CS166804B2 - - Google Patents

Info

Publication number
CS166804B2
CS166804B2 CS7061*A CS706174A CS166804B2 CS 166804 B2 CS166804 B2 CS 166804B2 CS 706174 A CS706174 A CS 706174A CS 166804 B2 CS166804 B2 CS 166804B2
Authority
CS
Czechoslovakia
Application number
CS7061*A
Other languages
Czech (cs)
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2105743A external-priority patent/DE2105743C3/de
Priority claimed from DE19712108954 external-priority patent/DE2108954A1/de
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of CS166804B2 publication Critical patent/CS166804B2/cs

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Furan Compounds (AREA)
CS7061*A 1971-02-08 1972-01-26 CS166804B2 (US08088918-20120103-C00476.png)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2105743A DE2105743C3 (de) 1971-02-08 1971-02-08 2-(Furylmethyl)- a -5,9-dialkyl -6,7benzomorphane, Verfahren zu ihrer Herstellung und deren Verwendung
DE19712108954 DE2108954A1 (en) 1971-02-25 1971-02-25 2-(furylmethyl)-6,7-benzomorphans - useful as cns active agents

Publications (1)

Publication Number Publication Date
CS166804B2 true CS166804B2 (US08088918-20120103-C00476.png) 1976-03-29

Family

ID=25760626

Family Applications (4)

Application Number Title Priority Date Filing Date
CS483A CS166801B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26
CS7061*A CS166804B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26
CS7060*A CS166803B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26
CS7059*A CS166802B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CS483A CS166801B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26

Family Applications After (2)

Application Number Title Priority Date Filing Date
CS7060*A CS166803B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26
CS7059*A CS166802B2 (US08088918-20120103-C00476.png) 1971-02-08 1972-01-26

Country Status (25)

Country Link
US (1) US3823150A (US08088918-20120103-C00476.png)
JP (1) JPS5545555B1 (US08088918-20120103-C00476.png)
AT (3) AT318602B (US08088918-20120103-C00476.png)
BE (1) BE779058A (US08088918-20120103-C00476.png)
BG (3) BG19600A3 (US08088918-20120103-C00476.png)
CA (1) CA969938A (US08088918-20120103-C00476.png)
CH (4) CH573933A5 (US08088918-20120103-C00476.png)
CS (4) CS166801B2 (US08088918-20120103-C00476.png)
DD (1) DD95847A5 (US08088918-20120103-C00476.png)
DK (1) DK129127B (US08088918-20120103-C00476.png)
ES (4) ES399536A1 (US08088918-20120103-C00476.png)
FI (1) FI57758C (US08088918-20120103-C00476.png)
FR (1) FR2124564B1 (US08088918-20120103-C00476.png)
GB (1) GB1384115A (US08088918-20120103-C00476.png)
HU (1) HU162946B (US08088918-20120103-C00476.png)
IE (1) IE36071B1 (US08088918-20120103-C00476.png)
IL (1) IL38699A (US08088918-20120103-C00476.png)
NL (1) NL171898C (US08088918-20120103-C00476.png)
NO (1) NO134054C (US08088918-20120103-C00476.png)
PH (1) PH10743A (US08088918-20120103-C00476.png)
PL (2) PL78312B1 (US08088918-20120103-C00476.png)
RO (5) RO59193A (US08088918-20120103-C00476.png)
SE (1) SE363630B (US08088918-20120103-C00476.png)
SU (4) SU469246A3 (US08088918-20120103-C00476.png)
YU (3) YU35016B (US08088918-20120103-C00476.png)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2229695A1 (de) * 1972-06-19 1974-01-31 Boehringer Sohn Ingelheim 2-(heteroaryl-methyl)-5,9 beta-dialkyl6,7-benzomorphane, deren saeureadditionssalze sowie verfahren zu deren herstellung
US4010164A (en) * 1973-03-28 1977-03-01 Boehringer Ingelheim Gmbh N-(furyl-methyl)-2-hydroxy-5,9,9-trimethyl-benzomorphans and salts thereof
SU510999A3 (ru) * 1973-10-27 1976-04-15 К.Х.Берингер Зон, (Фирма) Способ получени (метоксиметил-фурилметил)6,7-бензоморфанов илиморфинанов
US4087532A (en) * 1974-03-09 1978-05-02 Boehringer Ingelheim Gmbh Analgesically useful 2-tetrahydrofurfuryl-5-lower alkyl-2-oxy-6,7-benzomorphans and salts thereof
DE2437610A1 (de) * 1974-08-05 1976-02-26 Boehringer Sohn Ingelheim Neue 5,9-beta-disubstituierte 2-tetrahydrofurfuryl-6,7-benzomorphane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung
GB1575009A (en) * 1976-06-21 1980-09-17 Acf Chemiefarma Nv 6,7-benzomorphan derivatives
DE2716687A1 (de) * 1977-04-15 1978-10-19 Boehringer Sohn Ingelheim 2'-hydroxy-2-(5-isoxazolylmethyl)-6,7benzomorphane, deren saeureadditionssalze und diese enthaltende arzneimittel
DE3839659A1 (de) * 1988-11-24 1990-05-31 Boehringer Ingelheim Kg Verwendung von benzomorphanen zur zytoprotektion
AR069545A1 (es) * 2007-11-16 2010-02-03 Boehringer Ingelheim Pharma Derivados de aril y heteroarilcarbonilo de benzomorfanos y estructuras relacionadas, composiciones farmaceuticas que contienen dichos compuestos, obtencion de las mismas, su uso en el tratamiento de enfermedades mediadas por la inhibicion de la enzima 11beta-hidroxiesteroide deshidrogenasa (hsd) 1 y
EP2245014B1 (en) * 2008-02-12 2011-11-02 Boehringer Ingelheim International GmbH Urea derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use
TW200950780A (en) 2008-05-13 2009-12-16 Boehringer Ingelheim Int Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use
WO2013025664A1 (en) 2011-08-17 2013-02-21 Boehringer Ingelheim International Gmbh Indenopyridine derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1281227A (fr) * 1958-09-22 1962-01-12 Smith Kline French Lab Perfectionnements apportés aux procédés pour la préparation de dérivés d'aralcoylbenzomorphane
FR1538362A (fr) * 1966-05-20 1968-09-06 Merck & Co Inc Dérivés du benzomorphane

Also Published As

Publication number Publication date
CH574442A5 (US08088918-20120103-C00476.png) 1976-04-15
RO59165A (US08088918-20120103-C00476.png) 1976-02-15
CS166803B2 (US08088918-20120103-C00476.png) 1976-03-29
YU172078A (en) 1980-04-30
SE363630B (US08088918-20120103-C00476.png) 1974-01-28
NL171898B (nl) 1983-01-03
PL78312B1 (en) 1975-06-30
CS166802B2 (US08088918-20120103-C00476.png) 1976-03-29
CS166801B2 (US08088918-20120103-C00476.png) 1976-03-29
ES408276A1 (es) 1975-11-16
CH573934A5 (US08088918-20120103-C00476.png) 1976-03-31
ES408274A1 (es) 1976-02-01
YU35255B (en) 1980-10-31
NO134054B (US08088918-20120103-C00476.png) 1976-05-03
JPS5545555B1 (US08088918-20120103-C00476.png) 1980-11-18
IE36071B1 (en) 1976-08-04
DK129127C (US08088918-20120103-C00476.png) 1975-02-10
HU162946B (US08088918-20120103-C00476.png) 1973-05-28
RO63052A (fr) 1978-06-15
FR2124564B1 (US08088918-20120103-C00476.png) 1975-10-31
CH573935A5 (US08088918-20120103-C00476.png) 1976-03-31
IE36071L (en) 1973-06-08
ES399536A1 (es) 1974-11-01
IL38699A (en) 1975-12-31
BG19800A3 (US08088918-20120103-C00476.png) 1975-10-10
DK129127B (da) 1974-08-26
ES408275A1 (es) 1976-02-16
PL84115B3 (en) 1976-03-31
SU469246A3 (ru) 1975-04-30
BE779058A (fr) 1972-08-07
SU421187A3 (ru) 1974-03-25
PH10743A (en) 1977-09-01
FI57758B (fi) 1980-06-30
BG20792A3 (US08088918-20120103-C00476.png) 1975-12-20
CH573933A5 (US08088918-20120103-C00476.png) 1976-03-31
CA969938A (en) 1975-06-24
YU27972A (en) 1979-12-31
SU479290A3 (ru) 1975-07-30
US3823150A (en) 1974-07-09
RO58981A (US08088918-20120103-C00476.png) 1975-11-15
RO59251A (US08088918-20120103-C00476.png) 1976-05-15
NL171898C (nl) 1983-06-01
FR2124564A1 (US08088918-20120103-C00476.png) 1972-09-22
AT318602B (de) 1974-11-11
GB1384115A (en) 1975-02-19
BG19600A3 (US08088918-20120103-C00476.png) 1975-06-25
AT318601B (de) 1974-11-11
YU35016B (en) 1980-06-30
NO134054C (US08088918-20120103-C00476.png) 1976-08-11
RO59193A (US08088918-20120103-C00476.png) 1976-01-15
FI57758C (fi) 1980-10-10
DD95847A5 (US08088918-20120103-C00476.png) 1973-02-20
AT312587B (de) 1974-01-10
NL7201551A (US08088918-20120103-C00476.png) 1972-08-10
SU467519A3 (ru) 1975-04-15
IL38699A0 (en) 1972-04-27

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