CN110520110A - 包含5-氯-n4-[2-(二甲基磷酰基)苯基]-n2-{2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯基}嘧啶-2,4-二胺的药物制剂 - Google Patents
包含5-氯-n4-[2-(二甲基磷酰基)苯基]-n2-{2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯基}嘧啶-2,4-二胺的药物制剂 Download PDFInfo
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- CN110520110A CN110520110A CN201880021866.7A CN201880021866A CN110520110A CN 110520110 A CN110520110 A CN 110520110A CN 201880021866 A CN201880021866 A CN 201880021866A CN 110520110 A CN110520110 A CN 110520110A
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- brigatinib
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- phenyl
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Landscapes
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- Chemical & Material Sciences (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
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| US201762468696P | 2017-03-08 | 2017-03-08 | |
| US62/468,696 | 2017-03-08 | ||
| US201762491179P | 2017-04-27 | 2017-04-27 | |
| US62/491,179 | 2017-04-27 | ||
| US201762569954P | 2017-10-09 | 2017-10-09 | |
| US62/569,954 | 2017-10-09 | ||
| PCT/US2018/021128 WO2018165145A1 (en) | 2017-03-08 | 2018-03-06 | Pharmaceutical formulations comprising 5-chloro-n4-[2-(dimethylphosphoryl) phenyl]-n2-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl} pyrimidine-2,4-diamine |
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| TW (1) | TWI794214B (enExample) |
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CN115154473A (zh) * | 2022-08-04 | 2022-10-11 | 中国人民解放军陆军特色医学中心 | 布格替尼作为axl、c-met、st3gal4抑制剂的新应用 |
| CN115484937A (zh) * | 2020-04-14 | 2022-12-16 | 詹森生物科技公司 | 用于口服的包含氨基嘧啶衍生物或其药学上可接受的盐、水合物或溶剂化物的药物组合物 |
| CN116407512A (zh) * | 2021-12-31 | 2023-07-11 | 南京艾德凯腾生物医药有限责任公司 | 一种布格替尼冻干口崩片及其制备方法 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2019182936A1 (en) * | 2018-03-19 | 2019-09-26 | Ariad Pharmaceuticals, Inc. | Methods of treating cancer in pediatric patients |
| AU2022306151B2 (en) * | 2021-07-05 | 2024-11-14 | Qilu Pharmaceutical Co., Ltd. | Pharmaceutical composition, and preparation method therefor and application thereof |
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- 2018-03-06 CA CA3055109A patent/CA3055109A1/en active Pending
- 2018-03-06 EP EP18712759.2A patent/EP3592338A1/en not_active Withdrawn
- 2018-03-07 US US15/914,899 patent/US20180256610A1/en not_active Abandoned
- 2018-03-08 TW TW107107838A patent/TWI794214B/zh active
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2022
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- 2022-12-19 JP JP2022201704A patent/JP2023027312A/ja active Pending
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2023
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115484937A (zh) * | 2020-04-14 | 2022-12-16 | 詹森生物科技公司 | 用于口服的包含氨基嘧啶衍生物或其药学上可接受的盐、水合物或溶剂化物的药物组合物 |
| CN116407512A (zh) * | 2021-12-31 | 2023-07-11 | 南京艾德凯腾生物医药有限责任公司 | 一种布格替尼冻干口崩片及其制备方法 |
| CN115154473A (zh) * | 2022-08-04 | 2022-10-11 | 中国人民解放军陆军特色医学中心 | 布格替尼作为axl、c-met、st3gal4抑制剂的新应用 |
Also Published As
| Publication number | Publication date |
|---|---|
| TWI794214B (zh) | 2023-03-01 |
| US20210401860A1 (en) | 2021-12-30 |
| US20180256610A1 (en) | 2018-09-13 |
| JP2020510027A (ja) | 2020-04-02 |
| US20240082275A1 (en) | 2024-03-14 |
| TW201840320A (zh) | 2018-11-16 |
| EP3592338A1 (en) | 2020-01-15 |
| WO2018165145A1 (en) | 2018-09-13 |
| US20210186994A1 (en) | 2021-06-24 |
| CA3055109A1 (en) | 2018-09-13 |
| US20220249524A1 (en) | 2022-08-11 |
| JP2023027312A (ja) | 2023-03-01 |
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