CO4910160A1 - Formulaciones y formas polimorficas de desferrioxamina y su preparacion - Google Patents

Formulaciones y formas polimorficas de desferrioxamina y su preparacion

Info

Publication number
CO4910160A1
CO4910160A1 CO97072069A CO97072069A CO4910160A1 CO 4910160 A1 CO4910160 A1 CO 4910160A1 CO 97072069 A CO97072069 A CO 97072069A CO 97072069 A CO97072069 A CO 97072069A CO 4910160 A1 CO4910160 A1 CO 4910160A1
Authority
CO
Colombia
Prior art keywords
preparation
despherrioxamine
formulations
polymorphic forms
desferrioxamine
Prior art date
Application number
CO97072069A
Other languages
English (en)
Inventor
Ian Francis-Hass
Nicholas Lowther
Joanne Nicklin
Alan Steward
Peter Van Hoogevest
Erwim Marti
Andre Joseph Geoffroy
Hans Hirt
Andreas Burkhard
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9625878.5A external-priority patent/GB9625878D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CO4910160A1 publication Critical patent/CO4910160A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
    • C07C259/06Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

Una composición parenteralmente inyectable quecomprende partículas de una sal de desferrioxamina-B de un ácido sulfónico alifático que tiene cuando menos 8 átomos de carbono, suspendida en un aceite parenteralmente administrable.8- Un método para la preparación de una composición de acuerdo con cualquiera de las reivindicaciones 1 a 7, el cual comprende mezclar partículas de la sal de desferrioxamina-B con el aceite parenteralmente administrable, y en donde esté presente, el tensoactivo.
CO97072069A 1996-12-10 1997-12-10 Formulaciones y formas polimorficas de desferrioxamina y su preparacion CO4910160A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH302496 1996-12-10
GBGB9625878.5A GB9625878D0 (en) 1996-12-12 1996-12-12 Compositions

Publications (1)

Publication Number Publication Date
CO4910160A1 true CO4910160A1 (es) 2000-04-24

Family

ID=25691970

Family Applications (1)

Application Number Title Priority Date Filing Date
CO97072069A CO4910160A1 (es) 1996-12-10 1997-12-10 Formulaciones y formas polimorficas de desferrioxamina y su preparacion

Country Status (15)

Country Link
EP (1) EP0944586A2 (es)
KR (1) KR20000069376A (es)
CN (1) CN1239946A (es)
AR (1) AR009655A1 (es)
AU (1) AU5983998A (es)
BR (1) BR9713570A (es)
CA (1) CA2274761A1 (es)
CO (1) CO4910160A1 (es)
CZ (1) CZ204499A3 (es)
ID (1) ID22388A (es)
IL (1) IL130203A0 (es)
PE (1) PE27799A1 (es)
PL (1) PL334316A1 (es)
TR (1) TR199901260T2 (es)
WO (1) WO1998025887A2 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001085093A2 (en) * 1999-12-23 2001-11-15 Neurochem, Inc. Compounds and methods for modulating cerebral amyloid angiopathy
GB0117645D0 (en) 2001-07-19 2001-09-12 Isis Innovation Therapeutic stratergies for prevention and treatment of alzheimers disease
DE10223913A1 (de) * 2002-05-29 2003-12-11 Bayer Cropscience Ag Verfahren zur Herstellung spezifischer Kristallmodifikationen polymorpher Substanzen
TWI722031B (zh) 2015-10-23 2021-03-21 瑞士商威佛(國際)股份有限公司 新穎的膜鐵運輸蛋白(ferroportin)抑制劑
JOP20180036A1 (ar) 2017-04-18 2019-01-30 Vifor Int Ag أملاح لمثبطات فروبورتين جديدة
TW202102478A (zh) 2019-04-01 2021-01-16 瑞士商威佛(國際)股份有限公司 新穎的鐵螯合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH438351A (de) * 1959-09-25 1967-06-30 Ciba Geigy Verfahren zur Herstellung neuer Wuchsstoffe
FR1898M (fr) * 1961-04-07 1963-07-08 Ciba Geigy Nouvelle substance utilisable en thérapeutique.
GB9211779D0 (en) * 1992-06-03 1992-07-15 Ciba Geigy Ag Amine salts

Also Published As

Publication number Publication date
CN1239946A (zh) 1999-12-29
PL334316A1 (en) 2000-02-14
AU5983998A (en) 1998-07-03
WO1998025887A2 (en) 1998-06-18
PE27799A1 (es) 1999-03-18
EP0944586A2 (en) 1999-09-29
KR20000069376A (ko) 2000-11-25
TR199901260T2 (xx) 1999-10-21
IL130203A0 (en) 2000-06-01
WO1998025887A3 (en) 1998-08-13
BR9713570A (pt) 2000-03-14
ID22388A (id) 1999-10-07
CZ204499A3 (cs) 1999-09-15
AR009655A1 (es) 2000-04-26
CA2274761A1 (en) 1998-06-18

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