CN110382481A - 作为激酶抑制剂的杂环化合物 - Google Patents
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| PCT/US2017/062643 WO2018094362A1 (en) | 2016-11-21 | 2017-11-20 | Heterocyclic compounds as kinase inhibitors |
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| CN110382481A true CN110382481A (zh) | 2019-10-25 |
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| EP (1) | EP3541806A4 (https=) |
| JP (1) | JP2020502066A (https=) |
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| AU (1) | AU2017362571A1 (https=) |
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| IL (1) | IL266789A (https=) |
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021093795A1 (zh) * | 2019-11-15 | 2021-05-20 | 武汉朗来科技发展有限公司 | 一种rock抑制剂及其制备方法和用途 |
| WO2021115495A1 (zh) * | 2019-12-12 | 2021-06-17 | 维眸生物科技（上海）有限公司 | 一种小分子含硫杂环化合物 |
| CN113121443A (zh) * | 2019-12-31 | 2021-07-16 | 财团法人工业技术研究院 | β-氨基酸衍生物、含其之激酶抑制剂与医药组合物以及其用途 |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102758256B1 (ko) * | 2019-12-31 | 2025-01-21 | 인더스트리얼 테크놀로지 리서치 인스티튜트 | β-아미노산 유도체, 키나아제 억제제 및 이를 함유하는 약학 조성물 |
| EP4192828A1 (en) * | 2020-08-04 | 2023-06-14 | Nura Bio, Inc. | Substituted pyridine derivatives as sarm1 inhibitors |
| CN116438171A (zh) | 2020-09-16 | 2023-07-14 | 努拉生物公司 | 作为sarm1抑制剂的取代的吡啶衍生物 |
| US20240285621A1 (en) * | 2020-09-23 | 2024-08-29 | Nerviano Medical Sciences S.R.L. | Pyrazolyl-pyrimidine derivatives as kinase inhibitors |
| MX2024001322A (es) | 2021-07-28 | 2024-04-30 | Nura Bio Inc | Derivados de piridina sustituida como inhibidores de sarm1. |
| CR20250520A (es) * | 2023-05-09 | 2025-12-19 | Amgen Inc | Alcoholes y éteres bicíclicos 5,6-condensados y 6,6-condensados y composiciones para su uso como moduladores de la 15-prostaglandina deshidrogenasa |
Citations (8)
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- 2017-11-20 EP EP17872851.5A patent/EP3541806A4/en not_active Withdrawn
- 2017-11-20 JP JP2019527417A patent/JP2020502066A/ja not_active Withdrawn
- 2017-11-20 WO PCT/US2017/062643 patent/WO2018094362A1/en not_active Ceased
- 2017-11-20 CN CN201780084129.7A patent/CN110382481A/zh active Pending
- 2017-11-20 CA CA3082254A patent/CA3082254A1/en not_active Abandoned
- 2017-11-20 AU AU2017362571A patent/AU2017362571A1/en not_active Abandoned
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| WO2021093795A1 (zh) * | 2019-11-15 | 2021-05-20 | 武汉朗来科技发展有限公司 | 一种rock抑制剂及其制备方法和用途 |
| WO2021115495A1 (zh) * | 2019-12-12 | 2021-06-17 | 维眸生物科技（上海）有限公司 | 一种小分子含硫杂环化合物 |
| CN112979675A (zh) * | 2019-12-12 | 2021-06-18 | 维眸生物科技（上海）有限公司 | 一种小分子含硫杂环化合物 |
| CN112979675B (zh) * | 2019-12-12 | 2023-12-19 | 维眸生物科技（上海）有限公司 | 一种小分子含硫杂环化合物 |
| CN113121443A (zh) * | 2019-12-31 | 2021-07-16 | 财团法人工业技术研究院 | β-氨基酸衍生物、含其之激酶抑制剂与医药组合物以及其用途 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP3541806A4 (en) | 2020-07-01 |
| US20190284157A1 (en) | 2019-09-19 |
| JP2020502066A (ja) | 2020-01-23 |
| CA3082254A1 (en) | 2018-05-24 |
| AU2017362571A1 (en) | 2019-07-11 |
| US10807966B2 (en) | 2020-10-20 |
| EP3541806A1 (en) | 2019-09-25 |
| WO2018094362A1 (en) | 2018-05-24 |
| IL266789A (en) | 2019-07-31 |
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