CN113116749A - 一种用于修复女性阴道松弛的组合物配方及其配制方法 - Google Patents
一种用于修复女性阴道松弛的组合物配方及其配制方法 Download PDFInfo
- Publication number
- CN113116749A CN113116749A CN202110444656.2A CN202110444656A CN113116749A CN 113116749 A CN113116749 A CN 113116749A CN 202110444656 A CN202110444656 A CN 202110444656A CN 113116749 A CN113116749 A CN 113116749A
- Authority
- CN
- China
- Prior art keywords
- parts
- fiber
- citric acid
- vaginal
- forming peptide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/194—Carboxylic acids, e.g. valproic acid having two or more carboxyl groups, e.g. succinic, maleic or phthalic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/19—Cosmetics or similar toiletry preparations characterised by the composition containing inorganic ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
- A61K8/36—Carboxylic acids; Salts or anhydrides thereof
- A61K8/365—Hydroxycarboxylic acids; Ketocarboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/73—Polysaccharides
- A61K8/731—Cellulose; Quaternized cellulose derivatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/73—Polysaccharides
- A61K8/732—Starch; Amylose; Amylopectin; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/72—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds
- A61K8/84—Cosmetics or similar toiletry preparations characterised by the composition containing organic macromolecular compounds obtained by reactions otherwise than those involving only carbon-carbon unsaturated bonds
- A61K8/86—Polyethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/005—Preparations for sensitive skin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Birds (AREA)
- Engineering & Computer Science (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Inorganic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Emergency Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
本发明公开了一种用于修复女性阴道松弛的组合物配方及其配制方法,所述修复女性阴道松弛的组合物由以下重量份的原料制备而成:酸性成纤维肽1份、碱性成纤维肽1份、羧丙甲基纤维素2份、水溶性淀粉1份、枸橼酸2份、碳酸氢钠2份、聚乙二醇6000 2份。本发明通过阴道给药,经阴道吸收,促进阴道细胞饱满,修复老化的组织、拉伤的肌肉纤维组织,增加阴道弹性,保护阴道粘膜。
Description
技术领域
本发明涉及保健品药妆技术领域,具体涉及一种用于修复女性阴道松弛的组合物配方及其配制方法。
背景技术
目前,用于女性阴道松弛和产后盆底肌修复的产品大都为物理方法,例如:阴道哑铃、低频电刺激;利用生物多肽进行治疗和改善女性阴道松弛、盆底肌松弛的产品较少。
发明内容
本发明的目的是提供一种用于修复女性阴道松弛的组合物配方及其配制方法,本发明的配制方法得到的组合物,其通过阴道给药,经阴道吸收,促进阴道细胞饱满,修复老化的组织、拉伤的肌肉纤维组织,增加阴道弹性,保护阴道粘膜。
为解决上述技术问题,本发明采用如下技术方案:
本发明提供一种用于修复女性阴道松弛的组合物,其特征在于,由以下重量份的原料制备而成:酸性成纤维肽1份、碱性成纤维肽1份、羧丙甲基纤维素2份、水溶性淀粉1份、枸橼酸2份、碳酸氢钠2份、聚乙二醇6000 2份。
本发明还涉及一种用于修复女性阴道松弛的组合物的配制方法,其特征在于,具体步骤如下:
1)按重量份取酸性成纤维肽、碱性成纤维肽、羧丙甲基纤维素、水溶性淀粉、枸橼酸、碳酸氢钠、聚乙二醇6000;
