CN111163839B - 苯并咪唑酮衍生的bcl6抑制剂 - Google Patents

苯并咪唑酮衍生的bcl6抑制剂 Download PDF

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Publication number
CN111163839B
CN111163839B CN201880047061.XA CN201880047061A CN111163839B CN 111163839 B CN111163839 B CN 111163839B CN 201880047061 A CN201880047061 A CN 201880047061A CN 111163839 B CN111163839 B CN 111163839B
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methyl
amino
chloro
alkyl
hydroxy
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CN111163839A (zh
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B·R·贝勒妮
M·K·卡特
张桂明
O·A·戴维斯
S·霍尔德
M·G·劳埃德
罗德里格斯 A·瓦雷拉
A·瓦雷拉罗德里格斯
H·伍德沃德
P·诺森蒂
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Institute of Cancer Research Royal Cancer Hospital
Cancer Research Technology Ltd
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Institute of Cancer Research Royal Cancer Hospital
Cancer Research Technology Ltd
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Priority claimed from GBGB1806130.9A external-priority patent/GB201806130D0/en
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Priority to CN202410618580.4A priority Critical patent/CN118561812A/zh
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN201880047061.XA 2017-05-26 2018-05-25 苯并咪唑酮衍生的bcl6抑制剂 Active CN111163839B (zh)

Priority Applications (1)

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CN202410618580.4A CN118561812A (zh) 2017-05-26 2018-05-25 苯并咪唑酮衍生的bcl6抑制剂

Applications Claiming Priority (5)

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GB1708502.8 2017-05-26
GBGB1708502.8A GB201708502D0 (en) 2017-05-26 2017-05-26 Inhibitor compounds
GB1806130.9 2018-04-13
GBGB1806130.9A GB201806130D0 (en) 2018-04-13 2018-04-13 Inhibitor compounds
PCT/GB2018/051447 WO2018215801A1 (en) 2017-05-26 2018-05-25 Benzimidazolone derived inhibitors of bcl6

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CN111163839B true CN111163839B (zh) 2024-05-28

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US (2) US12110286B2 (https=)
EP (2) EP3630291B9 (https=)
JP (2) JP7202315B2 (https=)
KR (2) KR102828518B1 (https=)
CN (2) CN111163839B (https=)
AU (2) AU2018274723B2 (https=)
CA (1) CA3065005A1 (https=)
ES (1) ES2975690T3 (https=)
IL (2) IL270869B2 (https=)
MX (1) MX2023005636A (https=)
WO (1) WO2018215801A1 (https=)
ZA (1) ZA202405646B (https=)

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