CN116209659A - 方法 - Google Patents

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Publication number
CN116209659A
CN116209659A CN202180052436.3A CN202180052436A CN116209659A CN 116209659 A CN116209659 A CN 116209659A CN 202180052436 A CN202180052436 A CN 202180052436A CN 116209659 A CN116209659 A CN 116209659A
Authority
CN
China
Prior art keywords
formula
compound
reaction
alkyl
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN202180052436.3A
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English (en)
Chinese (zh)
Inventor
M·洛夫齐克
T·格拉尼尔
N·乔塞特
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Givaudan SA
Original Assignee
Givaudan SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Givaudan SA filed Critical Givaudan SA
Priority to CN202511947370.0A priority Critical patent/CN121717789A/zh
Publication of CN116209659A publication Critical patent/CN116209659A/zh
Pending legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Seasonings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Glass Compositions (AREA)
  • Iron Core Of Rotating Electric Machines (AREA)
CN202180052436.3A 2020-08-26 2021-08-24 方法 Pending CN116209659A (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN202511947370.0A CN121717789A (zh) 2020-08-26 2021-08-24 由2-哌啶酸原位形成清凉剂的方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2013383.1 2020-08-26
GBGB2013383.1A GB202013383D0 (en) 2020-08-26 2020-08-26 Process
PCT/EP2021/073378 WO2022043320A1 (en) 2020-08-26 2021-08-24 Process

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CN202511947370.0A Division CN121717789A (zh) 2020-08-26 2021-08-24 由2-哌啶酸原位形成清凉剂的方法

Publications (1)

Publication Number Publication Date
CN116209659A true CN116209659A (zh) 2023-06-02

Family

ID=72660759

Family Applications (2)

Application Number Title Priority Date Filing Date
CN202180052436.3A Pending CN116209659A (zh) 2020-08-26 2021-08-24 方法
CN202511947370.0A Pending CN121717789A (zh) 2020-08-26 2021-08-24 由2-哌啶酸原位形成清凉剂的方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN202511947370.0A Pending CN121717789A (zh) 2020-08-26 2021-08-24 由2-哌啶酸原位形成清凉剂的方法

Country Status (13)

Country Link
US (1) US20230312506A1 (https=)
EP (1) EP4204407B1 (https=)
JP (1) JP7818578B2 (https=)
KR (1) KR20230058096A (https=)
CN (2) CN116209659A (https=)
BR (1) BR112023002055A2 (https=)
CO (1) CO2023003013A2 (https=)
ES (1) ES2985349T3 (https=)
GB (1) GB202013383D0 (https=)
IL (1) IL300613A (https=)
MX (1) MX2023002234A (https=)
PL (1) PL4204407T3 (https=)
WO (1) WO2022043320A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB202105661D0 (en) * 2021-04-21 2021-06-02 Givaudan Sa Organic compounds
WO2022207944A2 (en) 2022-07-11 2022-10-06 Symrise Ag Novel mixtures and uses of (2e)-3-(1,3-benzodioxol-5-yl)-n-phenyl-n-(tetrahydro-3-furanyl)-2-propenamide

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013163270A1 (en) * 2012-04-25 2013-10-31 Theravance, Inc. Hepatitis c virus inhibitors
WO2015047973A1 (en) * 2013-09-27 2015-04-02 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
WO2015054087A1 (en) * 2013-10-07 2015-04-16 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
CN108129476A (zh) * 2017-11-27 2018-06-08 华中农业大学 一种杂环内酰胺衍生物及其用于作物病原菌杀菌剂的用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA987383B (en) * 1997-08-19 2000-02-17 Lilly Co Eli Treatment of congestive heart failure with growth hormone secretagogues.
WO2006091731A2 (en) * 2005-02-24 2006-08-31 Teva Pharmaceutical Industries Ltd. Processes for the preparation of linezolid intermediate
JP2009535327A (ja) * 2006-04-25 2009-10-01 ディシュマン・ファーマシューティカルズ・アンド・ケミカルズ・リミテッド ロピバカイン塩酸塩無水物およびその調製
TWI610916B (zh) * 2012-08-03 2018-01-11 廣東東陽光藥業有限公司 作爲丙型肝炎抑制劑的橋環化合物及其在藥物中的應用
EP4045491A1 (en) * 2019-10-17 2022-08-24 Givaudan SA Substituted azacyles as trmp8 modulators

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013163270A1 (en) * 2012-04-25 2013-10-31 Theravance, Inc. Hepatitis c virus inhibitors
WO2015047973A1 (en) * 2013-09-27 2015-04-02 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
WO2015054087A1 (en) * 2013-10-07 2015-04-16 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
CN108129476A (zh) * 2017-11-27 2018-06-08 华中农业大学 一种杂环内酰胺衍生物及其用于作物病原菌杀菌剂的用途

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CHANDRABALAN, ARUNDHASA等: "N-Cinnamoylanthranilates as human TRPA1 modulators: Structure-activity relationships and channel binding sites", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 170, 4 March 2019 (2019-03-04), pages 141 - 156 *

Also Published As

Publication number Publication date
IL300613A (en) 2023-04-01
JP2023538761A (ja) 2023-09-11
US20230312506A1 (en) 2023-10-05
WO2022043320A1 (en) 2022-03-03
ES2985349T3 (es) 2024-11-05
BR112023002055A2 (pt) 2023-03-07
KR20230058096A (ko) 2023-05-02
JP7818578B2 (ja) 2026-02-20
CO2023003013A2 (es) 2023-04-17
EP4204407B1 (en) 2024-06-19
EP4204407A1 (en) 2023-07-05
GB202013383D0 (en) 2020-10-07
PL4204407T3 (pl) 2024-11-04
CN121717789A (zh) 2026-03-24
MX2023002234A (es) 2023-03-15

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