CO6341514A2 - Método para reducir la variabilidad de la absorción de paracetamol en pacientes con dismotilidad gástrica - Google Patents

Método para reducir la variabilidad de la absorción de paracetamol en pacientes con dismotilidad gástrica

Info

Publication number
CO6341514A2
CO6341514A2 CO11009937A CO11009937A CO6341514A2 CO 6341514 A2 CO6341514 A2 CO 6341514A2 CO 11009937 A CO11009937 A CO 11009937A CO 11009937 A CO11009937 A CO 11009937A CO 6341514 A2 CO6341514 A2 CO 6341514A2
Authority
CO
Colombia
Prior art keywords
agent
gastric
patients
reducing
patient
Prior art date
Application number
CO11009937A
Other languages
English (en)
Inventor
Duke Edwuard Clarke Geoffrey
James Grattan Timothy
Burnett Ian
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Publication of CO6341514A2 publication Critical patent/CO6341514A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención está dirigida a un método novedoso para reducir a variabilidad intrapaciente en un agente farmacéuticamente activo que de manera adecuada no es absorbido en el estómago, tal como formulaciones que contienen paracetamol en pacientes que tienen dismotilidad gástrica, o un método para mejorar la analgesia en un paciente diabético, o mejorar la absorción de un agente activo en un paciente con dismotilidad gástrica, dichos métodos comprenden administrar oralmente a dicho paciente que lo necesita una forma de dosificación farmacéutica que comprende un primer agente activo, carbonato de calcio, al menos un primer agente aglutinante, y al menos un agente desintegrante como componentes intragranulares en forma de un material granulado, y como un componente extragranular al menos un coloide hidrofílico, de manera opcional un segundo agente aglutinante, carbonato de calcio, un superdesintegrante, y un segundo agente activo.
CO11009937A 2008-07-30 2011-01-28 Método para reducir la variabilidad de la absorción de paracetamol en pacientes con dismotilidad gástrica CO6341514A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0813929.7A GB0813929D0 (en) 2008-07-30 2008-07-30 Novel method

Publications (1)

Publication Number Publication Date
CO6341514A2 true CO6341514A2 (es) 2011-11-21

Family

ID=39747175

Family Applications (1)

Application Number Title Priority Date Filing Date
CO11009937A CO6341514A2 (es) 2008-07-30 2011-01-28 Método para reducir la variabilidad de la absorción de paracetamol en pacientes con dismotilidad gástrica

Country Status (12)

Country Link
US (2) US8604084B2 (es)
EP (1) EP2309852A4 (es)
CN (1) CN102170782A (es)
AU (1) AU2009276664B2 (es)
BR (1) BRPI0916597A2 (es)
CO (1) CO6341514A2 (es)
GB (1) GB0813929D0 (es)
MX (1) MX2011001124A (es)
MY (1) MY151230A (es)
NZ (1) NZ591408A (es)
RU (1) RU2517139C2 (es)
WO (1) WO2010014661A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2811202A1 (en) 2010-09-13 2012-03-22 Bev-Rx, Inc. Aqueous drug delivery system comprising off-flavor masking agent
JP6539274B2 (ja) 2013-08-12 2019-07-03 ファーマシューティカル マニュファクチュアリング リサーチ サービシズ,インコーポレーテッド 押出成形された即放性乱用抑止性丸剤
WO2015095391A1 (en) 2013-12-17 2015-06-25 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
US9492444B2 (en) 2013-12-17 2016-11-15 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
DK3169315T3 (da) 2014-07-17 2020-08-10 Pharmaceutical Manufacturing Res Services In Væskefyldt doseringsform til forhindring af misbrug med øjeblikkelig frigivelse
EP3209282A4 (en) 2014-10-20 2018-05-23 Pharmaceutical Manufacturing Research Services, Inc. Extended release abuse deterrent liquid fill dosage form
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
CN115444823B (zh) * 2022-10-12 2024-02-23 苏州中化药品工业有限公司 一种含瑞巴派特颗粒及其制备方法和应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1182049A (en) * 1981-07-13 1985-02-05 Francis J. Sterbenz Apap antacid composition
US6264983B1 (en) * 1999-09-16 2001-07-24 Rhodia, Inc. Directly compressible, ultra fine acetaminophen compositions and process for producing same
GB0114069D0 (en) 2001-06-08 2001-08-01 Smithkline Beecham Plc Composition
JP2006510593A (ja) * 2002-09-12 2006-03-30 ザ ユニヴァーシティ オヴ シカゴ 胃内容排出及び胃不全麻痺のモニタリング及び診断
US20050108021A1 (en) 2003-07-31 2005-05-19 Greg Anderson System and method for routing and managing service requests
US8216610B2 (en) * 2004-05-28 2012-07-10 Imaginot Pty Ltd. Oral paracetamol formulations
CN101048155A (zh) * 2004-10-28 2007-10-03 诺瓦提斯公司 含有对乙酰氨基酚、咖啡因和任选的阿司匹林以及用于增强吸收的碱性剂的组合物
GB0607085D0 (en) * 2006-04-07 2006-05-17 Smithkline Beecham Corp Novel compositions
US7863275B2 (en) * 2006-10-30 2011-01-04 The Board Of Regents Of The University Of Texas System Uses of tetrahydrobiopterin and derivatives thereof

Also Published As

Publication number Publication date
BRPI0916597A2 (pt) 2015-08-04
RU2011107285A (ru) 2012-09-10
MY151230A (en) 2014-04-30
EP2309852A1 (en) 2011-04-20
US20140066516A1 (en) 2014-03-06
GB0813929D0 (en) 2008-09-03
EP2309852A4 (en) 2011-08-24
NZ591408A (en) 2012-12-21
CN102170782A (zh) 2011-08-31
AU2009276664B2 (en) 2013-02-07
MX2011001124A (es) 2011-03-29
WO2010014661A1 (en) 2010-02-04
US20110301243A1 (en) 2011-12-08
AU2009276664A1 (en) 2010-02-04
US8604084B2 (en) 2013-12-10
RU2517139C2 (ru) 2014-05-27

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