CN1328464A - 膦酰基甲酸衍生物在治疗感染中的应用 - Google Patents
膦酰基甲酸衍生物在治疗感染中的应用 Download PDFInfo
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- CN1328464A CN1328464A CN99813747A CN99813747A CN1328464A CN 1328464 A CN1328464 A CN 1328464A CN 99813747 A CN99813747 A CN 99813747A CN 99813747 A CN99813747 A CN 99813747A CN 1328464 A CN1328464 A CN 1328464A
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- KJAMZCVTJDTESW-UHFFFAOYSA-N tiracizine Chemical compound C1CC2=CC=CC=C2N(C(=O)CN(C)C)C2=CC(NC(=O)OCC)=CC=C21 KJAMZCVTJDTESW-UHFFFAOYSA-N 0.000 description 1
- 229960000707 tobramycin Drugs 0.000 description 1
- NLVFBUXFDBBNBW-PBSUHMDJSA-S tobramycin(5+) Chemical compound [NH3+][C@@H]1C[C@H](O)[C@@H](C[NH3+])O[C@@H]1O[C@H]1[C@H](O)[C@@H](O[C@@H]2[C@@H]([C@@H]([NH3+])[C@H](O)[C@@H](CO)O2)O)[C@H]([NH3+])C[C@@H]1[NH3+] NLVFBUXFDBBNBW-PBSUHMDJSA-S 0.000 description 1
- FUSNMLFNXJSCDI-UHFFFAOYSA-N tolnaftate Chemical compound C=1C=C2C=CC=CC2=CC=1OC(=S)N(C)C1=CC=CC(C)=C1 FUSNMLFNXJSCDI-UHFFFAOYSA-N 0.000 description 1
- 229960004880 tolnaftate Drugs 0.000 description 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 description 1
- 125000002088 tosyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1C([H])([H])[H])S(*)(=O)=O 0.000 description 1
- VSQQQLOSPVPRAZ-RRKCRQDMSA-N trifluridine Chemical compound C1[C@H](O)[C@@H](CO)O[C@H]1N1C(=O)NC(=O)C(C(F)(F)F)=C1 VSQQQLOSPVPRAZ-RRKCRQDMSA-N 0.000 description 1
- 229960003962 trifluridine Drugs 0.000 description 1
- 125000002221 trityl group Chemical group [H]C1=C([H])C([H])=C([H])C([H])=C1C([*])(C1=C(C(=C(C(=C1[H])[H])[H])[H])[H])C1=C([H])C([H])=C([H])C([H])=C1[H] 0.000 description 1
- 229960003281 tyrothricin Drugs 0.000 description 1
- 230000036269 ulceration Effects 0.000 description 1
- 229960003165 vancomycin Drugs 0.000 description 1
- MYPYJXKWCTUITO-UHFFFAOYSA-N vancomycin Natural products O1C(C(=C2)Cl)=CC=C2C(O)C(C(NC(C2=CC(O)=CC(O)=C2C=2C(O)=CC=C3C=2)C(O)=O)=O)NC(=O)C3NC(=O)C2NC(=O)C(CC(N)=O)NC(=O)C(NC(=O)C(CC(C)C)NC)C(O)C(C=C3Cl)=CC=C3OC3=CC2=CC1=C3OC1OC(CO)C(O)C(O)C1OC1CC(C)(N)C(O)C(C)O1 MYPYJXKWCTUITO-UHFFFAOYSA-N 0.000 description 1
- 230000009385 viral infection Effects 0.000 description 1
- BCEHBSKCWLPMDN-MGPLVRAMSA-N voriconazole Chemical compound C1([C@H](C)[C@](O)(CN2N=CN=C2)C=2C(=CC(F)=CC=2)F)=NC=NC=C1F BCEHBSKCWLPMDN-MGPLVRAMSA-N 0.000 description 1
- 238000009333 weeding Methods 0.000 description 1
- 125000005023 xylyl group Chemical group 0.000 description 1
- 229960000523 zalcitabine Drugs 0.000 description 1
- HBOMLICNUCNMMY-XLPZGREQSA-N zidovudine Chemical compound O=C1NC(=O)C(C)=CN1[C@@H]1O[C@H](CO)[C@@H](N=[N+]=[N-])C1 HBOMLICNUCNMMY-XLPZGREQSA-N 0.000 description 1
- 239000011787 zinc oxide Substances 0.000 description 1
- 239000002132 β-lactam antibiotic Chemical class 0.000 description 1
- 229940124586 β-lactam antibiotics Drugs 0.000 description 1
- 229940126085 β‑Lactamase Inhibitor Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/665—Phosphorus compounds having oxygen as a ring hetero atom, e.g. fosfomycin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/04—Amoebicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19854310A DE19854310A1 (de) | 1998-11-25 | 1998-11-25 | Verwendung von Phosphonoameisensäurederivaten zur therapeutischen und prophylaktischen Behandlung von Infektionen |
| DE19854310.7 | 1998-11-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1328464A true CN1328464A (zh) | 2001-12-26 |
Family
ID=7888924
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN99813747A Pending CN1328464A (zh) | 1998-11-25 | 1999-11-20 | 膦酰基甲酸衍生物在治疗感染中的应用 |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP1133302A2 (no) |
| JP (1) | JP2002530343A (no) |
