CN112384513A - Gabaa正变构调节剂化合物、其制备方法和用途 - Google Patents
Gabaa正变构调节剂化合物、其制备方法和用途 Download PDFInfo
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113840610A (zh) * | 2019-03-18 | 2021-12-24 | 纽罗塞克医疗公司 | Gabaａ受体调节剂用于治疗疼痛的用途 |
| CN114981266A (zh) * | 2019-10-22 | 2022-08-30 | 纽罗塞克医疗公司 | Gabaa正向变构调节剂化合物、其制备方法和用途 |
| CN115003301A (zh) * | 2019-10-23 | 2022-09-02 | 纽罗塞克医疗公司 | 用gabaa受体调节剂的癫痫状况的治疗 |
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| JP7449272B2 (ja) * | 2018-04-18 | 2024-03-13 | ニューロサイクル・セラピューティクス・インコーポレイテッド | Ｇａｂａａ陽性アロステリックモジュレーター化合物、その作製の方法および使用 |
| US12233070B2 (en) * | 2020-06-30 | 2025-02-25 | University Of Mississippi Medical Center | Methods for treating benzodiazepine misuse/use disorder |
| AU2023356939A1 (en) * | 2022-10-04 | 2025-04-10 | Engrail Therapeutics, Inc. | Gaba a receptor modulators and uses thereof |
| WO2025175214A1 (en) * | 2024-02-16 | 2025-08-21 | Engrail Therapeutics, Inc. | Methods of treating generalized anxiety disorder |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113840610A (zh) * | 2019-03-18 | 2021-12-24 | 纽罗塞克医疗公司 | Gabaａ受体调节剂用于治疗疼痛的用途 |
| CN114981266A (zh) * | 2019-10-22 | 2022-08-30 | 纽罗塞克医疗公司 | Gabaa正向变构调节剂化合物、其制备方法和用途 |
| CN115003301A (zh) * | 2019-10-23 | 2022-09-02 | 纽罗塞克医疗公司 | 用gabaa受体调节剂的癫痫状况的治疗 |
| CN115003301B (zh) * | 2019-10-23 | 2025-05-06 | 纽罗塞克医疗公司 | 用gabaa受体调节剂的癫痫状况的治疗 |
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| BR112020021104A2 (pt) | 2021-02-23 |
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| TW202012402A (zh) | 2020-04-01 |
| CL2020002663A1 (es) | 2021-06-11 |
| EP3781566A1 (en) | 2021-02-24 |
| US11542263B2 (en) | 2023-01-03 |
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