CS239942B2 - Processing of oxazinbenzothiazin-6,6 dioxide derivatives - Google Patents

Processing of oxazinbenzothiazin-6,6 dioxide derivatives Download PDF

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Publication number
CS239942B2
CS239942B2 CS834311A CS431183A CS239942B2 CS 239942 B2 CS239942 B2 CS 239942B2 CS 834311 A CS834311 A CS 834311A CS 431183 A CS431183 A CS 431183A CS 239942 B2 CS239942 B2 CS 239942B2
Authority
CS
Czechoslovakia
Prior art keywords
methyl
formula
ethyl
het
radical
Prior art date
Application number
CS834311A
Other languages
Czech (cs)
English (en)
Inventor
Soler-Jose Esteve
Original Assignee
Provesan Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Provesan Sa filed Critical Provesan Sa
Publication of CS239942B2 publication Critical patent/CS239942B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Cephalosporin Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
CS834311A 1982-06-15 1983-06-14 Processing of oxazinbenzothiazin-6,6 dioxide derivatives CS239942B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8210409A FR2528433A1 (fr) 1982-06-15 1982-06-15 Nouveaux derives d'oxazinobenzothiazine-6,6-dioxyde, leur preparation et leur application en tant que medicaments

Publications (1)

Publication Number Publication Date
CS239942B2 true CS239942B2 (en) 1986-01-16

Family

ID=9275018

Family Applications (1)

Application Number Title Priority Date Filing Date
CS834311A CS239942B2 (en) 1982-06-15 1983-06-14 Processing of oxazinbenzothiazin-6,6 dioxide derivatives

Country Status (18)

Country Link
US (1) US4563452A (fi)
EP (1) EP0099770B1 (fi)
JP (1) JPS5980687A (fi)
AT (1) ATE21700T1 (fi)
BR (1) BR8303143A (fi)
CA (1) CA1257589A (fi)
CS (1) CS239942B2 (fi)
DE (1) DE3365631D1 (fi)
ES (1) ES8402842A1 (fi)
FR (1) FR2528433A1 (fi)
GR (1) GR78613B (fi)
HU (1) HU187086B (fi)
MX (1) MX157060A (fi)
PL (1) PL142244B1 (fi)
PT (1) PT76861B (fi)
RO (1) RO86084B (fi)
SU (1) SU1195910A3 (fi)
YU (1) YU45135B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4656265A (en) * 1984-06-21 1987-04-07 Pfizer Inc. Cyclic prodrugs of antiinflammatory oxicams
FR2597103B1 (fr) * 1986-04-15 1988-12-16 Provesan Sa Procede de preparation de derives d'oxazinobenzothiazine 6,6-dioxyde
US5196410A (en) * 1986-10-31 1993-03-23 Pfizer Inc. Transdermal flux enhancing compositions
US5244981A (en) * 1990-04-10 1993-09-14 Permeable Technologies, Inc. Silicone-containing contact lens polymers, oxygen permeable contact lenses and methods for making these lenses and treating patients with visual impairment
US5371147A (en) * 1990-10-11 1994-12-06 Permeable Technologies, Inc. Silicone-containing acrylic star polymers, block copolymers and macromonomers
WO2002076463A1 (en) * 2001-03-23 2002-10-03 Smithkline Beecham Corporation Compounds useful as kinase inhibitors for the treatment of hyperproliferative diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3492298A (en) * 1968-02-21 1970-01-27 Mcneilab Inc Oxazino-benzothiazine-6,6-dioxides
US3855216A (en) * 1973-05-29 1974-12-17 Warner Lambert Co Substituted pyrano(3,2-c)(1,2)benzothiazine 6,6-dioxides
US3923801A (en) * 1974-09-23 1975-12-02 Mcneilab Inc Oxazinobenzothiazine 6,6-dioxides
EP0043961A1 (en) * 1980-07-14 1982-01-20 MEDIOLANUM FARMACEUTICI s.r.l. 1,2-Benzothiazinopyrazoles having pharmacological activity

Also Published As

Publication number Publication date
PL242536A1 (en) 1984-08-13
US4563452A (en) 1986-01-07
DE3365631D1 (en) 1986-10-02
GR78613B (fi) 1984-09-27
EP0099770B1 (fr) 1986-08-27
RO86084A (ro) 1985-02-25
JPH0113713B2 (fi) 1989-03-07
RO86084B (ro) 1985-03-02
SU1195910A3 (ru) 1985-11-30
MX157060A (es) 1988-10-25
JPS5980687A (ja) 1984-05-10
ES523120A0 (es) 1984-03-16
YU45135B (en) 1992-03-10
PT76861A (fr) 1983-07-01
EP0099770A1 (fr) 1984-02-01
FR2528433A1 (fr) 1983-12-16
ES8402842A1 (es) 1984-03-16
ATE21700T1 (de) 1986-09-15
FR2528433B1 (fi) 1984-12-28
PL142244B1 (en) 1987-10-31
YU126483A (en) 1986-02-28
CA1257589A (en) 1989-07-18
BR8303143A (pt) 1984-01-31
HU187086B (en) 1985-11-28
PT76861B (fr) 1985-12-16

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