CN1592620A - 与心脏胰岛素抵抗相关的疾病的治疗和预防方法 - Google Patents
与心脏胰岛素抵抗相关的疾病的治疗和预防方法 Download PDFInfo
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- CN1592620A CN1592620A CNA008197679A CN00819767A CN1592620A CN 1592620 A CN1592620 A CN 1592620A CN A008197679 A CNA008197679 A CN A008197679A CN 00819767 A CN00819767 A CN 00819767A CN 1592620 A CN1592620 A CN 1592620A
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- analeptic
- heart failure
- insulin resistant
- chemical compound
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- 125000001188 haloalkyl group Chemical group 0.000 description 1
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- 238000005984 hydrogenation reaction Methods 0.000 description 1
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- NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical compound [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 description 1
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- XAEFZNCEHLXOMS-UHFFFAOYSA-M potassium benzoate Chemical compound [K+].[O-]C(=O)C1=CC=CC=C1 XAEFZNCEHLXOMS-UHFFFAOYSA-M 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
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- 229960004919 procaine Drugs 0.000 description 1
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- 239000004405 propyl p-hydroxybenzoate Substances 0.000 description 1
- QELSKZZBTMNZEB-UHFFFAOYSA-N propylparaben Chemical compound CCCOC(=O)C1=CC=C(O)C=C1 QELSKZZBTMNZEB-UHFFFAOYSA-N 0.000 description 1
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- 229910052708 sodium Inorganic materials 0.000 description 1
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- 235000010356 sorbitol Nutrition 0.000 description 1
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- 239000005720 sucrose Substances 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/GB2000/002347 WO2001095906A1 (en) | 2000-06-16 | 2000-06-16 | Treatment and prevention of cardiac insulin resistance associated conditions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1592620A true CN1592620A (zh) | 2005-03-09 |
Family
ID=9884792
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA008197679A Pending CN1592620A (zh) | 2000-06-16 | 2000-06-16 | 与心脏胰岛素抵抗相关的疾病的治疗和预防方法 |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP1292301A1 (hu) |
| JP (1) | JP2004503499A (hu) |
| CN (1) | CN1592620A (hu) |
| AP (1) | AP2002002688A0 (hu) |
| BG (1) | BG107384A (hu) |
| BR (1) | BR0017254A (hu) |
| CA (1) | CA2436116A1 (hu) |
| DZ (1) | DZ3389A1 (hu) |
| EA (1) | EA200300028A1 (hu) |
| HU (1) | HUP0301103A2 (hu) |
| IL (1) | IL153452A0 (hu) |
| MX (1) | MXPA02012619A (hu) |
| NO (1) | NO20026000L (hu) |
| WO (1) | WO2001095906A1 (hu) |
| YU (1) | YU1203A (hu) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7041691B1 (en) | 1999-06-30 | 2006-05-09 | Amgen Inc. | Compounds for the modulation of PPARγ activity |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9218830D0 (en) * | 1992-09-05 | 1992-10-21 | Smithkline Beecham Plc | Novel compounds |
| US5902726A (en) * | 1994-12-23 | 1999-05-11 | Glaxo Wellcome Inc. | Activators of the nuclear orphan receptor peroxisome proliferator-activated receptor gamma |
| WO1998005331A2 (en) * | 1996-08-02 | 1998-02-12 | Ligand Pharmaceuticals Incorporated | Prevention or treatment of type 2 diabetes or cardiovascular disease with ppar modulators |
| WO1999059586A1 (en) * | 1998-05-19 | 1999-11-25 | Regents Of The University Of California | Thiazolidine and oxazolidine derivatives for the treatment of acute myocardial infarction and inhibition of cardiomyocyte apoptosis |
| MA26662A1 (fr) * | 1998-07-21 | 2004-12-20 | Smithkline Beecham Plc | Derives de thiazolidinedione, compositions pharmaceutiques les contenant et leur utilisation |
-
2000
- 2000-06-16 EA EA200300028A patent/EA200300028A1/ru unknown
- 2000-06-16 YU YU1203A patent/YU1203A/sh unknown
- 2000-06-16 DZ DZ003389A patent/DZ3389A1/xx active
- 2000-06-16 MX MXPA02012619A patent/MXPA02012619A/es unknown
- 2000-06-16 JP JP2002510084A patent/JP2004503499A/ja active Pending
- 2000-06-16 IL IL15345200A patent/IL153452A0/xx unknown
- 2000-06-16 EP EP00938933A patent/EP1292301A1/en not_active Withdrawn
- 2000-06-16 CN CNA008197679A patent/CN1592620A/zh active Pending
- 2000-06-16 AP APAP/P/2002/002688A patent/AP2002002688A0/en unknown
- 2000-06-16 CA CA002436116A patent/CA2436116A1/en not_active Abandoned
- 2000-06-16 WO PCT/GB2000/002347 patent/WO2001095906A1/en not_active Application Discontinuation
- 2000-06-16 BR BR0017254-5A patent/BR0017254A/pt not_active IP Right Cessation
- 2000-06-16 HU HU0301103A patent/HUP0301103A2/hu unknown
-
2002
- 2002-12-12 BG BG107384A patent/BG107384A/bg unknown
- 2002-12-13 NO NO20026000A patent/NO20026000L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NO20026000L (no) | 2003-02-11 |
| MXPA02012619A (es) | 2003-04-10 |
| IL153452A0 (en) | 2003-07-06 |
| WO2001095906A1 (en) | 2001-12-20 |
| CA2436116A1 (en) | 2001-12-20 |
| AP2002002688A0 (en) | 2002-12-31 |
| EA200300028A1 (ru) | 2003-04-24 |
| YU1203A (sh) | 2006-05-25 |
| EP1292301A1 (en) | 2003-03-19 |
| HUP0301103A2 (hu) | 2003-08-28 |
| DZ3389A1 (fr) | 2001-12-20 |
| NO20026000D0 (no) | 2002-12-13 |
| BR0017254A (pt) | 2004-01-06 |
| JP2004503499A (ja) | 2004-02-05 |
| BG107384A (bg) | 2003-09-30 |
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| C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
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