CS223845B2 - Method of making the 5,6,7,8-tetrahydropyrazolo /3,4-b/1,5 diazepin-1h,4h-5,7-dion - Google Patents

Method of making the 5,6,7,8-tetrahydropyrazolo /3,4-b/1,5 diazepin-1h,4h-5,7-dion Download PDF

Info

Publication number
CS223845B2
CS223845B2 CS817964A CS796481A CS223845B2 CS 223845 B2 CS223845 B2 CS 223845B2 CS 817964 A CS817964 A CS 817964A CS 796481 A CS796481 A CS 796481A CS 223845 B2 CS223845 B2 CS 223845B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
alkyl
tetrahydropyrazolo
compound
hydrogen
Prior art date
Application number
CS817964A
Other languages
Czech (cs)
English (en)
Inventor
Gerhard Rackur
Irmgard Hoffamnn
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of CS223845B2 publication Critical patent/CS223845B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C07D231/40—Acylated on said nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CS817964A 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazolo /3,4-b/1,5 diazepin-1h,4h-5,7-dion CS223845B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19792932835 DE2932835A1 (de) 1979-08-14 1979-08-14 Neue 4-aryl-5,6,7,8-tetrahydropyrazolo(3,4-b)diazepin-1h,4h-5,7-dione und verfahren zu ihrer darstellung

Publications (1)

Publication Number Publication Date
CS223845B2 true CS223845B2 (en) 1983-11-25

Family

ID=6078398

Family Applications (4)

Application Number Title Priority Date Filing Date
CS805580A CS223833B2 (en) 1979-08-14 1980-08-13 Method of making the new 4-aryl-5,6,7,8-tetrahydropyrazolo /3,4-b/ dlazepin-1h,4h-5,7-dion
CS817966A CS223847B2 (en) 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazolo/3,4-b/1,5-diazepin-1h,4h-5,7-dions
CS817964A CS223845B2 (en) 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazolo /3,4-b/1,5 diazepin-1h,4h-5,7-dion
CS817965A CS223846B2 (en) 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazole /3,4-b/

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CS805580A CS223833B2 (en) 1979-08-14 1980-08-13 Method of making the new 4-aryl-5,6,7,8-tetrahydropyrazolo /3,4-b/ dlazepin-1h,4h-5,7-dion
CS817966A CS223847B2 (en) 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazolo/3,4-b/1,5-diazepin-1h,4h-5,7-dions

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS817965A CS223846B2 (en) 1979-08-14 1980-08-13 Method of making the 5,6,7,8-tetrahydropyrazole /3,4-b/

Country Status (21)

Country Link
US (1) US4302468A (fi)
EP (2) EP0024038B1 (fi)
JP (1) JPS5630977A (fi)
AR (1) AR226860A1 (fi)
AT (2) ATE3040T1 (fi)
AU (1) AU535884B2 (fi)
CA (1) CA1151645A (fi)
CS (4) CS223833B2 (fi)
DD (3) DD159699A5 (fi)
DE (3) DE2932835A1 (fi)
DK (1) DK350180A (fi)
ES (4) ES8103748A1 (fi)
FI (1) FI802536A (fi)
GR (1) GR69798B (fi)
HU (1) HU180163B (fi)
IL (1) IL60828A (fi)
NO (1) NO802425L (fi)
NZ (1) NZ194633A (fi)
PH (1) PH18209A (fi)
PT (1) PT71692B (fi)
ZA (1) ZA804959B (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5198436A (en) * 1989-10-17 1993-03-30 Ellinwood Jr Everett H Intraoral dosing method of administering trifluorobenzodiazepines

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3558605A (en) * 1969-05-14 1971-01-26 Parke Davis & Co Pyrazolo(3,4-e)(1,4)diazepin-7-(1h)-one compounds
AT325052B (de) * 1972-12-07 1975-10-10 Degussa Verfahren zur herstellung von neuen 6-azabenzo-1,5-diazepinen und ihren salzen

