CN1410420A - 链烷磺酰基吡啶的制备方法 - Google Patents

链烷磺酰基吡啶的制备方法 Download PDF

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Publication number
CN1410420A
CN1410420A CN02143532A CN02143532A CN1410420A CN 1410420 A CN1410420 A CN 1410420A CN 02143532 A CN02143532 A CN 02143532A CN 02143532 A CN02143532 A CN 02143532A CN 1410420 A CN1410420 A CN 1410420A
Authority
CN
China
Prior art keywords
alkyl
general formula
acid
compound
reagent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN02143532A
Other languages
English (en)
Chinese (zh)
Inventor
J·诺瓦科斯基
D·C·哈格
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of CN1410420A publication Critical patent/CN1410420A/zh
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/76—Nitrogen atoms to which a second hetero atom is attached
    • C07D213/77—Hydrazine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CN02143532A 2001-09-28 2002-09-27 链烷磺酰基吡啶的制备方法 Pending CN1410420A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32564801P 2001-09-28 2001-09-28
US60/325,648 2001-09-28

Publications (1)

Publication Number Publication Date
CN1410420A true CN1410420A (zh) 2003-04-16

Family

ID=23268791

Family Applications (1)

Application Number Title Priority Date Filing Date
CN02143532A Pending CN1410420A (zh) 2001-09-28 2002-09-27 链烷磺酰基吡啶的制备方法

Country Status (14)

Country Link
US (1) US6590103B2 (enExample)
EP (1) EP1298116A1 (enExample)
JP (1) JP2003160564A (enExample)
KR (1) KR20030027869A (enExample)
CN (1) CN1410420A (enExample)
BR (1) BR0203861A (enExample)
CA (1) CA2405328A1 (enExample)
HU (1) HUP0203242A2 (enExample)
IL (1) IL151836A0 (enExample)
MX (1) MXPA02009565A (enExample)
PL (1) PL356317A1 (enExample)
RU (1) RU2224747C1 (enExample)
YU (1) YU67702A (enExample)
ZA (1) ZA200207740B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20060058728A (ko) 2003-10-02 2006-05-30 파마시아 앤드 업존 캄파니 엘엘씨 피롤-치환된 인돌리논 화합물의 염 및 다형체

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668539A (en) * 1970-07-29 1972-06-06 Bell Telephone Labor Inc Low level amplifier
US4511857A (en) * 1982-09-17 1985-04-16 Gunderson Steven J Output following intermediate cascode circuit
FI100751B (fi) * 1996-06-11 1998-02-13 Nikolay Tchamov Pienikohinainen vahvistin
US6262273B1 (en) * 1996-09-12 2001-07-17 Basf Aktiengesellschaft Substituted thiopyridines
US6069534A (en) * 1997-12-04 2000-05-30 Trw Inc. Balance photo-receiver with complementary HBT common-base push pull pre-amplifier
ES2200787T3 (es) * 1999-12-03 2004-03-16 Pfizer Products Inc. Derivados de acetileno como agentes antiinflamatorios/analgesicos.
AP2002002532A0 (en) * 1999-12-03 2002-06-30 Pfizer Prod Inc Heterocyclo-alkylsulfonyl pyrazole derivatives as ant-inflammatory/analgesic agents.

Also Published As

Publication number Publication date
ZA200207740B (en) 2004-03-26
HU0203242D0 (enExample) 2002-11-28
EP1298116A1 (en) 2003-04-02
CA2405328A1 (en) 2003-03-28
HUP0203242A2 (hu) 2003-08-28
RU2224747C1 (ru) 2004-02-27
KR20030027869A (ko) 2003-04-07
US20030092914A1 (en) 2003-05-15
US6590103B2 (en) 2003-07-08
PL356317A1 (en) 2003-04-07
MXPA02009565A (es) 2003-03-12
JP2003160564A (ja) 2003-06-03
RU2002125831A (ru) 2004-03-27
BR0203861A (pt) 2003-09-16
YU67702A (sh) 2004-12-31
IL151836A0 (en) 2003-04-10

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