2)将羧丙甲基纤维素、枸橼酸、羧丙甲基纤维素、水溶性淀粉、枸橼酸、碳酸氢钠、聚乙二醇6000分别用纯化水溶解;
3)将步骤2溶解好的液体放入过滤机中过滤,之后加入聚六亚甲基双胍,搅拌均匀,检测后即可回灌装。
4)将步骤3得到的产物烘干—检验—压片—检验—包装—入库。
使用方法:本组合物为片状,每片0.3g或0.6g,每日一次,每次1-2片,7-10天为一疗程。
本发明的有益效果在于:通过阴道给药,经阴道吸收,促进阴道细胞饱满,修复老化的组织、拉伤的肌肉纤维组织,增加阴道弹性,保护阴道粘膜。
以下结合本发明中的主要成分的功效对本发明的有益效果作进一步说明:
酸性成纤维肽:对促进成纤维细胞的代谢和胶原蛋白的形成发挥着重要功能。能促进皮肤组织的生长繁殖,通过与细胞表面特异受体结合,调控皮肤上皮,内皮和基质细胞的分裂、繁殖和生长分化,促进细胞代谢,增强氧化作用;能促进与皮肤损伤有关细胞的迅速生长繁殖,并调节细胞间基质的合成、分泌及分解;能促进角质层细胞的再生,加速皮肤角质层和基质层的修复,促进人体皮肤细胞的生长;能增强皮肤细胞的蛋白质的合成和细胞代谢,具有延缓皮肤细胞衰老、促进表皮细胞的修复和生长作用,使皮肤光滑丰润。
碱性成纤维肽:能促进中胚层和神经外胚层细胞分裂的多肽。具有强烈的血管生成作用。在体外,能刺激细胞增殖、迁移,诱导纤溶酶原激活物及胶原酶活性,是与肝素有高亲和力的细胞促分裂原。
羧丙甲基纤维素:可形成高粘度的胶体、溶液、有粘着、增稠、流动、乳化分散、赋形、保水、保护胶体、薄膜成型、耐酸、耐盐、悬浊等特性,且生理无害,因此在食品、医药、日化、石油、造纸、纺织、建筑等领域生产中得到广泛应用。
水溶性淀粉:是一种介于淀粉和淀粉糖之间,经控制而成的低程度水解产品,该产品水化力较强,在常温下即可溶解,有良好湿度的粘性,有很好的载体作用,几乎没有甜度或不甜,耐热性强,不易褐变,有很好的乳化作用和增稠效果,吸湿性小,不易结团,成膜性好等优点。
枸橼酸:1.用于食品工业,因为柠檬酸有温和爽快的酸味;2、用于化妆品,加快角质更新;3、用于杀菌,柠檬酸与80℃温度联合作用具有良好杀灭细菌芽孢的作用,并可有效杀灭血液透析机管路中污染的细菌芽孢;4、用于医药,在凝血酶原激活物的形成及以后的凝血过程中,必须有钙离子参加。
碳酸氢钠:碳酸氢钠为弱碱,内服后能迅速中和胃酸,其抗酸作用弱而短暂,此外尚有碱化尿液的作用,适用于胃酸过多,消化不良及碱化尿液等。
聚乙二醇6000:无毒、无刺激性,味微苦,具有良好的水溶性,并与许多有机物组份有良好的相溶性。它们具有优良的润滑性、保湿性、分散性、粘接剂、抗静电剂及柔软剂等,在化妆品、制药、化纤、橡胶、塑料、造纸、油漆、电镀、农药、金属加工及食品加工等行业中均有着极为广泛的应用。
具体实施方式
下面将结合本发明实施例中对本发明的技术方案进行清楚、完整地描述,显然,所描述的实施例仅仅是本发明一部分实施例,而不是全部的实施例。基于本发明中的实施例,本领域普通技术人员在没有做出创造性劳动前提下所获得的所有其他实施例,都属于本发明保护的范围。
一种用于修复女性阴道松弛的组合物,由以下重量的原料制备而成:酸性成纤维肽500g、碱性成纤维肽500g、羧丙甲基纤维素1000g、水溶性淀粉500g、枸橼酸1000g、碳酸氢钠1000g、聚乙二醇6000 1000g。
其配制方法具体步骤如下:
1)取酸性成纤维肽500g、碱性成纤维肽500g、羧丙甲基纤维素1000g、水溶性淀粉500g、枸橼酸1000g、碳酸氢钠1000g、聚乙二醇6000 1000g;
2)将羧丙甲基纤维素、枸橼酸、羧丙甲基纤维素、水溶性淀粉、枸橼酸、碳酸氢钠、聚乙二醇6000分别用纯化水溶解;
3)将步骤2溶解好的液体放入过滤机中过滤,之后加入500ml聚六亚甲基双胍,搅拌均匀,检测后即可回灌装。
4)将步骤3得到的产物烘干—检验—压片—检验—包装—入库。
应用本发明临床试验:
试验人员100例产后阴道松弛的女性,年龄20-55岁,将100例试验人员分为4组,使4组尽量相似,使其具有可比性。
使用方法:本组合物为片状,每片0.3g,每日一次,每次2片,7-10天为一疗程,连续使用三个疗程。
诊断标准
有效:阴道松弛现象改善。
结果:100位产后阴道松弛女性,99位有效,有效率99%。
显然,本领域的技术人员可以对本发明进行各种改动和变型而不脱离本发明的精神和范围。这样,倘若本发明的这些修改和变型属于本发明权利要求及其等同技术的范围之内,则本发明也意图包含这些改动和变型在内。
Claims (2)
1.一种用于修复女性阴道松弛的组合物,其特征在于,由以下重量份的原料制备而成:酸性成纤维肽1份、碱性成纤维肽1份、羧丙甲基纤维素2份、水溶性淀粉1份、枸橼酸2份、碳酸氢钠2份、聚乙二醇6000 2份。
2.如权利要求1所述的修复女性阴道松弛的组合物的配制方法,其特征在于,具体步骤如下:
1)按重量份取酸性成纤维肽、碱性成纤维肽、羧丙甲基纤维素、水溶性淀粉、枸橼酸、碳酸氢钠、聚乙二醇6000;
2)将羧丙甲基纤维素、枸橼酸、羧丙甲基纤维素、水溶性淀粉、枸橼酸、碳酸氢钠、聚乙二醇6000分别用纯化水溶解;
3)将步骤2溶解好的液体放入过滤机中过滤,之后加入聚六亚甲基双胍,搅拌均匀,检测后即可回灌装。
4)将步骤3得到的产物烘干—检验—压片—检验—包装—入库。
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN202110444656.2A CN113116749A (zh) | 2021-04-24 | 2021-04-24 | 一种用于修复女性阴道松弛的组合物配方及其配制方法 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN202110444656.2A CN113116749A (zh) | 2021-04-24 | 2021-04-24 | 一种用于修复女性阴道松弛的组合物配方及其配制方法 |
Publications (1)
