CR20110195A - Compuestos heteroaromáticos espirocíclicos fusionados para el tratamiento de infecciones bacterianas - Google Patents

Compuestos heteroaromáticos espirocíclicos fusionados para el tratamiento de infecciones bacterianas

Info

Publication number
CR20110195A
CR20110195A CR20110195A CR20110195A CR20110195A CR 20110195 A CR20110195 A CR 20110195A CR 20110195 A CR20110195 A CR 20110195A CR 20110195 A CR20110195 A CR 20110195A CR 20110195 A CR20110195 A CR 20110195A
Authority
CR
Costa Rica
Prior art keywords
bacterial infections
fusioned
treatment
heteroaromatic compounds
spirocyclic
Prior art date
Application number
CR20110195A
Other languages
English (en)
Inventor
Kevin Barvian
Gregory Steven Basarab
Madhusudhan Reddy Gowravaram
Sheila Irene Hauck
Fei Zhou
Original Assignee
Cayman Chem Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cayman Chem Co filed Critical Cayman Chem Co
Publication of CR20110195A publication Critical patent/CR20110195A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains four or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)

Abstract

La presente invención se refiere a compuestos de la fórmula I, a sales farmacéuticamente aceptables de estos, a métodos de utilización de estos para tratar infecciones bacterianas y métodos para su preparación.
CR20110195A 2008-10-14 2011-04-14 Compuestos heteroaromáticos espirocíclicos fusionados para el tratamiento de infecciones bacterianas CR20110195A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10518908P 2008-10-14 2008-10-14

Publications (1)

Publication Number Publication Date
CR20110195A true CR20110195A (es) 2011-06-08

Family

ID=41668347

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20110195A CR20110195A (es) 2008-10-14 2011-04-14 Compuestos heteroaromáticos espirocíclicos fusionados para el tratamiento de infecciones bacterianas

Country Status (24)

Country Link
US (1) US8658641B2 (es)
EP (1) EP2350077B1 (es)
JP (2) JP5749169B2 (es)
KR (1) KR101676886B1 (es)
CN (2) CN104086565A (es)
AR (1) AR073862A1 (es)
AU (1) AU2009305203B2 (es)
BR (1) BRPI0920180B1 (es)
CA (1) CA2736335C (es)
CL (1) CL2011000838A1 (es)
CO (1) CO6382126A2 (es)
CR (1) CR20110195A (es)
CU (1) CU20110083A7 (es)
DO (1) DOP2011000102A (es)
EA (1) EA201100613A1 (es)
EC (1) ECSP11010980A (es)
ES (1) ES2565611T3 (es)
HK (2) HK1160127A1 (es)
IL (1) IL211728A0 (es)
MX (1) MX2011003598A (es)
TW (1) TW201020258A (es)
UY (1) UY32174A (es)
WO (1) WO2010043893A1 (es)
ZA (1) ZA201103533B (es)

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JP6540971B2 (ja) * 2014-08-25 2019-07-10 日産化学株式会社 Ｓｏｃパターン上でのパターン反転のための被覆用組成物
EP3215510B1 (en) 2014-11-06 2023-06-07 Bial-R&D Investments, S.A. Substituted imidazo[1,5-a]pyrimidines and their use in the treatment of medical disorders
FI3215511T3 (fi) 2014-11-06 2024-05-16 Bial R&D Invest S A Substituoituja pyratsolo(1,5-a)pyrimidiinejä ja niiden käyttö lääketieteellisten häiriöiden hoitamisessa
WO2016073891A1 (en) 2014-11-06 2016-05-12 Lysosomal Therapeutics Inc. Substituted pyrrolo[1,2-a]pyrimidines and their use in the treatment of medical disorders
SG11201708622UA (en) 2015-02-02 2017-11-29 Forma Therapeutics Inc 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as hdac inhibitors
WO2016126726A1 (en) 2015-02-02 2016-08-11 Forma Therapeutics, Inc. Bicyclic [4,6,0] hydroxamic acids as hdac6 inhibitors
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CN105152962B (zh) * 2015-09-30 2017-06-16 淄博亿丰高分子材料科技股份有限公司 N‑异丙基羟胺的制备方法
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CA3008809A1 (en) 2015-12-17 2017-06-22 Janssen Pharmaceutica Nv Antibodies to risperidone and use thereof
WO2017176961A1 (en) 2016-04-06 2017-10-12 Lysosomal Therapeutics Inc. Imidazo [1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
KR20180133461A (ko) 2016-04-06 2018-12-14 리소소말 테라퓨틱스 인크. 피라졸로[1,5-a]피리미디닐 카르복스아미드 화합물 및 의학적 장애의 치료에서의 그의 용도
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AU2017261291C1 (en) * 2016-05-05 2022-05-26 Bial - R&D Investments, S.A. Substituted imidazo[1,2-b]pyridazines, substituted imidazo[1,5-b]pyridazines, related compounds, and their use in the treatment of medical disorders
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Also Published As

Publication number Publication date
KR101676886B1 (ko) 2016-11-16
EP2350077B1 (en) 2016-01-27
BRPI0920180B1 (pt) 2021-10-26
HK1203483A1 (en) 2015-10-30
UY32174A (es) 2010-05-31
CN102245605B (zh) 2016-01-27
CA2736335C (en) 2017-05-09
US8658641B2 (en) 2014-02-25
JP2012505261A (ja) 2012-03-01
IL211728A0 (en) 2011-06-30
CO6382126A2 (es) 2012-02-15
KR20110090895A (ko) 2011-08-10
MX2011003598A (es) 2011-04-27
AR073862A1 (es) 2010-12-09
CA2736335A1 (en) 2010-04-22
HK1160127A1 (zh) 2012-08-10
ZA201103533B (en) 2012-01-25
WO2010043893A1 (en) 2010-04-22
CU20110083A7 (es) 2013-05-31
JP2015178510A (ja) 2015-10-08
CN102245605A (zh) 2011-11-16
BRPI0920180A2 (pt) 2020-12-29
EP2350077A1 (en) 2011-08-03
AU2009305203A1 (en) 2010-04-22
DOP2011000102A (es) 2011-05-15
ES2565611T3 (es) 2016-04-05
TW201020258A (en) 2010-06-01
US20110245224A1 (en) 2011-10-06
AU2009305203B2 (en) 2013-03-07
ECSP11010980A (es) 2011-05-31
JP5749169B2 (ja) 2015-07-15
CL2011000838A1 (es) 2011-10-21
EA201100613A1 (ru) 2011-12-30
CN104086565A (zh) 2014-10-08

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