CO4770978A1 - Empleo de epinastina para el tratamiento de dolores - Google Patents

Empleo de epinastina para el tratamiento de dolores

Info

Publication number
CO4770978A1
CO4770978A1 CO96060061A CO96060061A CO4770978A1 CO 4770978 A1 CO4770978 A1 CO 4770978A1 CO 96060061 A CO96060061 A CO 96060061A CO 96060061 A CO96060061 A CO 96060061A CO 4770978 A1 CO4770978 A1 CO 4770978A1
Authority
CO
Colombia
Prior art keywords
epinastine
pain treatment
pain
racemate
enantiomers
Prior art date
Application number
CO96060061A
Other languages
English (en)
Inventor
Birgit Jung
Meade Christopher John Montague
Michael Pairet
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of CO4770978A1 publication Critical patent/CO4770978A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Empleo de epinastina en forma de sus enantiómeros, sus mezclas odel racemato como medicamentos para el tratamiento de dolores. Empleo de epinastina como racemato o en forma de sus enantiómeros que se presenta como base libre o como sal por adición de ácidos con un ácido farmacológicamente inocuo para la preparación de un medicamento para el tratamiento terapéutico de dolores.
CO96060061A 1995-11-14 1996-11-14 Empleo de epinastina para el tratamiento de dolores CO4770978A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19542281A DE19542281C2 (de) 1995-11-14 1995-11-14 Verwendung von Epinastin für die Behandlung der Migräne

Publications (1)

Publication Number Publication Date
CO4770978A1 true CO4770978A1 (es) 1999-04-30

Family

ID=7777343

Family Applications (1)

Application Number Title Priority Date Filing Date
CO96060061A CO4770978A1 (es) 1995-11-14 1996-11-14 Empleo de epinastina para el tratamiento de dolores

Country Status (32)

Country Link
US (1) US5942503A (es)
EP (1) EP0861081B1 (es)
JP (2) JP4264850B2 (es)
KR (1) KR100435611B1 (es)
CN (1) CN1104242C (es)
AR (1) AR004321A1 (es)
AT (1) ATE213160T1 (es)
AU (1) AU706112B2 (es)
BG (1) BG62511B1 (es)
BR (1) BR9611502A (es)
CA (1) CA2232008C (es)
CO (1) CO4770978A1 (es)
CZ (1) CZ290115B6 (es)
DE (2) DE19542281C2 (es)
DK (1) DK0861081T3 (es)
EE (1) EE03512B1 (es)
ES (1) ES2171746T3 (es)
HK (1) HK1015280A1 (es)
HU (1) HU225759B1 (es)
IL (1) IL123601A (es)
NO (1) NO982172D0 (es)
NZ (1) NZ322467A (es)
PL (1) PL186615B1 (es)
PT (1) PT861081E (es)
RO (1) RO118373B1 (es)
RU (2) RU2238733C2 (es)
SK (1) SK61398A3 (es)
TR (1) TR199800853T2 (es)
TW (1) TW575423B (es)
UY (1) UY24354A1 (es)
WO (1) WO1997017971A1 (es)
ZA (1) ZA969520B (es)

