CS375591A3 - Aminoalkylketone derivatives, process of their preparation and pharmaceutical composition comprising thereof - Google Patents

Aminoalkylketone derivatives, process of their preparation and pharmaceutical composition comprising thereof Download PDF

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Publication number
CS375591A3
CS375591A3 CS913755A CS375591A CS375591A3 CS 375591 A3 CS375591 A3 CS 375591A3 CS 913755 A CS913755 A CS 913755A CS 375591 A CS375591 A CS 375591A CS 375591 A3 CS375591 A3 CS 375591A3
Authority
CS
Czechoslovakia
Prior art keywords
group
compounds
solution
mol
thienyl
Prior art date
Application number
CS913755A
Other languages
Czech (cs)
English (en)
Inventor
Louis Lafon
Original Assignee
Lafon Labor
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lafon Labor filed Critical Lafon Labor
Publication of CS375591A3 publication Critical patent/CS375591A3/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Steroid Compounds (AREA)
  • Peptides Or Proteins (AREA)
CS913755A 1990-12-12 1991-12-11 Aminoalkylketone derivatives, process of their preparation and pharmaceutical composition comprising thereof CS375591A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9015591A FR2670492B1 (fr) 1990-12-12 1990-12-12 Nouveaux derives d'aminoalkylcetone, leur procede de preparation et leurs applications en therapeutique.

Publications (1)

Publication Number Publication Date
CS375591A3 true CS375591A3 (en) 1992-06-17

Family

ID=9403177

Family Applications (1)

Application Number Title Priority Date Filing Date
CS913755A CS375591A3 (en) 1990-12-12 1991-12-11 Aminoalkylketone derivatives, process of their preparation and pharmaceutical composition comprising thereof

Country Status (23)

Country Link
US (1) US5446060A (es)
EP (1) EP0490769B1 (es)
JP (1) JPH04334379A (es)
KR (1) KR920012074A (es)
CN (1) CN1029737C (es)
AT (1) ATE121397T1 (es)
AU (1) AU648126B2 (es)
CA (1) CA2057138A1 (es)
CS (1) CS375591A3 (es)
DE (1) DE69109072T2 (es)
DK (1) DK0490769T3 (es)
ES (1) ES2071955T3 (es)
FI (1) FI915809A7 (es)
FR (1) FR2670492B1 (es)
HU (1) HUT62002A (es)
IE (1) IE914311A1 (es)
LT (1) LTIP614A (es)
LV (1) LV10266B (es)
MX (1) MX9102514A (es)
NO (1) NO914845L (es)
NZ (1) NZ240809A (es)
PT (1) PT99726A (es)
ZA (1) ZA919754B (es)

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3189600A (en) * 1963-01-03 1965-06-15 Ciba Geigy Corp Alpha-halogen-gamma tertiary aminobutyrophenones and the corresponding thophenes
DE1217396B (de) * 1963-07-04 1966-05-26 Laboratorie Roger Bellon, Neuilly-sur-Seine (Frankreich) Verfahren zur Herstellung von 1 - (Thienyl-21) - l-oxo-2-amino-propanen
US3417087A (en) * 1965-12-27 1968-12-17 Research Corp 3(aminopropionyl)benzothiophenes
FR2134218A1 (en) * 1971-04-27 1972-12-08 Penciolelli Madeleine Phloroglucinol aminoketones - vasodilators and antispasmodics
FR2184503A2 (en) * 1972-05-19 1973-12-28 Cluzel Roger Alkyl 2-amino-3-(2-thenoyl)propionates - with antibacterial activity
US4009184A (en) * 1974-06-06 1977-02-22 Kali-Chemie Aktiengesellschaft Amino carbonyl derivatives of benzofurans, processes for their production, and pharmaceutical compositions containing the same 2-phenyl-3-[3-dialkylaminopropanoyl]benzofuran compounds
FR2291755A2 (fr) * 1974-11-21 1976-06-18 Delalande Sa Nouveaux benzoyl-2' eth-1' yl)-1 (cinnamyl-4'' piperazin-1'' yl methyl)-2 benzimidazoles, leur procede de preparation et leur application en therapeutique
FR2305982A1 (fr) * 1975-04-03 1976-10-29 Innothera Lab Sa Nouvelles benzothienyl amino (propyl et butyl) cetones, leur procede de preparation et leur application en therapeutique
FR2305981A1 (fr) * 1975-04-03 1976-10-29 Innothera Lab Sa Nouvelles benzothienyl aminoethyl cetones, leur procede de preparation et leur application en therapeutique
FR2453172A1 (fr) * 1979-04-06 1980-10-31 Innothera Lab Sa Nouvelles (thienyl-2) amino-1 butyl cetones, leur procede de preparation et leur application en therapeutique
US4299769A (en) * 1980-04-28 1981-11-10 American Cyanamid Company ω-Heteroaroyl(propionyl or butyryl)-L-prolines
JPS6028973A (ja) * 1983-07-28 1985-02-14 Kaken Pharmaceut Co Ltd チオフェン誘導体
DE3508398A1 (de) * 1985-03-08 1986-11-06 Hoechst Ag, 6230 Frankfurt Fungizide mittel auf der basis von 3-(hetero)-arylpropylaminen sowie neue (hetero)-aryl-propylamine und verfahren zu ihrer herstellung
FR2655043B1 (fr) * 1989-11-24 1992-02-07 Adir Nouveaux derives du thiophene, leur procede de preparation et les compositions pharmaceutiques les renfermant.

Also Published As

Publication number Publication date
DE69109072D1 (de) 1995-05-24
FR2670492A1 (fr) 1992-06-19
ZA919754B (en) 1993-06-11
FI915809L (fi) 1992-06-13
ATE121397T1 (de) 1995-05-15
PT99726A (pt) 1992-10-30
LTIP614A (en) 1994-12-27
CN1029737C (zh) 1995-09-13
DK0490769T3 (da) 1995-07-17
JPH04334379A (ja) 1992-11-20
CA2057138A1 (en) 1992-06-13
AU8894091A (en) 1992-07-09
EP0490769B1 (fr) 1995-04-19
FI915809A0 (fi) 1991-12-10
CN1062353A (zh) 1992-07-01
HU913903D0 (en) 1992-02-28
FI915809A7 (fi) 1992-06-13
NZ240809A (en) 1992-11-25
KR920012074A (ko) 1992-07-25
AU648126B2 (en) 1994-04-14
NO914845L (no) 1992-06-15
MX9102514A (es) 1992-09-01
IE914311A1 (en) 1992-06-17
HUT62002A (en) 1993-03-29
ES2071955T3 (es) 1995-07-01
LV10266A (lv) 1994-10-20
US5446060A (en) 1995-08-29
EP0490769A1 (fr) 1992-06-17
NO914845D0 (no) 1991-12-10
LV10266B (en) 1995-04-20
DE69109072T2 (de) 1995-09-14
FR2670492B1 (fr) 1994-11-04

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