Publication Number | Publication Date |
---|---|
CN113116749A true CN113116749A (zh) | 2021-07-16 |
Family
ID=76779612
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN202110444656.2A Pending CN113116749A (zh) | 2021-04-24 | 2021-04-24 | 一种用于修复女性阴道松弛的组合物配方及其配制方法 |
Country Status (1)
Country | Link |
---|---|
CN (1) | CN113116749A (zh) |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102048708A (zh) * | 2010-12-08 | 2011-05-11 | 赵磊 | 替硝唑阴道泡腾片及其制备方法 |
CN111789937A (zh) * | 2020-07-06 | 2020-10-20 | 江苏艾特美科技有限公司 | 一种具有阴道紧缩功效的抑菌片 |
-
2021
- 2021-04-24 CN CN202110444656.2A patent/CN113116749A/zh active Pending
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102048708A (zh) * | 2010-12-08 | 2011-05-11 | 赵磊 | 替硝唑阴道泡腾片及其制备方法 |
CN111789937A (zh) * | 2020-07-06 | 2020-10-20 | 江苏艾特美科技有限公司 | 一种具有阴道紧缩功效的抑菌片 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FI94767C (fi) | Ei-terapeuttisesti käytettävät hyaluronihapon täydelliset ja osittaiset esterit | |
JP4542300B2 (ja) | ヒアルロン酸蓄積促進剤 | |
CN105107007B (zh) | 一种阳离子医用护创敷料及其制备方法 | |
JP5646446B2 (ja) | 医療用化合物あるいは医療用製品を作成するための生体適合性ポリマーの使用方法 | |
CN106344956A (zh) | 一种壳聚糖抑菌促愈合凝胶及其制备方法 | |
US20020172712A1 (en) | Antiemetic, anti-motion sustained release drug delivery system | |
CN103483625A (zh) | 可吸收降解的多用途生物相容性材料 | |
CN107184961A (zh) | 一种活性细胞修复剂及其制备方法 | |
CN108686255A (zh) | 一种预防疤痕形成的生物敷料及其制备方法 | |
CN107982277B (zh) | 一种复合抗菌气雾剂及其制备方法和应用 | |
CN108743921A (zh) | 一种预防疤痕形成的修复液及其制备方法和应用 | |
EP0285856B1 (de) | Verwendung von Dihydroergotamin und seinen Salzen zur lokalen Behandlung trophischer Störungen | |
CN104147108B (zh) | 含有褐藻寡糖的抑菌凝胶 | |
CN105013001A (zh) | 一种妇科医用生物水凝胶功能敷料及其制备方法 | |
CN109700998A (zh) | 一种复方肌肤损伤再生修复剂及其制备方法 | |
CN104307031B (zh) | 一种皮肤外用修复材料的制备方法及用途 | |
CN108744024A (zh) | 一种复配防疤痕液剂生物敷料及其制备方法 | |
CN113116749A (zh) | 一种用于修复女性阴道松弛的组合物配方及其配制方法 | |
CN100360141C (zh) | 小牛血清去蛋白凝胶和小牛血清去蛋白眼用凝胶 | |
CN111012944A (zh) | 一种基于藻酸盐和透明质酸的液体敷料及其制备方法 | |
CN107823256A (zh) | 一种低聚壳聚糖‑聚六亚甲基双胍伤口护理膜及其制备方法 | |
CN111760067A (zh) | 一种含艾考糊精的组合物及其应用 | |
CN106729954A (zh) | 一种含丝胶蛋白的医用敷料的制备方法 | |
CN106420399A (zh) | 一套激光美容术护理剂及其制备与使用方法 | |
CN112386531A (zh) | 一种皂荚低聚糖面膜及其制备方法 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PB01 | Publication | ||
PB01 | Publication | ||
SE01 | Entry into force of request for substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
RJ01 | Rejection of invention patent application after publication | ||
RJ01 | Rejection of invention patent application after publication |
Application publication date: 20210716 |