| CN (1) | CN1328464A (no) |
| AP (1) | AP2001002164A0 (no) |
| AU (1) | AU1859100A (no) |
| BR (1) | BR9915605A (no) |
| CA (1) | CA2352511A1 (no) |
| CZ (1) | CZ20011819A3 (no) |
| DE (1) | DE19854310A1 (no) |
| EA (1) | EA200100585A1 (no) |
| IL (1) | IL142775A0 (no) |
| NO (1) | NO20012540L (no) |
| OA (1) | OA11718A (no) |
| PL (1) | PL348354A1 (no) |
| TR (1) | TR200101431T2 (no) |
| WO (1) | WO2000030653A2 (no) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104940211A (zh) * | 2015-06-08 | 2015-09-30 | 曹晓宏 | 白桦脂酸在制备抗真菌生物被膜药物中的应用 |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100906018B1 (ko) | 2001-07-20 | 2009-07-06 | 바이오에이전시 아게 | 감마/델타 ｔ세포 활성화를 위한 유기-인 화합물 |
| EP1603542A1 (en) * | 2003-03-14 | 2005-12-14 | Epistem Limited | Treatment and/or prevention of non-viral epithelial damage |
| US20050171063A1 (en) * | 2003-10-20 | 2005-08-04 | Pawan Malhotra | Use of phosphono derivatives as anti-malarials |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1995012604A1 (en) * | 1993-11-05 | 1995-05-11 | Aktiebolaget Astra | Novel amino acid derivatives |
| SE9604582D0 (sv) * | 1996-12-13 | 1996-12-13 | Astra Ab | Novel compounds |
| RU2116790C1 (ru) * | 1997-07-02 | 1998-08-10 | Закрытое акционерное общество "Рефарм" | Наружное противоинфекционное средство "рефарм" |
| DE19859668A1 (de) * | 1998-06-24 | 1999-12-30 | Hassan Jomaa | Verwendung von Bisphosphonaten zur Prophylaxe und zur Behandlung von infektiösen Prozessen |
-
1998
- 1998-11-25 DE DE19854310A patent/DE19854310A1/de not_active Withdrawn
-
1999
- 1999-11-20 TR TR2001/01431T patent/TR200101431T2/xx unknown
- 1999-11-20 AP APAP/P/2001/002164A patent/AP2001002164A0/en unknown
- 1999-11-20 EP EP99962147A patent/EP1133302A2/de not_active Withdrawn
- 1999-11-20 BR BR9915605-9A patent/BR9915605A/pt not_active IP Right Cessation
- 1999-11-20 WO PCT/EP1999/008964 patent/WO2000030653A2/de not_active Application Discontinuation
- 1999-11-20 JP JP2000583536A patent/JP2002530343A/ja active Pending
- 1999-11-20 EA EA200100585A patent/EA200100585A1/ru unknown
- 1999-11-20 PL PL99348354A patent/PL348354A1/xx unknown
- 1999-11-20 CZ CZ20011819A patent/CZ20011819A3/cs unknown
- 1999-11-20 AU AU18591/00A patent/AU1859100A/en not_active Abandoned
- 1999-11-20 OA OA1200100130A patent/OA11718A/en unknown
- 1999-11-20 CA CA002352511A patent/CA2352511A1/en not_active Abandoned
- 1999-11-20 CN CN99813747A patent/CN1328464A/zh active Pending
- 1999-11-20 IL IL14277599A patent/IL142775A0/xx unknown
-
2001
- 2001-05-23 NO NO20012540A patent/NO20012540L/no not_active Application Discontinuation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104940211A (zh) * | 2015-06-08 | 2015-09-30 | 曹晓宏 | 白桦脂酸在制备抗真菌生物被膜药物中的应用 |
Also Published As
| Publication number | Publication date |
|---|---|
| IL142775A0 (en) | 2002-03-10 |
| AU1859100A (en) | 2000-06-13 |
| OA11718A (en) | 2005-01-26 |
| TR200101431T2 (tr) | 2001-10-22 |
| DE19854310A1 (de) | 2000-06-29 |
| WO2000030653A2 (de) | 2000-06-02 |
| BR9915605A (pt) | 2001-08-14 |
| CA2352511A1 (en) | 2000-06-02 |
| PL348354A1 (en) | 2002-05-20 |
| CZ20011819A3 (cs) | 2001-12-12 |
| EA200100585A1 (ru) | 2002-04-25 |
| JP2002530343A (ja) | 2002-09-17 |
| WO2000030653A3 (de) | 2000-11-16 |
| NO20012540L (no) | 2001-07-24 |
| EP1133302A2 (de) | 2001-09-19 |
| NO20012540D0 (no) | 2001-05-23 |
| AP2001002164A0 (en) | 2001-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| C10 | Entry into substantive examination | ||
| PB01 | Publication | ||
| SE01 | Entry into force of request for substantive examination | ||
| C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
| WD01 | Invention patent application deemed withdrawn after publication |