HUP0203242A2 - Eljárás alkánszulfonil-piridinek előállítására - Google Patents

Eljárás alkánszulfonil-piridinek előállítására

Info

Publication number
HUP0203242A2
HUP0203242A2 HU0203242A HUP0203242A HUP0203242A2 HU P0203242 A2 HUP0203242 A2 HU P0203242A2 HU 0203242 A HU0203242 A HU 0203242A HU P0203242 A HUP0203242 A HU P0203242A HU P0203242 A2 HUP0203242 A2 HU P0203242A2
Authority
HU
Hungary
Prior art keywords
pyridines
alkanesulfonyl
preparing
reacted
general formula
Prior art date
Application number
HU0203242A
Other languages
English (en)
Inventor
Dieter Christian Haag
Jolanta Nowakowski
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of HU0203242D0 publication Critical patent/HU0203242D0/hu
Publication of HUP0203242A2 publication Critical patent/HUP0203242A2/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/76—Nitrogen atoms to which a second hetero atom is attached
    • C07D213/77—Hydrazine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A találmány szerinti eljárással (1) általános képletű alkánszulfonil-piridineket állítanak elő, ahol R1 jelentése helyettesítetlenalkilcsoport. Az (1) általános képletű vegyületek előállítása során(a) egy (2) képletű vegyületet egy Grignard-reagenssel reagáltatnak,és (b) az (a) lépésben kapott terméket egy 1-6 szénatomosalkilszulfonilező szerrel reagáltatják. Ó
HU0203242A 2001-09-28 2002-09-27 Eljárás alkánszulfonil-piridinek előállítására HUP0203242A2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US32564801P 2001-09-28 2001-09-28

Publications (2)

Publication Number Publication Date
HU0203242D0 HU0203242D0 (hu) 2002-11-28
HUP0203242A2 true HUP0203242A2 (hu) 2003-08-28

Family

ID=23268791

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203242A HUP0203242A2 (hu) 2001-09-28 2002-09-27 Eljárás alkánszulfonil-piridinek előállítására

Country Status (14)

Country Link
US (1) US6590103B2 (hu)
EP (1) EP1298116A1 (hu)
JP (1) JP2003160564A (hu)
KR (1) KR20030027869A (hu)
CN (1) CN1410420A (hu)
BR (1) BR0203861A (hu)
CA (1) CA2405328A1 (hu)
HU (1) HUP0203242A2 (hu)
IL (1) IL151836A0 (hu)
MX (1) MXPA02009565A (hu)
PL (1) PL356317A1 (hu)
RU (1) RU2224747C1 (hu)
YU (1) YU67702A (hu)
ZA (1) ZA200207740B (hu)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA06003661A (es) 2003-10-02 2006-06-05 Pharmacia & Upjohn Co Llc Sales y polimorfos de un compuesto de indolinona sustituido con pirrol.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668539A (en) * 1970-07-29 1972-06-06 Bell Telephone Labor Inc Low level amplifier
US4511857A (en) * 1982-09-17 1985-04-16 Gunderson Steven J Output following intermediate cascode circuit
FI100751B (fi) * 1996-06-11 1998-02-13 Nikolay Tchamov Pienikohinainen vahvistin
US6069534A (en) * 1997-12-04 2000-05-30 Trw Inc. Balance photo-receiver with complementary HBT common-base push pull pre-amplifier
ES2200787T3 (es) * 1999-12-03 2004-03-16 Pfizer Products Inc. Derivados de acetileno como agentes antiinflamatorios/analgesicos.
CN1423646A (zh) * 1999-12-03 2003-06-11 辉瑞产品公司 作为抗炎/镇痛剂的杂环－烷基磺酰基吡唑衍生物

Also Published As

Publication number Publication date
US20030092914A1 (en) 2003-05-15
KR20030027869A (ko) 2003-04-07
YU67702A (sh) 2004-12-31
CA2405328A1 (en) 2003-03-28
PL356317A1 (en) 2003-04-07
CN1410420A (zh) 2003-04-16
JP2003160564A (ja) 2003-06-03
MXPA02009565A (es) 2003-03-12
ZA200207740B (en) 2004-03-26
US6590103B2 (en) 2003-07-08
RU2002125831A (ru) 2004-03-27
RU2224747C1 (ru) 2004-02-27
IL151836A0 (en) 2003-04-10
EP1298116A1 (en) 2003-04-02
BR0203861A (pt) 2003-09-16
HU0203242D0 (hu) 2002-11-28

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Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees