring Bv | composição farmacêutica de dissolução rápida |
RU2497505C1 (ru) * | 2012-11-07 | 2013-11-10 | Максим Эдуардович Запольский | Новая лекарственная композиция для лечения болевого синдрома при спазме гладкой мускулатуры |
RU2503447C1 (ru) * | 2012-11-20 | 2014-01-10 | Максим Эдуардович Запольский | Лекарственное средство в форме ородисперсной таблетки и способ получения лекарственного средства |
EP2952200A1 (en) | 2014-06-04 | 2015-12-09 | Alk-Abelló A/S | Allergen for prophylactic treatment of allergy |
CN106259891A (zh) * | 2015-05-28 | 2017-01-04 | 上海旺旺食品集团有限公司 | 一种益生菌口含片及其制备方法 |
RU2674765C2 (ru) * | 2016-10-03 | 2018-12-13 | Михаил Лукич Ткаченко | Антигрибковая композиция эвтектического типа (варианты) |
FI3562486T3 (fi) | 2016-12-31 | 2024-06-04 | Bioxcel Therapeutics Inc | Kielenalaisen deksmedetomidiinin käyttö agitaation hoidossa |
SG11202012772XA (en) | 2018-06-27 | 2021-01-28 | Bioxcel Therapeutics Inc | Film formulations containing dexmedetomidine and methods of producing them |
US20240024288A1 (en) | 2019-07-19 | 2024-01-25 | Bioxcel Therapeutics, Inc. | Non-sedating dexmedetomidine treatment regimens |
US11806334B1 (en) | 2023-01-12 | 2023-11-07 | Bioxcel Therapeutics, Inc. | Non-sedating dexmedetomidine treatment regimens |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE45770B1 (en) * | 1976-10-06 | 1982-11-17 | Wyeth John & Brother Ltd | Pharmaceutical dosage forms |
GB1548022A (en) * | 1976-10-06 | 1979-07-04 | Wyeth John & Brother Ltd | Pharmaceutial dosage forms |
NL8304133A (nl) * | 1983-12-01 | 1985-07-01 | Unilever Nv | Water-in-olie emulsies die gehydrateerde zetmeelkorrels bevatten. |
DE4018247A1 (de) * | 1990-06-07 | 1991-12-12 | Lohmann Therapie Syst Lts | Herstellungsverfahren fuer schnellzerfallende folienfoermige darreichungsformen |
DE69429119T2 (de) * | 1993-07-09 | 2002-07-18 | R.P. Scherer Corp., Troy | Verfahren zur herstellung von gefriergetrockneten arzneistoffdosierungsformen |
GB9401892D0 (en) * | 1994-02-01 | 1994-03-30 | Boots Co Plc | Therapeutic agents |
AU713462B2 (en) * | 1996-07-12 | 1999-12-02 | Daiichi Pharmaceutical Co., Ltd. | Quickly disintegrable compression-molded materials and process for producing the same |
JP4292588B2 (ja) * | 1997-01-31 | 2009-07-08 | 日産化学工業株式会社 | ピリダジノン化合物類の経口製剤 |
-
1999
- 1999-01-27 GB GBGB9901819.4A patent/GB9901819D0/en not_active Ceased
-
2000
- 2000-01-27 CZ CZ20012700A patent/CZ301249B6/cs not_active IP Right Cessation
- 2000-01-27 IL IL14441200A patent/IL144412A0/xx active IP Right Grant
- 2000-01-27 AU AU29729/00A patent/AU768121B2/en not_active Expired
- 2000-01-27 CA CA002360647A patent/CA2360647C/en not_active Expired - Lifetime
- 2000-01-27 RU RU2001123681/15A patent/RU2242968C2/ru not_active IP Right Cessation
- 2000-01-27 ES ES00908371T patent/ES2298129T3/es not_active Expired - Lifetime
- 2000-01-27 DE DE60037653T patent/DE60037653T2/de not_active Expired - Lifetime
- 2000-01-27 KR KR1020017009411A patent/KR100852015B1/ko active IP Right Grant
- 2000-01-27 DK DK00908371T patent/DK1154757T3/da active
- 2000-01-27 CN CNB008031592A patent/CN1193740C/zh not_active Expired - Lifetime
- 2000-01-27 EP EP00908371A patent/EP1154757B1/en not_active Expired - Lifetime
- 2000-01-27 WO PCT/US2000/001868 patent/WO2000044351A1/en active IP Right Grant
- 2000-01-27 PT PT00908371T patent/PT1154757E/pt unknown
- 2000-01-27 JP JP2000595655A patent/JP4863336B2/ja not_active Expired - Fee Related
- 2000-01-27 TR TR2001/02504T patent/TR200102504T2/xx unknown
- 2000-01-27 AT AT00908371T patent/ATE382334T1/de active
- 2000-01-27 HU HU0105107A patent/HU226557B1/hu unknown
- 2000-01-27 PL PL349666A patent/PL197462B1/pl unknown
-
2001
- 2001-07-18 IL IL144412A patent/IL144412A/en not_active IP Right Cessation
- 2001-07-18 ZA ZA200105930A patent/ZA200105930B/en unknown
- 2001-07-25 IS IS6023A patent/IS2678B/is unknown
- 2001-07-26 NO NO20013679A patent/NO331253B1/no not_active IP Right Cessation
- 2001-07-26 BG BG105739A patent/BG65413B1/bg unknown
- 2001-12-04 HK HK01108496A patent/HK1037536A1/xx not_active IP Right Cessation
-
2008
- 2008-04-02 CY CY20081100372T patent/CY1107384T1/el unknown
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