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DE19954516A1 (de) * 1999-11-12 2001-05-17 Boehringer Ingelheim Int Epinastin-haltige Lösungen
DE19958460A1 (de) * 1999-12-03 2001-06-07 Boehringer Ingelheim Pharma Verfahren zur Herstellung von Epinastine-Hydrochlorid in der hochschmelzenden Kristallmodifikation
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US20030104017A1 (en) * 2001-10-26 2003-06-05 Boehringer Ingelheim International Gmbh Epinastine formulation for oral administration
DE10152973A1 (de) * 2001-10-26 2003-05-08 Boehringer Ingelheim Int Neue trockene und wässrige Epinastin-Sirup-Formulierung
BR0313175A (pt) * 2002-08-02 2005-06-14 Boehringer Ingelheim Int Formulações farmacêuticas compreendendo combinações de epinastina, pseudoefedrina e metilefedrina
AU2003303631B2 (en) 2002-12-26 2008-05-29 Nuvo Pharmaceuticals (Ireland) Designated Activity Company Multilayer Dosage Forms Containing NSAIDs and Triptans
EP1452177A1 (en) * 2003-02-27 2004-09-01 Boehringer Ingelheim International GmbH Pharmaceutical formulations comprising sodium laurylsulfate as bitterness masking agent
EP1901724A1 (en) * 2005-07-08 2008-03-26 Senju Pharmaceutical Co., Ltd. Percutaneously absorptive ophthalmic preparation comprising epinastine
US7247623B2 (en) * 2005-08-19 2007-07-24 Inspire Pharmaceuticals, Inc. Method of treating dry eye disease with non-drying antihistamines
WO2007110380A1 (en) * 2006-03-25 2007-10-04 Boehringer Ingelheim International Gmbh Insect bite relief preparation comprising epinastine
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US20080102097A1 (en) * 2006-10-31 2008-05-01 Zanella John M Device and method for treating osteolysis using a drug depot to deliver an anti-inflammatory agent
US8470360B2 (en) 2008-04-18 2013-06-25 Warsaw Orthopedic, Inc. Drug depots having different release profiles for reducing, preventing or treating pain and inflammation
RU2464984C2 (ru) * 2007-11-22 2012-10-27 Общество с ограниченной ответственностью "МС-Вита" Нестероидное противовоспалительное лекарственное средство
US8557273B2 (en) * 2008-04-18 2013-10-15 Medtronic, Inc. Medical devices and methods including polymers having biologically active agents therein
US8956641B2 (en) * 2008-04-18 2015-02-17 Warsaw Orthopedic, Inc. Alpha adrenergic receptor agonists for treatment of inflammatory diseases
US20090263489A1 (en) * 2008-04-18 2009-10-22 Warsaw Orthopedic, Inc. Analgesic and anti-inflammatory compositions and methods for reducing, preventing or treating pain and inflammation
US8883768B2 (en) * 2008-04-18 2014-11-11 Warsaw Orthopedic, Inc. Fluocinolone implants to protect against undesirable bone and cartilage destruction
US20090263451A1 (en) * 2008-04-18 2009-10-22 Warsaw Orthopedic, Inc. Anti-Inflammatory and/or Analgesic Agents for Treatment of Myofascial Pain
US9072727B2 (en) 2008-04-18 2015-07-07 Warsaw Orthopedic, Inc. Alpha adrenergic receptor agonists for treatment of degenerative disc disease
USRE48948E1 (en) 2008-04-18 2022-03-01 Warsaw Orthopedic, Inc. Clonidine compounds in a biodegradable polymer
US8722079B2 (en) 2008-04-18 2014-05-13 Warsaw Orthopedic, Inc. Methods for treating conditions such as dystonia and post-stroke spasticity with clonidine
US8889173B2 (en) * 2008-04-18 2014-11-18 Warsaw Orthopedic, Inc. Alpha adrenergic receptor agonists for treatment of pain and/or inflammation
US20090264477A1 (en) * 2008-04-18 2009-10-22 Warsaw Orthopedic, Inc., An Indiana Corporation Beta adrenergic receptor agonists for treatment of pain and/or inflammation
US8946277B2 (en) * 2008-04-18 2015-02-03 Warsaw Orthopedic, Inc. Clonidine formulations in a biodegradable polymer carrier
US8629172B2 (en) * 2008-04-18 2014-01-14 Warsaw Orthopedic, Inc. Methods and compositions for treating post-operative pain comprising clonidine
US20090264489A1 (en) * 2008-04-18 2009-10-22 Warsaw Orthopedic, Inc. Method for Treating Acute Pain with a Formulated Drug Depot in Combination with a Liquid Formulation
US9610243B2 (en) 2008-04-18 2017-04-04 Warsaw Orthopedic, Inc. Clonidine compounds in a biodegradable polymer
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US9132119B2 (en) * 2008-04-18 2015-09-15 Medtronic, Inc. Clonidine formulation in a polyorthoester carrier
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US9988445B2 (en) 2013-09-02 2018-06-05 The University Of Melbourne Method of treatment of pain by administration of a CCL17 specific antibody
CN105708840A (zh) * 2014-12-01 2016-06-29 重庆安格龙翔医药科技有限公司 一种盐酸依匹斯汀组合物
GB2571696B (en) 2017-10-09 2020-05-27 Compass Pathways Ltd Large scale method for the preparation of Psilocybin and formulations of Psilocybin so produced
KR102041389B1 (ko) 2017-12-12 2019-11-27 (주)프론트바이오 N-(9,13b-디하이드로-1H-디벤조[c,f]이미다조[1,5-a]아제핀-3-일)-2-하이드록시벤즈아미드 및 2-((9,13b-디하이드로-1H-디벤조[c,f]이미다조[1,5-a]아제핀-3-일) 카바모일)페닐 아세테이트의 화합물, 이의 제조방법 및 이를 포함하는 항염증 및 진통제 조성물
AU2020257625A1 (en) 2019-04-17 2021-11-04 Compass Pathfinder Limited Methods for treating anxiety disorders, headache disorders, and eating disorders with psilocybin
JP6963651B2 (ja) * 2020-04-16 2021-11-10 参天製薬株式会社 エピナスチン又はその塩を含有する水性組成物
JP7118579B1 (ja) 2020-04-16 2022-08-16 参天製薬株式会社 エピナスチン又はその塩を含有する水性組成物

