CS240974B2 - Production method of n formyl a n-hydroxymethyl-3-phenoxy-1-azetidincarboxamides - Google Patents

Production method of n formyl a n-hydroxymethyl-3-phenoxy-1-azetidincarboxamides Download PDF

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Publication number
CS240974B2
CS240974B2 CS836141A CS614183A CS240974B2 CS 240974 B2 CS240974 B2 CS 240974B2 CS 836141 A CS836141 A CS 836141A CS 614183 A CS614183 A CS 614183A CS 240974 B2 CS240974 B2 CS 240974B2
Authority
CS
Czechoslovakia
Prior art keywords
phenoxy
formyl
trifluoromethyl
compounds
formula
Prior art date
Application number
CS836141A
Other languages
Czech (cs)
English (en)
Other versions
CS614183A2 (en
Inventor
George J Wright
Lina Ch Teng
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of CS614183A2 publication Critical patent/CS614183A2/cs
Publication of CS240974B2 publication Critical patent/CS240974B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS836141A 1982-09-02 1983-08-23 Production method of n formyl a n-hydroxymethyl-3-phenoxy-1-azetidincarboxamides CS240974B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/414,101 US4505907A (en) 1982-09-02 1982-09-02 N-Formyl and N-hydroxymethyl-3-phenoxy-1-azetidinecarboxamides

Publications (2)

Publication Number Publication Date
CS614183A2 CS614183A2 (en) 1985-06-13
CS240974B2 true CS240974B2 (en) 1986-03-13

Family

ID=23639965

Family Applications (1)

Application Number Title Priority Date Filing Date
CS836141A CS240974B2 (en) 1982-09-02 1983-08-23 Production method of n formyl a n-hydroxymethyl-3-phenoxy-1-azetidincarboxamides

Country Status (25)

Country Link
US (1) US4505907A (fr)
EP (1) EP0102740B1 (fr)
JP (1) JPS601161A (fr)
KR (1) KR900005131B1 (fr)
AU (1) AU553472B2 (fr)
CA (1) CA1185983A (fr)
CS (1) CS240974B2 (fr)
DE (1) DE3367385D1 (fr)
DK (1) DK166297C (fr)
EG (1) EG16473A (fr)
ES (2) ES8504697A1 (fr)
FI (1) FI77226C (fr)
GR (1) GR79337B (fr)
HK (1) HK47587A (fr)
HU (1) HU189740B (fr)
IE (1) IE55770B1 (fr)
IL (1) IL68743A0 (fr)
IN (1) IN161222B (fr)
NO (1) NO157977C (fr)
NZ (1) NZ205448A (fr)
PH (1) PH20572A (fr)
PL (2) PL145986B1 (fr)
PT (1) PT77281B (fr)
YU (1) YU44747B (fr)
ZA (1) ZA834410B (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4571393A (en) * 1982-08-19 1986-02-18 A. H. Robins Company, Incorporated 3-Phenoxy-1-azetidinecarboxamides
US4594189A (en) * 1983-07-06 1986-06-10 A. H. Robins Company, Inc. Process for preparing 3-phenoxy-1-azetidines and carboxamide derivatives
ZA861210B (en) * 1985-02-28 1987-10-28 Robins Co Inc A H 3-aryloxyazetidinecarboxamides as anticonvulsants and antiepileptics
US4956359A (en) * 1985-02-28 1990-09-11 A. H. Robins Company, Inc. 3-aryloxy and 3-arylthioazetidinecarboxamides as anticonvulsants and antiepileptics
FI87559C (fi) * 1985-02-28 1993-01-25 Robins Co Inc A H Foerfarande foer framstaellning av aktiva 3-fenyloxiazetidinkarboxamider
IN162808B (fr) * 1985-02-28 1988-07-09 Robins Co Inc A H
US5068231A (en) * 1985-02-28 1991-11-26 A. H. Robins Company Incorporated Method of treating muscular tension, muscle spasticity and anxiety with 3-aryloxy and 3-arylthioazetidinecarboxamides
US5130309A (en) * 1991-04-12 1992-07-14 A. H. Robins Company, Incorporated Aryloxy and aryloxyalklazetidines as antiarrhythmic and anticonvulsant agents
JP3178922B2 (ja) * 1992-12-03 2001-06-25 小松ゼノア株式会社 エンジンの吸気装置
GB9801501D0 (en) 1998-01-23 1998-03-18 Cerebrus Ltd Chemical compounds - II
EP1049672B1 (fr) 1998-01-23 2003-09-17 Vernalis Research Limited Derives d'azetidinecarboxamides utilises pour traiter des troubles du systeme nerveux central
DK1049670T3 (da) 1998-01-23 2002-11-11 Vernalis Res Ltd Azetidincarboxamidderivater til behandling af CNS-lidelser
GB9917386D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-II
GB9917385D0 (en) * 1999-07-23 1999-09-22 Cerebrus Ltd Chemical compounds-I
EP2202223B1 (fr) * 2007-10-18 2017-01-25 Takeda Pharmaceutical Company Limited Composé hétérocyclique en tant qu'agent diminuant les rpb4 sanguines
US10365007B2 (en) 2014-09-30 2019-07-30 Fujitsu General Limited Ceiling-embedded air conditioner
JP6504349B2 (ja) 2015-03-31 2019-04-24 株式会社富士通ゼネラル 天井埋込型空気調和機
US10288302B2 (en) 2015-03-31 2019-05-14 Fujitsu General Limited Ceiling-embedded air conditioner with airflow guide vane
JP6516095B2 (ja) 2015-04-27 2019-05-22 株式会社富士通ゼネラル 天井埋込型空気調和機

