CN117427079A - 含氰基取代的大环类化合物的用途 - Google Patents
含氰基取代的大环类化合物的用途 Download PDFInfo
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- CN117427079A CN117427079A CN202310893963.8A CN202310893963A CN117427079A CN 117427079 A CN117427079 A CN 117427079A CN 202310893963 A CN202310893963 A CN 202310893963A CN 117427079 A CN117427079 A CN 117427079A
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202210861773 | 2022-07-20 | ||
| CN2022108617733 | 2022-07-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN117427079A true CN117427079A (zh) | 2024-01-23 |
Family
ID=89554261
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202310893963.8A Pending CN117427079A (zh) | 2022-07-20 | 2023-07-19 | 含氰基取代的大环类化合物的用途 |
Country Status (2)
| Country | Link |
|---|---|
| CN (1) | CN117427079A (fr) |
| WO (1) | WO2024017305A1 (fr) |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017075107A1 (fr) * | 2015-10-26 | 2017-05-04 | Nanda Nisha | Mutations ponctuelles dans le cancer résistant aux inhibiteurs de trk et méthodes associées |
| WO2019144885A1 (fr) * | 2018-01-23 | 2019-08-01 | 深圳市塔吉瑞生物医药有限公司 | Composé macrocyclique de pyrazolo [1,5-a]pyrimidine substitué |
| JP7323748B2 (ja) * | 2018-02-28 | 2023-08-09 | ナンジン ザイミン ファーマシューティカル カンパニー リミテッド | ピラゾロピリミジン誘導体及びその使用 |
| CN110577549A (zh) * | 2018-06-08 | 2019-12-17 | 焦玉奇 | 大环化合物 |
| CN113773335A (zh) * | 2019-06-21 | 2021-12-10 | 成都海博为药业有限公司 | 一种作为蛋白质激酶抑制剂的化合物及其制备方法和用途 |
| US20230002410A1 (en) * | 2019-11-18 | 2023-01-05 | Guangzhou Joyo Pharmatech Co., Ltd. | Compound as highly selective ros1 inhibitor and use thereof |
-
2023
- 2023-07-19 CN CN202310893963.8A patent/CN117427079A/zh active Pending
- 2023-07-19 WO PCT/CN2023/108205 patent/WO2024017305A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2024017305A1 (fr) | 2024-01-25 |
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