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Also Published As

Publication number Publication date
SK61398A3 (en) 1998-09-09
BG62511B1 (bg) 2000-01-31
EE9800158A (et) 1998-12-15
AU7623096A (en) 1997-06-05
MX9803206A (es) 1998-09-30
CN1202111A (zh) 1998-12-16
CA2232008C (en) 2004-01-06
DE19542281A1 (de) 1997-05-15
UY24354A1 (es) 2001-10-25
DE59608738D1 (de) 2002-03-21
NZ322467A (en) 2000-01-28
ATE213160T1 (de) 2002-02-15
HUP9903489A2 (hu) 2000-03-28
HUP9903489A3 (en) 2001-12-28
HU225759B1 (en) 2007-08-28
RU2217144C2 (ru) 2003-11-27
WO1997017971A1 (de) 1997-05-22
PT861081E (pt) 2002-06-28
DK0861081T3 (da) 2002-05-27
PL326653A1 (en) 1998-10-12
CZ149898A3 (cs) 1998-10-14
JP4850880B2 (ja) 2012-01-11
AR004321A1 (es) 1998-11-04
BG102408A (en) 1998-12-30
KR19990067527A (ko) 1999-08-25
JP2000500446A (ja) 2000-01-18
TW575423B (en) 2004-02-11
PL186615B1 (pl) 2004-02-27
CZ290115B6 (cs) 2002-06-12
NO982172L (no) 1998-05-13
JP2009019050A (ja) 2009-01-29
CA2232008A1 (en) 1997-05-22
ZA969520B (en) 1997-05-14
RO118373B1 (ro) 2003-05-30
IL123601A (en) 2002-12-01
BR9611502A (pt) 1999-03-02
HK1015280A1 (en) 1999-10-15
ES2171746T3 (es) 2002-09-16
RU2238733C2 (ru) 2004-10-27
EE03512B1 (et) 2001-10-15
KR100435611B1 (ko) 2005-01-13
NO982172D0 (no) 1998-05-13
EP0861081B1 (de) 2002-02-13
IL123601A0 (en) 1998-10-30
US5942503A (en) 1999-08-24
CN1104242C (zh) 2003-04-02
AU706112B2 (en) 1999-06-10
EP0861081A1 (de) 1998-09-02
TR199800853T2 (xx) 1998-09-21
JP4264850B2 (ja) 2009-05-20
DE19542281C2 (de) 1997-12-04

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