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB872447A (en) * 1958-12-23 1961-07-12 Lepetit Spa 1-carbamyl-3-substituted azetidines
DE2053333A1 (de) * 1970-10-30 1972-05-04 Farbenfabriken Bayer Ag, 5090 Lever Kusen Herbizide Mittel
US4031221A (en) * 1974-06-17 1977-06-21 American Hoechst Corporation Method of treating pain and hypertension
US4379151A (en) * 1978-03-14 1983-04-05 A. H. Robins Company, Inc. 3-Phenoxyazetidines for anorexigenic activity
US4226861A (en) * 1978-04-18 1980-10-07 A. H. Robins Company, Inc. N-Lower-alkyl 3-phenoxy-1-azetidinecarboxamides

Also Published As

Publication number Publication date
HU189740B (en) 1986-07-28
ES537668A0 (es) 1985-09-16
FI77226B (fi) 1988-10-31
EG16473A (en) 1990-12-30
PH20572A (en) 1987-02-18
FI833126A (fi) 1984-03-03
JPS601161A (ja) 1985-01-07
CA1185983A (fr) 1985-04-23
NO157977C (no) 1988-06-22
JPH0452264B2 (fr) 1992-08-21
EP0102740A1 (fr) 1984-03-14
ES523194A0 (es) 1985-04-16
DK166297C (da) 1993-08-30
DE3367385D1 (en) 1986-12-11
NO157977B (no) 1988-03-14
NZ205448A (en) 1985-08-30
AU1459883A (en) 1984-03-08
IE831652L (en) 1984-03-02
FI833126A0 (fi) 1983-09-01
GR79337B (fr) 1984-10-22
IN161222B (fr) 1987-10-24
YU44747B (en) 1991-02-28
PL243555A1 (en) 1984-08-27
IE55770B1 (en) 1991-01-16
EP0102740B1 (fr) 1986-11-05
KR840006203A (ko) 1984-11-22
DK398783D0 (da) 1983-09-01
IL68743A0 (en) 1983-09-30
ES8504697A1 (es) 1985-04-16
FI77226C (fi) 1989-02-10
PL142643B1 (en) 1987-11-30
NO833135L (no) 1984-03-05
PT77281A (en) 1983-10-01
DK166297B (da) 1993-03-29
CS614183A2 (en) 1985-06-13
ES8600234A1 (es) 1985-09-16
KR900005131B1 (ko) 1990-07-20
PL145986B1 (en) 1988-12-31
HK47587A (en) 1987-06-26
AU553472B2 (en) 1986-07-17
YU170483A (en) 1986-04-30
US4505907A (en) 1985-03-19
DK398783A (da) 1984-03-03
PT77281B (en) 1986-02-04
ZA834410B (en) 1984-03-28

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