Also Published As

Publication number Publication date
ES494143A0 (es) 1981-03-16
PT71692A (de) 1980-09-01
AU535884B2 (en) 1984-04-12
ES8103749A1 (es) 1981-03-16
PT71692B (de) 1982-01-22
ES8103746A1 (es) 1981-03-16
FI802536A (fi) 1981-02-15
US4302468A (en) 1981-11-24
ES8103747A1 (es) 1981-03-16
EP0050376A1 (de) 1982-04-28
CS223847B2 (en) 1983-11-25
GR69798B (fi) 1982-07-12
CS223833B2 (en) 1983-11-25
NZ194633A (en) 1982-03-23
DE2966484D1 (en) 1984-01-12
ATE5536T1 (de) 1983-12-15
ZA804959B (en) 1981-08-26
NO802425L (no) 1981-02-16
ATE3040T1 (de) 1983-04-15
ES494141A0 (es) 1981-03-16
AU6142380A (en) 1981-02-19
DD152936A5 (de) 1981-12-16
DD159640A5 (de) 1983-03-23
DE2932835A1 (de) 1981-03-26
CA1151645A (en) 1983-08-09
DE3062746D1 (en) 1983-05-19
EP0024038A2 (de) 1981-02-18
EP0024038A3 (en) 1981-04-15
PH18209A (en) 1985-04-30
ES494144A0 (es) 1981-03-16
CS223846B2 (en) 1983-11-25
EP0050376B1 (de) 1983-12-07
DD159699A5 (de) 1983-03-30
EP0024038B1 (de) 1983-04-13
JPS5630977A (en) 1981-03-28
AR226860A1 (es) 1982-08-31
DK350180A (da) 1981-02-15
ES8103748A1 (es) 1981-03-16
HU180163B (en) 1983-02-28
IL60828A (en) 1984-04-30
ES494142A0 (es) 1981-03-16
IL60828A0 (en) 1980-10-26

Similar Documents

Publication Publication Date Title
US4208521A (en) Process for the preparation of imidazo[2,1-b]quinazolinones
US4507488A (en) N-Pyrazolylalkylenediamine intermediates
KR880000439A (ko) 1,8-다리 걸친 4-퀴놀론-3-카르복실산의 제조방법
Hegde et al. Synthesis of 1, 6‐dihydro‐5‐hydroxy‐6‐oxo‐3‐(trifluoromethyl)‐4‐pyridazinecarboxylates
IE48829B1 (en) Production of triazinones
Elnagdi et al. Studies on 3, 5-pyrazolidinediones. IV. Addition of 4-Arylazo-3, 5-pyrazolidinediones to Ethyl Acrylate
US4803270A (en) Process of producing fluoroaniline derivatives
CS223845B2 (en) Method of making the 5,6,7,8-tetrahydropyrazolo /3,4-b/1,5 diazepin-1h,4h-5,7-dion
Gardiner et al. Efficient One-Pot Conversion of 6-Methyl-2-nitroaniline into 1-Alkyloxy-2-alkyl-4-methyl-, 1-Benzyloxy-2-phenyl-4-Methyl-, and 1-Allyloxy-4-methyl-2-vinyl-benzimidazole
US3736316A (en) 1,2,5-benzotriazepin-4-ones and their preparation
JPS5829779A (ja) Ｎ−アミノアルキル−１，５−ベンゾチアゼピン誘導体の製造法
GB1595467A (en) 5-methyliso-oxazole-4-carboxylic acid anilides having pharmaceutical activity
US3158618A (en) Nu-(acylamino)-ephedrines
US3711483A (en) 1,3,6-substituted 5-halouracils
US4095024A (en) Process for the manufacture of 1-aryl-3-carboxypyrazolid-5-ones
US3472847A (en) Conversion of pyrazinoylcyanamides to pyrazinoylguanidines
CA1044240A (en) Process for the preparation of 2-arylamino-2-imidazoline derivatives
US3526628A (en) Process for the production of 5,6-dihydrocytosine compounds
US4895957A (en) Process for the preparation of 4-substituted 3-methyl-1-aryl-5-amino-pyrazoles
US4402876A (en) Production of 2-benzazepines
JPS58167574A (ja) ジカルバメ−ト類
CS224639B2 (en) Method for producing 3,6-disubstituted 4-amino-1,2,4-triazine-5-one
JPS62195366A (ja) ５−ヒドラジノ−１ｈ−ピラゾ−ル系化合物
US4395550A (en) Tetrahydro-2(1H)-quinazolinones and cyclohexene nitriles
ZǍLARU et al. New pyrazole derivatives with potential local anesthetic activity