CN114401946A - Magl抑制剂及其制备方法、用途 - Google Patents

Magl抑制剂及其制备方法、用途 Download PDF

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CN114401946A
CN114401946A CN202080061346.6A CN202080061346A CN114401946A CN 114401946 A CN114401946 A CN 114401946A CN 202080061346 A CN202080061346 A CN 202080061346A CN 114401946 A CN114401946 A CN 114401946A
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aryl
alkyl
maglz
group
radical
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张贵民
王进欣
姚景春
赵桂芳
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Lunan Pharmaceutical Group Corp
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Lunan Pharmaceutical Group Corp
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Priority claimed from CN201910836454.5A external-priority patent/CN111518020A/zh
Priority claimed from CN201910856962.XA external-priority patent/CN112552229A/zh
Priority claimed from CN201910854235.XA external-priority patent/CN112552228A/zh
Application filed by Lunan Pharmaceutical Group Corp filed Critical Lunan Pharmaceutical Group Corp
Publication of CN114401946A publication Critical patent/CN114401946A/zh
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Abstract

本发明属于药物领域，涉及一种作为MAGL抑制剂的式(Ⅰ)化合物及其药学上可接受的盐，及其制备方法、用途，和用于制备其的中间体。

Description

PCT国内申请，说明书已公开。

Claims (21)

  1. PCT国内申请，权利要求书已公开。
CN202080061346.6A 2019-09-05 2020-07-27 Magl抑制剂及其制备方法、用途 Pending CN114401946A (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
CN201910836454.5A CN111518020A (zh) 2019-02-01 2019-09-05 Magl抑制剂及其制备方法、用途
CN2019108364545 2019-09-05
CN201910856962X 2019-09-10
CN201910856962.XA CN112552229A (zh) 2019-09-10 2019-09-10 Magl抑制剂及制备方法和用途
CN201910854235X 2019-09-10
CN201910854235.XA CN112552228A (zh) 2019-09-10 2019-09-10 Magl抑制剂及其用途
PCT/CN2020/104989 WO2021042911A1 (zh) 2019-09-05 2020-07-27 Magl抑制剂及其制备方法、用途

Publications (1)

Publication Number Publication Date
CN114401946A true CN114401946A (zh) 2022-04-26

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US (1) US20230090255A1 (zh)
EP (1) EP4043436A4 (zh)
JP (1) JP2022546958A (zh)
KR (1) KR20220058553A (zh)
CN (1) CN114401946A (zh)
AU (1) AU2020343737A1 (zh)
BR (1) BR112022004068A2 (zh)
CA (1) CA3150147A1 (zh)
MX (1) MX2022002720A (zh)
WO (1) WO2021042911A1 (zh)

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